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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[4-(4-fluorophenyl)-2-(4-iminopiperidin-1-yl)-1,3-thiazol-5-yl]-N-[(1S)-1-phenylethyl]pyrimidin-2-amine —— C26H25FN6S
4-[4-(4-fluorophenyl)-2-(4-iminopiperidin-1-yl)-1,3-thiazol-5-yl]-N-[(1S)-1-phenylethyl]pyrimidin-2-amine
—— (17S)-N-(3-fluorophenyl)-15-methyl-13-phenyl-17-(4-propan-2-ylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C34H29FN6
(17S)-N-(3-fluorophenyl)-15-methyl-13-phenyl-17-(4-propan-2-ylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(2,4-dimethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C31H26N6O2S
(17R)-N-(2,4-dimethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— 1-[(3R,4S)-1-[2-(4-ethoxyphenyl)-1,3-benzoxazol-4-yl]-4-hydroxypentan-3-yl]imidazole-4-carboxamide;hydrochloride —— C24H27ClN4O4
1-[(3R,4S)-1-[2-(4-ethoxyphenyl)-1,3-benzoxazol-4-yl]-4-hydroxypentan-3-yl]imidazole-4-carboxamide;hydrochloride
—— (5S)-5-(3,4-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C29H32N4O6
(5S)-5-(3,4-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— (17S)-N-(4-ethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C31H26N6OS
(17S)-N-(4-ethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— 2-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl-[(1R)-1-phenylethyl]amino]acetic acid —— C29H30N2O4
2-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl-[(1R)-1-phenylethyl]amino]acetic acid
—— (17R)-17-(3-bromophenyl)-9-chloro-15-methyl-13-(4-nitrophenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaene —— C25H16BrClN6O2
(17R)-17-(3-bromophenyl)-9-chloro-15-methyl-13-(4-nitrophenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaene
—— (5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione —— C29H34N4O6
(5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione
—— (17S)-N-(2,4-dimethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C31H26N6O2S
(17S)-N-(2,4-dimethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-N-(1,3-benzodioxol-5-yl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C30H22N6O2S
(17S)-N-(1,3-benzodioxol-5-yl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(1,3-benzodioxol-5-yl)-15-methyl-13,17-diphenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H24N6O2
(17R)-N-(1,3-benzodioxol-5-yl)-15-methyl-13,17-diphenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— 1-(4-Methoxyphenyl)-7-methylsulfonyl-3-(phenoxymethyl)-4,5-dihydroimidazo[1,5-a]quinoline —— C26H24N2O4S
1-(4-Methoxyphenyl)-7-methylsulfonyl-3-(phenoxymethyl)-4,5-dihydroimidazo[1,5-a]quinoline
—— (5R)-5-(3,4-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C29H32N4O6
(5R)-5-(3,4-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— (17S)-N-(1,3-benzodioxol-5-yl)-15-methyl-13,17-diphenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H24N6O2
(17S)-N-(1,3-benzodioxol-5-yl)-15-methyl-13,17-diphenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(4-ethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C31H26N6OS
(17R)-N-(4-ethoxyphenyl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-17-(3-bromophenyl)-9-chloro-15-methyl-13-(4-nitrophenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaene —— C25H16BrClN6O2
(17S)-17-(3-bromophenyl)-9-chloro-15-methyl-13-(4-nitrophenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaene
—— 4-[3-[4-(1H-pyrrol-2-yl)phenyl]-4-(trifluoromethyl)-1H-pyrazol-5-yl]benzenesulfonamide —— C20H15F3N4O2S
