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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]-2-phenyl-5-thiophen-2-ylpyrazole-3-carboxamide —— C25H19N5O3S2
N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]-2-phenyl-5-thiophen-2-ylpyrazole-3-carboxamide
—— 1,5-dimethyl-4-[[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-2-phenylpyrazol-3-one —— C20H24N4O2
1,5-dimethyl-4-[[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-2-phenylpyrazol-3-one
—— [3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-[2-(1H-1,2,4-triazol-5-yl)phenyl]methanone —— C18H23N5O
[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-[2-(1H-1,2,4-triazol-5-yl)phenyl]methanone
—— 1-Benzyl-3-chloro-5-(4-methylsulfanylphenyl)pyrazole —— C17H15ClN2S
1-Benzyl-3-chloro-5-(4-methylsulfanylphenyl)pyrazole
—— (1S)-1-[4-cyclopentyl-5-(4-fluorophenyl)-1,3-thiazol-2-yl]-N-methylethanamine —— C17H21FN2S
(1S)-1-[4-cyclopentyl-5-(4-fluorophenyl)-1,3-thiazol-2-yl]-N-methylethanamine
—— 2-(3-fluorophenyl)-7-methoxy-1H-pyrazolo[4,3-c]quinolin-3-one —— C17H12FN3O2
2-(3-fluorophenyl)-7-methoxy-1H-pyrazolo[4,3-c]quinolin-3-one
—— N,N-dimethyl-2-[2-(3-phenyl-1H-pyrazol-5-yl)phenoxy]ethanamine —— C19H21N3O
N,N-dimethyl-2-[2-(3-phenyl-1H-pyrazol-5-yl)phenoxy]ethanamine
—— 1-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-4-(1H-imidazol-5-yl)piperidine —— C17H18FN5
1-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-4-(1H-imidazol-5-yl)piperidine
—— 3-(2,4-diphenylimidazol-1-yl)-N-methylpropanamide —— C19H19N3O
3-(2,4-diphenylimidazol-1-yl)-N-methylpropanamide
—— 1-(cyclohexylmethyl)-5-(1H-imidazol-5-ylmethyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazole —— C17H25N5O
1-(cyclohexylmethyl)-5-(1H-imidazol-5-ylmethyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazole
—— 4-[3-(oxan-4-yl)-5-[(4R)-2-oxoimidazolidin-4-yl]-1,2,4-triazol-1-yl]benzonitrile —— C17H18N6O2
4-[3-(oxan-4-yl)-5-[(4R)-2-oxoimidazolidin-4-yl]-1,2,4-triazol-1-yl]benzonitrile
—— 4-(1H-imidazol-5-yl)-1-(5-phenyl-1H-imidazol-2-yl)piperidine —— C17H19N5
4-(1H-imidazol-5-yl)-1-(5-phenyl-1H-imidazol-2-yl)piperidine
—— (Z)-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methyl-3-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C29H28N4O3
(Z)-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methyl-3-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— (3S)-3-(methylsulfanylmethyl)-N-[3-(2-methyltetrazol-5-yl)phenyl]piperidine-1-carboxamide —— C16H22N6OS
(3S)-3-(methylsulfanylmethyl)-N-[3-(2-methyltetrazol-5-yl)phenyl]piperidine-1-carboxamide
—— (E)-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methyl-2-(5-phenyltetrazol-1-yl)-3-thiophen-2-ylprop-2-enamide —— C24H22N6O3S
(E)-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methyl-2-(5-phenyltetrazol-1-yl)-3-thiophen-2-ylprop-2-enamide
—— 1,5-dimethyl-4-[[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-2-phenylpyrazol-3-one —— C20H24N4O2
1,5-dimethyl-4-[[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-2-phenylpyrazol-3-one
—— (E)-5-(3-benzyl-2-propylimidazol-4-yl)pent-4-enoic acid —— C18H22N2O2
(E)-5-(3-benzyl-2-propylimidazol-4-yl)pent-4-enoic acid
—— (3R)-1-[[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl]piperidine-3-carbonitrile —— C16H16FN3S
(3R)-1-[[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl]piperidine-3-carbonitrile
—— (Z)-N-[4-(tetrazol-1-yl)phenyl]-3-thiophen-2-ylprop-2-enamide —— C14H11N5OS
(Z)-N-[4-(tetrazol-1-yl)phenyl]-3-thiophen-2-ylprop-2-enamide
—— [3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]-[2-(1H-1,2,4-triazol-5-yl)phenyl]methanone —— C18H23N5O
[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]-[2-(1H-1,2,4-triazol-5-yl)phenyl]methanone
—— (6R)-1-(1-phenyltetrazol-5-yl)-1,4-diazepane-6-carboxylic acid —— C13H16N6O2
(6R)-1-(1-phenyltetrazol-5-yl)-1,4-diazepane-6-carboxylic acid
—— (Z)-N-[(3,4-dimethoxyphenyl)methyl]-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]-N-methylprop-2-enamide —— C29H29N3O4
(Z)-N-[(3,4-dimethoxyphenyl)methyl]-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]-N-methylprop-2-enamide
—— 5-O-tert-butyl 1-O-ethyl 6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-1,5-dicarboxylate —— C14H21N3O4
5-O-tert-butyl 1-O-ethyl 6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-1,5-dicarboxylate
—— 4-[3-(oxan-4-yl)-5-[(4S)-2-oxoimidazolidin-4-yl]-1,2,4-triazol-1-yl]benzonitrile —— C17H18N6O2
4-[3-(oxan-4-yl)-5-[(4S)-2-oxoimidazolidin-4-yl]-1,2,4-triazol-1-yl]benzonitrile
