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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H35ClN4O3S
(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2S,3R)-2,3-dimethyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]thiomorpholine-4-carboxamide —— C12H19N3OS2
(2S,3R)-2,3-dimethyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]thiomorpholine-4-carboxamide
—— 2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C28H37N5O2S2
2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H34F2N4O3S
(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H27ClN4O4S
2-[(4R)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C28H30N4O3S2
2-[(4R)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H34F2N4O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C31H29ClN4O4S
2-[(4S)-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— N-(furan-2-ylmethyl)-2-[(4R)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H28N4O3S2
N-(furan-2-ylmethyl)-2-[(4R)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H35ClN4O3S
2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— (4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H34F2N4O3S
(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C30H33N5O2S2
2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C32H34N4O4S
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-3-tert-butyl-1-(2-ethylphenyl)-4-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C30H38N4O4S
2-[(4R)-3-tert-butyl-1-(2-ethylphenyl)-4-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C29H35ClN4O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— (4S)-3-tert-butyl-1-(2-ethylphenyl)-4-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H38N4O4S
(4S)-3-tert-butyl-1-(2-ethylphenyl)-4-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C30H29ClN4O4S
2-[(4R)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H29ClN4O3S
2-[(4R)-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C29H36N4O3S2
2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C29H32N4O3S2
2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C31H29ClN4O4S
2-[(4R)-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C29H33ClN4O2S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4S)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C32H31ClN4O4S
2-[(4S)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (3S)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-2,3-dihydro-1-benzothiophene-3-carboxamide —— C15H16N2O2S
(3S)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-2,3-dihydro-1-benzothiophene-3-carboxamide
—— 3-phenyl-5-[2-(trifluoromethyl)phenyl]-1H-indazole —— C20H13F3N2
3-phenyl-5-[2-(trifluoromethyl)phenyl]-1H-indazole
—— 2-[(4S)-4-(2-chlorophenyl)-7-oxo-1,3-diphenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C29H27ClN4O2S
2-[(4S)-4-(2-chlorophenyl)-7-oxo-1,3-diphenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4R)-3-tert-butyl-1-(4-fluorophenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H36FN5O2S
2-[(4R)-3-tert-butyl-1-(4-fluorophenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C28H34N4O3S2
2-[(4S)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C31H37ClN4O3S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (4S)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H30N4O3S2
(4S)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H25Cl2FN4O2S
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C29H35ClN4O2S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C31H36F2N4O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C29H35ClN4O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H34ClN5O2S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C31H36F2N4O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C31H36F2N4O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C28H37N5O2S2
2-[(4R)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 3-(2-bromophenyl)-6-[(Z)-2-(4-methoxyphenyl)ethenyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C18H13BrN4OS
3-(2-bromophenyl)-6-[(Z)-2-(4-methoxyphenyl)ethenyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (1R,2R,4R)-N-[2-(4-methyl-1,3-thiazol-2-yl)propan-2-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide —— C15H20N2OS
(1R,2R,4R)-N-[2-(4-methyl-1,3-thiazol-2-yl)propan-2-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
—— (3R)-1-methyl-3-[(2-methyl-1,3-thiazol-5-yl)methylsulfanyl]pyrrolidin-2-one —— C10H14N2OS2
(3R)-1-methyl-3-[(2-methyl-1,3-thiazol-5-yl)methylsulfanyl]pyrrolidin-2-one
—— 6-[(Z)-2-(4-methoxyphenyl)ethenyl]-3-(4-methylphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C19H16N4OS
6-[(Z)-2-(4-methoxyphenyl)ethenyl]-3-(4-methylphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (Z)-3-(5-bromothiophen-3-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]prop-2-enamide —— C12H11BrN2OS2
(Z)-3-(5-bromothiophen-3-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]prop-2-enamide
—— 3-(6-Aminopyridin-3-yl)-2-[1-(2-phenylethyl)imidazol-4-yl]propanoic acid —— C19H20N4O2
3-(6-Aminopyridin-3-yl)-2-[1-(2-phenylethyl)imidazol-4-yl]propanoic acid
—— (1R,2S,4R)-N-[2-(4-methyl-1,3-thiazol-2-yl)propan-2-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide —— C15H20N2OS
(1R,2S,4R)-N-[2-(4-methyl-1,3-thiazol-2-yl)propan-2-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
—— 3-(4-fluorophenyl)-6-[(Z)-2-phenylethenyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C17H11FN4S
3-(4-fluorophenyl)-6-[(Z)-2-phenylethenyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (3S)-1-methyl-3-[(2-methyl-1,3-thiazol-5-yl)methylsulfanyl]pyrrolidin-2-one —— C10H14N2OS2
(3S)-1-methyl-3-[(2-methyl-1,3-thiazol-5-yl)methylsulfanyl]pyrrolidin-2-one
—— 6-[(Z)-2-(furan-2-yl)ethenyl]-3-(4-methylphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C16H12N4OS
6-[(Z)-2-(furan-2-yl)ethenyl]-3-(4-methylphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 4-(4-Methoxyphenyl)-5-methyl-2-[1-(3-methylpyridin-2-yl)cyclopropyl]-1,3-thiazole —— C20H20N2OS
4-(4-Methoxyphenyl)-5-methyl-2-[1-(3-methylpyridin-2-yl)cyclopropyl]-1,3-thiazole
—— N-[(1S,4R)-7-azabicyclo[2.2.1]heptan-2-yl]-2-(2,5-difluorophenyl)-1,3-thiazole-5-carboxamide —— C16H15F2N3OS
N-[(1S,4R)-7-azabicyclo[2.2.1]heptan-2-yl]-2-(2,5-difluorophenyl)-1,3-thiazole-5-carboxamide