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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-2-(2-oxo-1,3-benzoxazol-3-yl)-N-[2-(triazol-1-yl)phenyl]propanamide —— C18H15N5O3
(2S)-2-(2-oxo-1,3-benzoxazol-3-yl)-N-[2-(triazol-1-yl)phenyl]propanamide
—— N-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]-3-[[(S)-methylsulfinyl]methyl]aniline —— C18H18FN3OS
N-[[1-(4-fluorophenyl)pyrazol-3-yl]methyl]-3-[[(S)-methylsulfinyl]methyl]aniline
—— (2S)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-N-(2-hydroxy-2-methylpropyl)-N-methylpropanamide —— C15H24F3N3O2
(2S)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-N-(2-hydroxy-2-methylpropyl)-N-methylpropanamide
—— 1-[(3S)-3-[[methyl-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]amino]methyl]pyrrolidin-1-yl]ethanone —— C17H22N4O2
1-[(3S)-3-[[methyl-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]amino]methyl]pyrrolidin-1-yl]ethanone
—— methyl (1S,2R)-2-[[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]carbamoyl]cyclopentane-1-carboxylate —— C17H24N2O3S
methyl (1S,2R)-2-[[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]carbamoyl]cyclopentane-1-carboxylate
—— 1-cyclopentyl-N-[(1S)-2-hydroxy-1-phenylethyl]-5-methylpyrazole-4-carboxamide —— C18H23N3O2
1-cyclopentyl-N-[(1S)-2-hydroxy-1-phenylethyl]-5-methylpyrazole-4-carboxamide
—— N-[(E)-[5-chloro-1-(3-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-(4-methylanilino)acetamide —— C20H19Cl2N5O
N-[(E)-[5-chloro-1-(3-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-(4-methylanilino)acetamide
—— (2R)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-1-(1,4-thiazepan-4-yl)propan-1-one —— C15H22F3N3OS
(2R)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-1-(1,4-thiazepan-4-yl)propan-1-one
—— N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-5-(trifluoromethyl)pyridin-2-amine —— C17H13ClF3N5
N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-5-(trifluoromethyl)pyridin-2-amine
—— methyl (1R,2S)-2-[[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]carbamoyl]cyclopentane-1-carboxylate —— C17H24N2O3S
methyl (1R,2S)-2-[[1-(4-methyl-1,3-thiazol-2-yl)cyclopentyl]carbamoyl]cyclopentane-1-carboxylate
—— (2R)-2-(2-oxo-1,3-benzoxazol-3-yl)-N-[2-(triazol-1-yl)phenyl]propanamide —— C18H15N5O3
(2R)-2-(2-oxo-1,3-benzoxazol-3-yl)-N-[2-(triazol-1-yl)phenyl]propanamide
—— 3-(4-methylphenyl)-N-[(2S)-4-methylsulfonylbutan-2-yl]-1,2,4-oxadiazol-5-amine —— C14H19N3O3S
3-(4-methylphenyl)-N-[(2S)-4-methylsulfonylbutan-2-yl]-1,2,4-oxadiazol-5-amine
—— N-[(1R)-2-hydroxy-1-phenylethyl]-2-[(2R)-oxolan-2-yl]-1,3-thiazole-5-carboxamide —— C16H18N2O3S
N-[(1R)-2-hydroxy-1-phenylethyl]-2-[(2R)-oxolan-2-yl]-1,3-thiazole-5-carboxamide
—— (2S)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-1-(1,4-thiazepan-4-yl)propan-1-one —— C15H22F3N3OS
(2S)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-1-(1,4-thiazepan-4-yl)propan-1-one
—— (2R)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-N-(2-hydroxy-2-methylpropyl)-N-methylpropanamide —— C15H24F3N3O2
(2R)-2-[3,5-dimethyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-N-(2-hydroxy-2-methylpropyl)-N-methylpropanamide
—— N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-5-(trifluoromethyl)pyridin-2-amine —— C18H16F3N5