—— (3R)-3-(methylsulfanylmethyl)-N-[3-(2-methyltetrazol-5-yl)phenyl]piperidine-1-carboxamide —— C16H22N6OS
(3R)-3-(methylsulfanylmethyl)-N-[3-(2-methyltetrazol-5-yl)phenyl]piperidine-1-carboxamide
—— (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]prop-2-enamide —— C27H27N3O4
(Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]prop-2-enamide
—— 5-(2-methoxyphenyl)-4-methyl-2-phenyl-3H-1,2,4-triazol-3-one —— C16H15N3O2
5-(2-methoxyphenyl)-4-methyl-2-phenyl-3H-1,2,4-triazol-3-one
—— Methyl 4-(2-phenyl-1,3-oxazol-5-yl)benzoate —— C17H13NO3
Methyl 4-(2-phenyl-1,3-oxazol-5-yl)benzoate
—— 2-(3-Chlorophenyl)-4-methyl-5-phenyl-1,2,4-triazol-3-one —— C15H12ClN3O
2-(3-Chlorophenyl)-4-methyl-5-phenyl-1,2,4-triazol-3-one
—— 3-ethylsulfanyl-5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazole —— C15H18FN3OS
3-ethylsulfanyl-5-(4-fluorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazole
—— 2-(3-Fluorophenyl)-3-pyridin-4-ylimidazo[4,5-b]pyridine —— C17H11FN4
2-(3-Fluorophenyl)-3-pyridin-4-ylimidazo[4,5-b]pyridine
—— 5-(4-Methoxyphenyl)-4-pyridin-4-yl-1,3-thiazol-2-amine —— C15H13N3OS
5-(4-Methoxyphenyl)-4-pyridin-4-yl-1,3-thiazol-2-amine
—— (Z)-N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-[3-(3,4-dimethylphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C31H34N4O2
(Z)-N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-[3-(3,4-dimethylphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— (3S)-1-[[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl]piperidine-3-carbonitrile —— C16H16FN3S
(3S)-1-[[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl]piperidine-3-carbonitrile
—— 5-(3,5-dimethyl-2-phenylethynyl-3H-imidazol-4-yl)-3-methyl-[1,2,4]oxadiazole —— C16H14N4O
5-(3,5-dimethyl-2-phenylethynyl-3H-imidazol-4-yl)-3-methyl-[1,2,4]oxadiazole
—— 2-Phenylimidazo[1,2-a]quinolin-1-amine —— C17H13N3
2-Phenylimidazo[1,2-a]quinolin-1-amine
—— (6S)-1-(1-phenyltetrazol-5-yl)-1,4-diazepane-6-carboxylic acid —— C13H16N6O2
(6S)-1-(1-phenyltetrazol-5-yl)-1,4-diazepane-6-carboxylic acid
—— (Z)-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-[3-(3,4-dimethylphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C31H34N4O2
(Z)-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-[3-(3,4-dimethylphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— (E,2S)-1-cyclohexyl-4-[(1R,2S)-2-(1H-imidazol-5-yl)cyclopropyl]but-3-en-2-amine —— C16H25N3
(E,2S)-1-cyclohexyl-4-[(1R,2S)-2-(1H-imidazol-5-yl)cyclopropyl]but-3-en-2-amine
—— [2-(2-methyl-6-propan-2-ylanilino)-2-oxoethyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C26H29N3O3
[2-(2-methyl-6-propan-2-ylanilino)-2-oxoethyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— [2-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5-yl)-2-oxoethyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C28H27N5O5
[2-(6-amino-1-benzyl-3-methyl-2,4-dioxopyrimidin-5-yl)-2-oxoethyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— [2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate —— C23H20N4O3S
[2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate —— C24H22N4O4S
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate
—— [2-(1-ethyl-2,5-dimethylpyrrol-3-yl)-2-oxoethyl] (Z)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C23H24ClN3O3
[2-(1-ethyl-2,5-dimethylpyrrol-3-yl)-2-oxoethyl] (Z)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— [2-oxo-2-[2-(4-sulfamoylphenyl)ethylamino]ethyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C24H26N4O5S
[2-oxo-2-[2-(4-sulfamoylphenyl)ethylamino]ethyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— (5-phenyl-1,3-oxazol-2-yl)methyl (Z)-3-quinolin-2-ylprop-2-enoate —— C22H16N2O3
(5-phenyl-1,3-oxazol-2-yl)methyl (Z)-3-quinolin-2-ylprop-2-enoate
—— [2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] (Z)-3-quinolin-2-ylprop-2-enoate —— C25H22N4O3
[2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] (Z)-3-quinolin-2-ylprop-2-enoate
—— [2-[(5-methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate —— C22H18N4O3S
[2-[(5-methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate
—— (3-phenyl-1,2,4-oxadiazol-5-yl)methyl (Z)-2-cyano-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]prop-2-enoate —— C23H24N4O3
(3-phenyl-1,2,4-oxadiazol-5-yl)methyl (Z)-2-cyano-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]prop-2-enoate
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate —— C24H22N4O4S
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate