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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-piperidin-1-ylethanone —— C22H30FN5O2
2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-piperidin-1-ylethanone
—— 3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(2R)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]propan-1-one —— C15H23N3O
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(2R)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]propan-1-one
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(2-methylpropyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H27FN4O
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(2-methylpropyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— [(2S)-1-[(5-methoxy-2-pyrazol-1-ylphenyl)methyl]azepan-2-yl]methanol —— C18H25N3O2
[(2S)-1-[(5-methoxy-2-pyrazol-1-ylphenyl)methyl]azepan-2-yl]methanol
—— 2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C23H32FN5O2
2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— N-[(2R)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide —— C16H23N3OS2
N-[(2R)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
—— 2-(2,4-dimethyl-1,3-thiazol-5-yl)-N-[(2S)-2-(furan-2-ylmethyl)-3-hydroxypropyl]acetamide —— C15H20N2O3S
2-(2,4-dimethyl-1,3-thiazol-5-yl)-N-[(2S)-2-(furan-2-ylmethyl)-3-hydroxypropyl]acetamide
—— N-[(2S)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide —— C16H23N3OS2
N-[(2S)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
—— 5-[(2S)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole —— C18H19ClN4O
5-[(2S)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole
—— 5-[[(3R)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid —— C11H17N3O4
5-[[(3R)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-(4-phenylmethoxypiperidin-1-yl)ethyl]-1,2,4-oxadiazole —— C23H26FN3O2
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-(4-phenylmethoxypiperidin-1-yl)ethyl]-1,2,4-oxadiazole
—— 1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-morpholin-4-ylethanone —— C21H28FN5O3
1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-morpholin-4-ylethanone
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-2-ethylhexyl]urea —— C17H32N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-2-ethylhexyl]urea
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(3-methoxyphenyl)methanone —— C23H25FN4O3
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(3-methoxyphenyl)methanone
—— [1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-pyrrolidin-1-ylmethanone —— C21H27FN4O2
[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-pyrrolidin-1-ylmethanone
—— 2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-piperidin-1-ylethanone —— C22H30FN5O2
2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-piperidin-1-ylethanone
—— [(2R)-1-[(5-methoxy-2-pyrazol-1-ylphenyl)methyl]azepan-2-yl]methanol —— C18H25N3O2
[(2R)-1-[(5-methoxy-2-pyrazol-1-ylphenyl)methyl]azepan-2-yl]methanol
—— 5-cyclopropyl-3-[4-[5-[(3R)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole —— C17H17N5O2
5-cyclopropyl-3-[4-[5-[(3R)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole
—— 4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N,N-dimethylpiperazine-1-carboxamide —— C18H24FN5O2
4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N,N-dimethylpiperazine-1-carboxamide
—— 5-[[(3S)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid —— C11H17N3O4
5-[[(3S)-3-methoxypiperidin-1-yl]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid
—— 5-cyclopropyl-3-[4-[5-[(3S)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole —— C17H17N5O2
5-cyclopropyl-3-[4-[5-[(3S)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]-1,2,4-oxadiazole
—— 2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C23H32FN5O2
2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 5-[(1R)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C21H23FN4O3S
5-[(1R)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(2R)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole —— C18H19ClN4O
5-[(2R)-1-[[1-(2-chlorophenyl)pyrazol-4-yl]methyl]pyrrolidin-2-yl]-3-methyl-1,2-oxazole
—— 5-[(1S)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H20FN3O
5-[(1S)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-2-ethylhexyl]urea —— C17H32N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-2-ethylhexyl]urea
—— (3-chlorophenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H22ClFN4O2
(3-chlorophenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-5-methylhexan-2-yl]urea —— C16H30N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-5-methylhexan-2-yl]urea
—— 1-[(2S)-2-ethylhexyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C15H27N3OS
1-[(2S)-2-ethylhexyl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 5-[(1S)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H24FN5O4S
5-[(1S)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-morpholin-4-ylethanone —— C21H28FN5O3
2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-morpholin-4-ylethanone
—— 2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-pyrrolidin-1-ylethanone —— C21H28FN5O2
2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-pyrrolidin-1-ylethanone
—— (4-chlorophenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H22ClFN4O2
(4-chlorophenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-pyrrolidin-1-ylethanone —— C21H28FN5O2
2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-pyrrolidin-1-ylethanone
—— 2-(2,4-dimethyl-1,3-thiazol-5-yl)-N-[(2R)-2-(furan-2-ylmethyl)-3-hydroxypropyl]acetamide —— C15H20N2O3S
2-(2,4-dimethyl-1,3-thiazol-5-yl)-N-[(2R)-2-(furan-2-ylmethyl)-3-hydroxypropyl]acetamide
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-octan-2-yl]urea —— C17H32N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-octan-2-yl]urea
—— 2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone —— C23H32FN5O2
2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(2-methylpropyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H27FN4O
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(2-methylpropyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-thiophen-2-ylmethanone —— C20H21FN4O2S
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-thiophen-2-ylmethanone
—— N-[[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-3-[(2R)-oxolan-2-yl]propan-1-amine —— C19H27N3O2
N-[[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-3-[(2R)-oxolan-2-yl]propan-1-amine
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-thiophen-2-ylmethanone —— C20H21FN4O2S
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-thiophen-2-ylmethanone
—— 5-[(1S)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C21H23FN4O3S
5-[(1S)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiophene-2-carboxamide —— C14H12N6OS
N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiophene-2-carboxamide
—— 1,3-benzodioxol-5-yl-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C23H23FN4O4
1,3-benzodioxol-5-yl-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one —— C23H21N5O5
5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-1-(2-nitrophenyl)pyrazolo[3,4-d]pyrimidin-4-one
—— [1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-pyrrolidin-1-ylmethanone —— C21H27FN4O2
[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-pyrrolidin-1-ylmethanone
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-6-methylheptan-2-yl]urea —— C17H32N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-6-methylheptan-2-yl]urea
—— 3-(4-methylphenyl)-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-5-carboxamide —— C16H18N6O
3-(4-methylphenyl)-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
—— 5-[(1R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H20FN3O
5-[(1R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H24FN5O4S
5-[(1R)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole