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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S,7aR)-N-[2-(3,5-dimethylpyrazol-1-yl)-5-(trifluoromethyl)phenyl]-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide —— C20H21F3N4O2S
(3S,7aR)-N-[2-(3,5-dimethylpyrazol-1-yl)-5-(trifluoromethyl)phenyl]-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide
—— 1-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone —— C24H26N2O3S
1-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone
—— 1-[4-[(S)-hydroxy(phenyl)methyl]piperidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone —— C24H26N2O3S
1-[4-[(S)-hydroxy(phenyl)methyl]piperidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone
—— N-[(2S)-1-hydroxypropan-2-yl]-2-pyrazol-1-ylbenzamide —— C13H15N3O2
N-[(2S)-1-hydroxypropan-2-yl]-2-pyrazol-1-ylbenzamide
—— 1-(4-chlorophenyl)-N-[(2S)-2-hydroxypropyl]pyrazole-4-carboxamide —— C13H14ClN3O2
1-(4-chlorophenyl)-N-[(2S)-2-hydroxypropyl]pyrazole-4-carboxamide
—— N-[(2R)-2-hydroxypropyl]-4-(4-methylpyrazol-1-yl)benzamide —— C14H17N3O2
N-[(2R)-2-hydroxypropyl]-4-(4-methylpyrazol-1-yl)benzamide
—— N-[(2S)-2-hydroxypropyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C15H18N2O3S
N-[(2S)-2-hydroxypropyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— 3-(2-cyclohexylethyl)-4-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C22H28N6S
3-(2-cyclohexylethyl)-4-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— N-[(2R)-2-hydroxypropyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C15H18N2O3S
N-[(2R)-2-hydroxypropyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— 1-(4-bromophenyl)-N-[(2R)-2-hydroxypropyl]pyrazole-4-carboxamide —— C13H14BrN3O2
1-(4-bromophenyl)-N-[(2R)-2-hydroxypropyl]pyrazole-4-carboxamide
—— N-[(2S)-2-hydroxypropyl]-2-pyrazol-1-ylbenzamide —— C13H15N3O2
N-[(2S)-2-hydroxypropyl]-2-pyrazol-1-ylbenzamide
—— N-[(2R)-2-hydroxypropyl]-2-pyrazol-1-ylbenzamide —— C13H15N3O2
N-[(2R)-2-hydroxypropyl]-2-pyrazol-1-ylbenzamide
—— N-[(2R,6S)-2,6-dimethylcyclohexyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C20H26N2O2S
N-[(2R,6S)-2,6-dimethylcyclohexyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-4-(4-methylpyrazol-1-yl)benzamide —— C20H28N4O3S
N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-4-(4-methylpyrazol-1-yl)benzamide
—— N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-2-pyrazol-1-ylbenzamide —— C19H26N4O2
N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-2-pyrazol-1-ylbenzamide
—— 2-[[(2R)-2-(2-bromo-4-methylphenoxy)propanoyl]amino]-1,3-thiazole-5-carboxamide —— C14H14BrN3O3S
2-[[(2R)-2-(2-bromo-4-methylphenoxy)propanoyl]amino]-1,3-thiazole-5-carboxamide
—— 2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]-N-[(1R)-1-phenyl-2-pyrrolidin-1-ylethyl]acetamide —— C24H27N3O2S
2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]-N-[(1R)-1-phenyl-2-pyrrolidin-1-ylethyl]acetamide
—— methyl N-[(E)-(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]carbamate —— C17H21N5O2
methyl N-[(E)-(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]carbamate
—— 1-(4-bromophenyl)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]pyrazole-4-carboxamide —— C20H21BrN4O
1-(4-bromophenyl)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]pyrazole-4-carboxamide
—— 4-(4-methylpyrazol-1-yl)-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)benzamide —— C21H23N3O2S
4-(4-methylpyrazol-1-yl)-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)benzamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-[(4-methoxyphenyl)methyl]-4-(4-methylpyrazol-1-yl)benzamide —— C23H25N3O4S
N-[(3S)-1,1-dioxothiolan-3-yl]-N-[(4-methoxyphenyl)methyl]-4-(4-methylpyrazol-1-yl)benzamide
—— N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-2-pyrazol-1-ylbenzamide —— C19H26N4O2
N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-2-pyrazol-1-ylbenzamide
—— 2-(1,1-dioxo-1,2-thiazolidin-2-yl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C15H19N5O3S
2-(1,1-dioxo-1,2-thiazolidin-2-yl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 2-[[(2R)-2-benzylsulfanylpropanoyl]amino]-1,3-thiazole-5-carboxamide —— C14H15N3O2S2
2-[[(2R)-2-benzylsulfanylpropanoyl]amino]-1,3-thiazole-5-carboxamide
—— N-[(R)-(3-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C24H24N4O3S
N-[(R)-(3-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— N-[3-(dimethylamino)propyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-4-(4-methylpyrazol-1-yl)benzamide —— C20H28N4O3S