4-[3-[4-(1H-pyrrol-2-yl)phenyl]-4-(trifluoromethyl)-1H-pyrazol-5-yl]benzenesulfonamide
—— N-cyclohexyl-N'-[8-(2,6-dichloro-4-methoxyphenyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-yl]ethane-1,2-diamine —— C22H28Cl2N6O
N-cyclohexyl-N'-[8-(2,6-dichloro-4-methoxyphenyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-yl]ethane-1,2-diamine
—— (17R)-N-(1,3-benzodioxol-5-yl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C30H22N6O2S
(17R)-N-(1,3-benzodioxol-5-yl)-15-methyl-13-phenyl-17-thiophen-2-yl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(3-fluorophenyl)-15-methyl-13-phenyl-17-(4-propan-2-ylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C34H29FN6
(17R)-N-(3-fluorophenyl)-15-methyl-13-phenyl-17-(4-propan-2-ylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-N-(4-ethoxyphenyl)-17-(2-fluorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C33H27FN6O
(17S)-N-(4-ethoxyphenyl)-17-(2-fluorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(3-chlorophenyl)-17-(2-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H25ClN6O
(17R)-N-(3-chlorophenyl)-17-(2-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-N-(1,3-benzodioxol-5-yl)-17-(2-fluorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H23FN6O2
(17S)-N-(1,3-benzodioxol-5-yl)-17-(2-fluorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-17-(4-chlorophenyl)-N-(3-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H25ClN6O
(17S)-17-(4-chlorophenyl)-N-(3-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-N-(3-chlorophenyl)-17-(2-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H25ClN6O
(17S)-N-(3-chlorophenyl)-17-(2-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (4-bromophenyl)-[(3R)-5-(1,3-diphenylpyrazol-4-yl)-3-phenyl-3,4-dihydropyrazol-2-yl]methanone —— C31H23BrN4O
(4-bromophenyl)-[(3R)-5-(1,3-diphenylpyrazol-4-yl)-3-phenyl-3,4-dihydropyrazol-2-yl]methanone
—— (17R)-17-(2-fluorophenyl)-N-(4-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H25FN6O
(17R)-17-(2-fluorophenyl)-N-(4-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17S)-17-(2-fluorophenyl)-N-(4-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H25FN6O
(17S)-17-(2-fluorophenyl)-N-(4-methoxyphenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(4-ethoxyphenyl)-17-(2-fluorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C33H27FN6O
(17R)-N-(4-ethoxyphenyl)-17-(2-fluorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— 4-[(3S)-2-(benzenesulfonyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-3-yl]-3-(4-methylphenyl)-1-phenylpyrazole —— C32H28N4O3S
4-[(3S)-2-(benzenesulfonyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-3-yl]-3-(4-methylphenyl)-1-phenylpyrazole
—— [3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-cyclopropylmethyl-(2-methoxy-ethyl)-amine —— C21H27BrN6O
[3-(2-Bromo-4-isopropyl-phenyl)-5-methyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl]-cyclopropylmethyl-(2-methoxy-ethyl)-amine
—— 3-[[2-(4,5-Diphenyl-1,3-oxazol-2-yl)cyclohexen-1-yl]methyl]benzoic acid —— C29H25NO3
3-[[2-(4,5-Diphenyl-1,3-oxazol-2-yl)cyclohexen-1-yl]methyl]benzoic acid
—— 5-methoxy-2-methyl-4-[2-[[(E)-1-[4-[(E)-C-methyl-N-prop-2-enoxycarbonimidoyl]phenyl]ethylideneamino]oxymethyl]phenyl]-1,2,4-triazol-3-one —— C24H27N5O4
5-methoxy-2-methyl-4-[2-[[(E)-1-[4-[(E)-C-methyl-N-prop-2-enoxycarbonimidoyl]phenyl]ethylideneamino]oxymethyl]phenyl]-1,2,4-triazol-3-one
