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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C31H38N4O5S
2-[(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C32H31ClN4O3S
2-[(4S)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H33FN4O3S
(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H29N5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H37N5O5S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C30H31FN4O3S
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2S)-butan-2-yl]acetamide —— C30H36N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2S)-butan-2-yl]acetamide
—— N-[2-(dimethylamino)ethyl]-2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C32H35N5O3S
N-[2-(dimethylamino)ethyl]-2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C31H36N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H34N4O5S
(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H34N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H34N4O4S
2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-[(2S)-butan-2-yl]-2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C32H34N4O3S
N-[(2S)-butan-2-yl]-2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H34N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C28H29ClN4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— (4R)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H34N4O2S
(4R)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C26H32ClN5O2S2
2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C32H34N4O4S
2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2R)-butan-2-yl]acetamide —— C30H36N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2R)-butan-2-yl]acetamide
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C28H28ClN5O2S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C32H33N5O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H38N4O4S
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C32H34N4O2S
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C32H34N4O2S
2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C27H30ClFN4O3S
2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2R)-butan-2-yl]acetamide —— C30H36N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2R)-butan-2-yl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C31H36N4O6S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[2-(dimethylamino)ethyl]-2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C33H37N5O2S
N-[2-(dimethylamino)ethyl]-2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H34N4O5S
(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C28H28ClN5O2S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C28H28ClN5O2S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C29H33ClN4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H33N5O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C25H29ClN4O3S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— (4S)-3-tert-butyl-1-(3-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C26H29ClN4O3S2
(4S)-3-tert-butyl-1-(3-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H32FN5O2S
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C25H29ClN4O3S2
2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H34N4O4S
2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H35FN4O3S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C28H28ClN5O2S2
2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H33N5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C31H36N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H37N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H28ClN5O2S
2-[(4S)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C27H31ClN4O3S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H32N4O5S
(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C30H36N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C29H35FN4O3S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H33ClN4O3S
(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C27H27ClN4O3S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide