中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C30H38FN5O4S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C31H40N4O6S |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4S)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C30H32N4O2S2 |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C29H35FN4O4S |
|
—— |
(4R)-3-tert-butyl-1,4-bis(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C28H30F2N4O3S |
|
—— |
(4R)-4-(3,4-dimethoxyphenyl)-1-(3-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C35H38N4O4S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H35ClN4O3S |
|
—— |
(4S)-3-tert-butyl-4-(2-fluorophenyl)-1-(2-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H37FN4O2S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H35ClN4O3S |
|
—— |
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C32H33FN4O5S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1,4-bis(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H29F2N5O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C30H37ClN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C34H37FN4O5S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H33FN4O4S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C29H35ClN4O4S |
|
—— |
(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H39ClN4O2S |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H35ClN4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C34H37FN4O5S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C31H40N4O5S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H29ClFN5O2S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C31H40N4O5S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C31H29ClF2N4O2S |
|
—— |
2-[(4S)-3-tert-butyl-1,4-bis(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C29H28F2N4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C29H32F2N4O3S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C28H34N4O3S2 |
|
—— |
(4S)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O6S |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H34FN5O5S |
|
—— |
(4S)-4-(4-fluorophenyl)-1-(3-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H33FN4O2S |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H33FN4O4S |
|
—— |
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C33H36N4O5S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C28H30N4O3S2 |
|
—— |
2-[(4S)-1-(2,3-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C32H33FN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C29H35ClN4O4S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C30H38FN5O4S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(3-methylphenyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H35N5O3S2 |
|
—— |
2-[(4R)-4-(2,4-difluorophenyl)-7-oxo-1,3-diphenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C30H28F2N4O3S |
|
—— |
2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C31H31ClN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C28H33ClFN5O2S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C29H35FN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C33H37N5O5S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C30H38N4O5S |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4R)-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H33ClN4O4S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C31H40N4O5S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C30H30F2N4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H35ClN4O3S |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C32H33FN4O5S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C30H28Cl2N4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H29ClFN5O2S |
|
—— |
(4S)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-(3-methylthiophen-2-yl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H34N4O2S2 |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C30H28Cl2N4O2S |
|