N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-5-(trifluoromethyl)pyridin-2-amine
—— N-[(2S)-1-hydroxybutan-2-yl]-2-methyl-4-(2-methylpropyl)-1,3-thiazole-5-carboxamide —— C13H22N2O2S
N-[(2S)-1-hydroxybutan-2-yl]-2-methyl-4-(2-methylpropyl)-1,3-thiazole-5-carboxamide
—— methyl (1R,2R)-2-[(2-imidazol-1-ylphenyl)carbamoyl]cyclopentane-1-carboxylate —— C17H19N3O3
methyl (1R,2R)-2-[(2-imidazol-1-ylphenyl)carbamoyl]cyclopentane-1-carboxylate
—— N-[(1S)-2-hydroxy-1-phenylethyl]-2-[(2R)-oxolan-2-yl]-1,3-thiazole-4-carboxamide —— C16H18N2O3S
N-[(1S)-2-hydroxy-1-phenylethyl]-2-[(2R)-oxolan-2-yl]-1,3-thiazole-4-carboxamide
—— 3-(4-methylphenyl)-N-[(2R)-4-methylsulfonylbutan-2-yl]-1,2,4-oxadiazol-5-amine —— C14H19N3O3S
3-(4-methylphenyl)-N-[(2R)-4-methylsulfonylbutan-2-yl]-1,2,4-oxadiazol-5-amine
—— N-[(1S)-2-hydroxy-1-phenylethyl]-2-[(2S)-oxolan-2-yl]-1,3-thiazole-4-carboxamide —— C16H18N2O3S
N-[(1S)-2-hydroxy-1-phenylethyl]-2-[(2S)-oxolan-2-yl]-1,3-thiazole-4-carboxamide
—— N-[(1R)-2-hydroxy-1-phenylethyl]-2-[(2S)-oxolan-2-yl]-1,3-thiazole-5-carboxamide —— C16H18N2O3S
N-[(1R)-2-hydroxy-1-phenylethyl]-2-[(2S)-oxolan-2-yl]-1,3-thiazole-5-carboxamide
—— methyl (1R,2S)-2-[(2-imidazol-1-ylphenyl)carbamoyl]cyclopentane-1-carboxylate —— C17H19N3O3
methyl (1R,2S)-2-[(2-imidazol-1-ylphenyl)carbamoyl]cyclopentane-1-carboxylate
—— N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]-1H-benzimidazol-2-amine —— C16H14N8
N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]-1H-benzimidazol-2-amine
—— 2,4-dimethyl-N-[(2R,4S)-2-pentan-3-yloxan-4-yl]-1,3-thiazole-5-carboxamide —— C16H26N2O2S
2,4-dimethyl-N-[(2R,4S)-2-pentan-3-yloxan-4-yl]-1,3-thiazole-5-carboxamide
—— 4-[(5-phenyltetrazol-2-yl)methyl]-N-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylideneamino]benzamide —— C22H22N8O
4-[(5-phenyltetrazol-2-yl)methyl]-N-[(E)-(1,3,5-trimethylpyrazol-4-yl)methylideneamino]benzamide
—— 2,4-dimethyl-N-[(2S,4R)-2-pentan-3-yloxan-4-yl]-1,3-thiazole-5-carboxamide —— C16H26N2O2S
2,4-dimethyl-N-[(2S,4R)-2-pentan-3-yloxan-4-yl]-1,3-thiazole-5-carboxamide
—— ethyl 3-[[(2S)-2-thiophen-2-ylpropanoyl]amino]-1H-pyrazole-5-carboxylate —— C13H15N3O3S
ethyl 3-[[(2S)-2-thiophen-2-ylpropanoyl]amino]-1H-pyrazole-5-carboxylate
—— 5-(2-fluorophenyl)-N-[(1R)-1-(1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C14H12FN5O2
5-(2-fluorophenyl)-N-[(1R)-1-(1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 2-[(R)-[(1S)-1-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)ethyl]sulfinyl]ethanol —— C10H12N2O3S2
2-[(R)-[(1S)-1-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)ethyl]sulfinyl]ethanol
—— N-[(1S)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide —— C14H14ClFN2O2S
N-[(1S)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
—— 5-(2-fluorophenyl)-N-[(1S)-1-(1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C14H12FN5O2
5-(2-fluorophenyl)-N-[(1S)-1-(1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 4-[1-methyl-4-[[[(1R)-1-[(2R)-4-methylmorpholin-2-yl]ethyl]amino]methyl]pyrazol-3-yl]benzonitrile —— C19H25N5O
4-[1-methyl-4-[[[(1R)-1-[(2R)-4-methylmorpholin-2-yl]ethyl]amino]methyl]pyrazol-3-yl]benzonitrile