—— 2-bromo-N-[(1R)-2,2,2-trichloro-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylamino]ethyl]benzamide —— C21H19BrCl3N5O2S
2-bromo-N-[(1R)-2,2,2-trichloro-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylamino]ethyl]benzamide
—— 4-[2-[[4-[(E)-N-[(Z)-3-chloroprop-2-enoxy]-C-methylcarbonimidoyl]-3-methylphenoxy]methyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one —— C23H25ClN4O4
4-[2-[[4-[(E)-N-[(Z)-3-chloroprop-2-enoxy]-C-methylcarbonimidoyl]-3-methylphenoxy]methyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one
—— 4-[4-Bromo-5-(4-methoxyphenyl)-3-methylpyrazol-1-yl]-2-(hydroxymethyl)benzenesulfonamide —— C18H18BrN3O4S
4-[4-Bromo-5-(4-methoxyphenyl)-3-methylpyrazol-1-yl]-2-(hydroxymethyl)benzenesulfonamide
—— 3-(5-aminopentyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1-(thiophen-3-ylmethyl)-1,3-diazinan-4-one —— C23H27N5OS2
3-(5-aminopentyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1-(thiophen-3-ylmethyl)-1,3-diazinan-4-one
—— N-[4-(8-benzyloxy-3-cyclohexylaminoimidazo[1,2-a]pyridin-2-yl)-phenyl]-acetamide —— C28H30N4O2
N-[4-(8-benzyloxy-3-cyclohexylaminoimidazo[1,2-a]pyridin-2-yl)-phenyl]-acetamide
—— 5-[4-[2-[5-methyl-2-(2-pyrimidinylthio)methyl-4-oxazolyl]ethoxy]benzyl]-2,4-thiazolidinedione —— C21H20N4O4S2
5-[4-[2-[5-methyl-2-(2-pyrimidinylthio)methyl-4-oxazolyl]ethoxy]benzyl]-2,4-thiazolidinedione
—— methyl (2E,4R,5S,6E)-3,5-dimethoxy-4-methyl-7-[4-[(Z)-C-methyl-N-phenylmethoxycarbonimidoyl]-1,3-thiazol-2-yl]hepta-2,6-dienoate —— C23H28N2O5S
methyl (2E,4R,5S,6E)-3,5-dimethoxy-4-methyl-7-[4-[(Z)-C-methyl-N-phenylmethoxycarbonimidoyl]-1,3-thiazol-2-yl]hepta-2,6-dienoate
—— N-(1-phenyltetrazol-5-yl)imino-N'-(4-propylanilino)-2,3-dihydro-1-benzofuran-5-carboximidamide —— C25H24N8O
N-(1-phenyltetrazol-5-yl)imino-N'-(4-propylanilino)-2,3-dihydro-1-benzofuran-5-carboximidamide
—— 4-(1,4-dihydroindeno[1,2-c]pyrazol-3-yl)-N-(2-morpholin-4-ylethyl)aniline;dihydrochloride —— C22H26Cl2N4O
4-(1,4-dihydroindeno[1,2-c]pyrazol-3-yl)-N-(2-morpholin-4-ylethyl)aniline;dihydrochloride
—— 3-[[4-[2-(4-Butylphenyl)tetrazol-5-yl]phenyl]sulfonylamino]-2-methylpropanoic acid —— C21H25N5O4S
3-[[4-[2-(4-Butylphenyl)tetrazol-5-yl]phenyl]sulfonylamino]-2-methylpropanoic acid
—— 8-(4-tert-butylphenyl)-5-(diethoxyphosphorylmethyl)-7H-[1,2,4]triazolo[5,1-f]purine —— C21H27N6O3P
8-(4-tert-butylphenyl)-5-(diethoxyphosphorylmethyl)-7H-[1,2,4]triazolo[5,1-f]purine
—— 3-(2,4-dichlorophenyl)-N-ethyl-1,5-dimethyl-N-[(4-methylphenyl)methyl]pyrazolo[4,3-b]pyridin-7-amine —— C24H24Cl2N4
3-(2,4-dichlorophenyl)-N-ethyl-1,5-dimethyl-N-[(4-methylphenyl)methyl]pyrazolo[4,3-b]pyridin-7-amine
—— 2-bromo-N-[(1S)-2,2,2-trichloro-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylamino]ethyl]benzamide —— C21H19BrCl3N5O2S
2-bromo-N-[(1S)-2,2,2-trichloro-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylamino]ethyl]benzamide
—— 3-[[2-(4,5-Diphenyl-1,3-oxazol-2-yl)cyclohex-2-en-1-yl]methyl]benzamide —— C29H26N2O2
3-[[2-(4,5-Diphenyl-1,3-oxazol-2-yl)cyclohex-2-en-1-yl]methyl]benzamide
—— 8,9-dimethoxy-1-phenyl-N-(2-phenylpropan-2-yl)-5,6-dihydroimidazo[5,1-a]isoquinolin-3-amine —— C28H29N3O2
8,9-dimethoxy-1-phenyl-N-(2-phenylpropan-2-yl)-5,6-dihydroimidazo[5,1-a]isoquinolin-3-amine
—— benzyl N-[(1S)-1-diethoxyphosphoryl-1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2,2,2-trifluoroethyl]carbamate —— C25H29F3N3O6P
benzyl N-[(1S)-1-diethoxyphosphoryl-1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2,2,2-trifluoroethyl]carbamate