N-[3-(dimethylamino)propyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-4-(4-methylpyrazol-1-yl)benzamide
—— N-[(2R,6R)-2,6-dimethylcyclohexyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C20H26N2O2S
N-[(2R,6R)-2,6-dimethylcyclohexyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— 3-nitro-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]aniline —— C15H13N7O2
3-nitro-N-[(E)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]aniline
—— 1-[(2S)-2-benzylpyrrolidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone —— C23H24N2O2S
1-[(2S)-2-benzylpyrrolidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone
—— 2-(1,1-dioxo-1,2-thiazolidin-2-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide —— C15H19N5O3S
2-(1,1-dioxo-1,2-thiazolidin-2-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]acetamide
—— 2-[[(2S)-2-benzylsulfanylpropanoyl]amino]-1,3-thiazole-5-carboxamide —— C14H15N3O2S2
2-[[(2S)-2-benzylsulfanylpropanoyl]amino]-1,3-thiazole-5-carboxamide
—— Ethyl 2-[[cyclohexyl(hexanoyl)amino]methyl]-1,3-thiazole-4-carboxylate —— C19H30N2O3S
Ethyl 2-[[cyclohexyl(hexanoyl)amino]methyl]-1,3-thiazole-4-carboxylate
—— 1-(4-bromophenyl)-N-[(1R)-2-(dimethylamino)-1-phenylethyl]pyrazole-4-carboxamide —— C20H21BrN4O
1-(4-bromophenyl)-N-[(1R)-2-(dimethylamino)-1-phenylethyl]pyrazole-4-carboxamide
—— 1-(4-chlorophenyl)-N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]pyrazole-4-carboxamide —— C19H25ClN4O3S
1-(4-chlorophenyl)-N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]pyrazole-4-carboxamide
—— N-[(2S,6S)-2,6-dimethylcyclohexyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C20H26N2O2S
N-[(2S,6S)-2,6-dimethylcyclohexyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— 2-[[(2S)-2-(2-bromo-4-methylphenoxy)propanoyl]amino]-1,3-thiazole-5-carboxamide —— C14H14BrN3O3S
2-[[(2S)-2-(2-bromo-4-methylphenoxy)propanoyl]amino]-1,3-thiazole-5-carboxamide
—— N-[(S)-(3-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C24H24N4O3S
N-[(S)-(3-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— 1-(4-chlorophenyl)-N-[3-(dimethylamino)propyl]-N-[(3S)-1,1-dioxothiolan-3-yl]pyrazole-4-carboxamide —— C19H25ClN4O3S
1-(4-chlorophenyl)-N-[3-(dimethylamino)propyl]-N-[(3S)-1,1-dioxothiolan-3-yl]pyrazole-4-carboxamide
—— 2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]acetamide —— C24H27N3O2S
2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]acetamide
—— 1-[(2R)-2-benzylpyrrolidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone —— C23H24N2O2S
1-[(2R)-2-benzylpyrrolidin-1-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]ethanone
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-[(4-methoxyphenyl)methyl]-4-(4-methylpyrazol-1-yl)benzamide —— C23H25N3O4S
N-[(3R)-1,1-dioxothiolan-3-yl]-N-[(4-methoxyphenyl)methyl]-4-(4-methylpyrazol-1-yl)benzamide
—— 4-(4-methylpyrazol-1-yl)-N-[[(2S)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)benzamide —— C21H23N3O2S
4-(4-methylpyrazol-1-yl)-N-[[(2S)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)benzamide
—— tert-butyl N-[(E)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]carbamate —— C16H18Cl2N4O2
tert-butyl N-[(E)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]carbamate
—— 3-[(2R)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]-5-methyl-1H-1,2,4-triazole —— C19H23FN6
3-[(2R)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]-5-methyl-1H-1,2,4-triazole
—— tert-butyl N-[(E)-(2-morpholin-4-yl-4-phenyl-1,3-thiazol-5-yl)methylideneamino]carbamate —— C19H24N4O3S
tert-butyl N-[(E)-(2-morpholin-4-yl-4-phenyl-1,3-thiazol-5-yl)methylideneamino]carbamate
—— 3-[(2S)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]-5-methyl-1H-1,2,4-triazole —— C19H23FN6
3-[(2S)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]-5-methyl-1H-1,2,4-triazole
—— 3-[(1R)-1-(2-fluorophenyl)ethyl]sulfanyl-4-methyl-5-(3-methylphenyl)-1,2,4-triazole —— C18H18FN3S
3-[(1R)-1-(2-fluorophenyl)ethyl]sulfanyl-4-methyl-5-(3-methylphenyl)-1,2,4-triazole
—— 1-(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)-3-[(1R)-2-imidazol-1-yl-1-phenylethyl]urea —— C20H26N6O
1-(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)-3-[(1R)-2-imidazol-1-yl-1-phenylethyl]urea
—— (2Z)-4-methyl-3-oxo-2-[(2-phenyl-1,3-thiazol-4-yl)methylidene]pentanenitrile —— C16H14N2OS
(2Z)-4-methyl-3-oxo-2-[(2-phenyl-1,3-thiazol-4-yl)methylidene]pentanenitrile
—— (2R)-4-N-(2-tert-butyl-4-phenylpyrazol-3-yl)morpholine-2,4-dicarboxamide —— C19H25N5O3
(2R)-4-N-(2-tert-butyl-4-phenylpyrazol-3-yl)morpholine-2,4-dicarboxamide