—— 4-[1-methyl-4-[[[(1R)-1-[(2S)-4-methylmorpholin-2-yl]ethyl]amino]methyl]pyrazol-3-yl]benzonitrile —— C19H25N5O
4-[1-methyl-4-[[[(1R)-1-[(2S)-4-methylmorpholin-2-yl]ethyl]amino]methyl]pyrazol-3-yl]benzonitrile
—— N-[(1R)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide —— C14H14ClFN2O2S
N-[(1R)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
—— 2,4-dimethyl-N-[(2R,4R)-2-pentan-3-yloxan-4-yl]-1,3-thiazole-5-carboxamide —— C16H26N2O2S
2,4-dimethyl-N-[(2R,4R)-2-pentan-3-yloxan-4-yl]-1,3-thiazole-5-carboxamide
—— ethyl 3-[[(2R)-2-thiophen-2-ylpropanoyl]amino]-1H-pyrazole-5-carboxylate —— C13H15N3O3S
ethyl 3-[[(2R)-2-thiophen-2-ylpropanoyl]amino]-1H-pyrazole-5-carboxylate
—— 4-[1-methyl-4-[[[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]amino]methyl]pyrazol-3-yl]benzonitrile —— C20H22N6
4-[1-methyl-4-[[[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]amino]methyl]pyrazol-3-yl]benzonitrile
—— 2-ethyl-5-[[(3S)-3-(3-phenyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl]-1,3,4-oxadiazole —— C18H22N6O
2-ethyl-5-[[(3S)-3-(3-phenyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl]-1,3,4-oxadiazole
—— 4-[1-methyl-4-[[[(1S)-1-[(2S)-4-methylmorpholin-2-yl]ethyl]amino]methyl]pyrazol-3-yl]benzonitrile —— C19H25N5O
4-[1-methyl-4-[[[(1S)-1-[(2S)-4-methylmorpholin-2-yl]ethyl]amino]methyl]pyrazol-3-yl]benzonitrile
—— N-[(E)-(4-chlorophenyl)methylideneamino]-4-[(5-phenyltetrazol-2-yl)methyl]benzamide —— C22H17ClN6O
N-[(E)-(4-chlorophenyl)methylideneamino]-4-[(5-phenyltetrazol-2-yl)methyl]benzamide
—— 4-[(5-phenyltetrazol-2-yl)methyl]-N-[(Z)-[(5S)-3,3,5-trimethylcyclohexylidene]amino]benzamide —— C24H28N6O
4-[(5-phenyltetrazol-2-yl)methyl]-N-[(Z)-[(5S)-3,3,5-trimethylcyclohexylidene]amino]benzamide
—— (2S,4R,5S)-1,2,5-trimethyl-N-[3-(4-methyl-1,3-oxazol-2-yl)phenyl]piperidin-4-amine —— C18H25N3O
(2S,4R,5S)-1,2,5-trimethyl-N-[3-(4-methyl-1,3-oxazol-2-yl)phenyl]piperidin-4-amine
—— 4-(8-methylimidazo[1,2-a]pyridin-2-yl)-N-[(2S)-1-methylsulfonylpropan-2-yl]aniline —— C18H21N3O2S
4-(8-methylimidazo[1,2-a]pyridin-2-yl)-N-[(2S)-1-methylsulfonylpropan-2-yl]aniline
—— 4-[1-methyl-4-[[[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]amino]methyl]pyrazol-3-yl]benzonitrile —— C20H22N6
4-[1-methyl-4-[[[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]amino]methyl]pyrazol-3-yl]benzonitrile
—— (2R,4R,5S)-1,2,5-trimethyl-N-[3-(4-methyl-1,3-oxazol-2-yl)phenyl]piperidin-4-amine —— C18H25N3O
(2R,4R,5S)-1,2,5-trimethyl-N-[3-(4-methyl-1,3-oxazol-2-yl)phenyl]piperidin-4-amine
—— 4-[4-[[[(2S)-2-hydroxy-3,3-dimethylbutyl]amino]methyl]-1-methylpyrazol-3-yl]benzonitrile —— C18H24N4O
4-[4-[[[(2S)-2-hydroxy-3,3-dimethylbutyl]amino]methyl]-1-methylpyrazol-3-yl]benzonitrile
—— 4-[4-[[[(2R)-2-hydroxy-3,3-dimethylbutyl]amino]methyl]-1-methylpyrazol-3-yl]benzonitrile —— C18H24N4O
4-[4-[[[(2R)-2-hydroxy-3,3-dimethylbutyl]amino]methyl]-1-methylpyrazol-3-yl]benzonitrile
—— (2S,4S,5S)-1,2,5-trimethyl-N-[3-(4-methyl-1,3-oxazol-2-yl)phenyl]piperidin-4-amine —— C18H25N3O
(2S,4S,5S)-1,2,5-trimethyl-N-[3-(4-methyl-1,3-oxazol-2-yl)phenyl]piperidin-4-amine
—— 2-[(S)-[(1R)-1-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)ethyl]sulfinyl]ethanol —— C10H12N2O3S2
2-[(S)-[(1R)-1-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)ethyl]sulfinyl]ethanol