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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-1-[2-[4-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetyl]piperidine-3-carboxamide —— C22H30N6O3
(3S)-1-[2-[4-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetyl]piperidine-3-carboxamide
—— 1-[(3R)-3-methylpiperidin-1-yl]-2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]ethanone —— C22H31N5O2
1-[(3R)-3-methylpiperidin-1-yl]-2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]ethanone
—— methyl 2-methyl-5-[[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]methyl]furan-3-carboxylate —— C22H26N4O4
methyl 2-methyl-5-[[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]methyl]furan-3-carboxylate
—— 1-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-3-(4-fluorophenyl)urea —— C23H25F2N5O2
1-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-3-(4-fluorophenyl)urea
—— N-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-2-methylbenzamide —— C24H27FN4O2
N-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-2-methylbenzamide
—— 1-[2-[4-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetyl]piperidine-4-carboxamide —— C22H30N6O3
1-[2-[4-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetyl]piperidine-4-carboxamide
—— 5-[(1R)-1-[4-[[5-(3-chlorophenyl)-1,3-oxazol-2-yl]methyl]piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole —— C24H24ClN5O2
5-[(1R)-1-[4-[[5-(3-chlorophenyl)-1,3-oxazol-2-yl]methyl]piperazin-1-yl]ethyl]-3-phenyl-1,2,4-oxadiazole
—— 2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]acetamide —— C19H19Cl2N3O3
2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]acetamide
—— N-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-2-methylbenzamide —— C24H27FN4O2
N-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-2-methylbenzamide
—— (2S)-1-(4-ethylpiperazin-1-yl)-2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]propan-1-one —— C23H34N6O2
(2S)-1-(4-ethylpiperazin-1-yl)-2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]propan-1-one
—— 2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C21H21ClFN3O2
2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-5-(4-methoxyphenyl)-1-phenylpyrazole-3-carboxamide —— C23H21N3O4
N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-5-(4-methoxyphenyl)-1-phenylpyrazole-3-carboxamide
—— N-methyl-N-[(2-methylphenyl)methyl]-2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetamide —— C25H31N5O2
N-methyl-N-[(2-methylphenyl)methyl]-2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetamide
—— (1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-ethyl-1-(3-methoxyphenyl)ethanamine —— C21H23F2N3O3
(1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-ethyl-1-(3-methoxyphenyl)ethanamine
—— N-methyl-N-[(2-methylphenyl)methyl]-2-[4-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetamide —— C25H31N5O2
N-methyl-N-[(2-methylphenyl)methyl]-2-[4-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetamide
—— 2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]acetamide —— C19H19Cl2N3O3
2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]acetamide
—— N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-2-pyrazol-1-ylbenzamide —— C16H15N3O3
N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-2-pyrazol-1-ylbenzamide
—— 2-(4-fluorophenoxy)-1-[4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]ethanone —— C21H23FN6O2
2-(4-fluorophenoxy)-1-[4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]ethanone
—— 2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]acetamide —— C19H19Cl2N3O3
2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]acetamide
—— 2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]acetamide —— C20H20F3N3O3
2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]acetamide
—— 2-(4-fluorophenoxy)-1-[4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]ethanone —— C21H23FN6O2
2-(4-fluorophenoxy)-1-[4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]ethanone
—— 1-(4-bromophenyl)-5-ethyl-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]pyrazole-4-carboxamide —— C18H18BrN3O3
1-(4-bromophenyl)-5-ethyl-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]pyrazole-4-carboxamide
—— 2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]acetamide —— C19H19Cl2N3O3
2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]acetamide
—— 1-[2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetyl]piperidine-4-carboxamide —— C22H30N6O3
1-[2-[4-[(1R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]acetyl]piperidine-4-carboxamide
—— 1-(4-bromophenyl)-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]pyrazole-4-carboxamide —— C18H15BrFN3O2
1-(4-bromophenyl)-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]pyrazole-4-carboxamide
—— [1-[(2R,3R)-2-(2,4-difluorophenyl)-2-hydroxy-3-[2-oxo-3-[4-(tetrazol-1-yl)phenyl]imidazolidin-1-yl]butyl]-1,2,4-triazol-4-ium-4-yl]methyl ethyl carbonate —— C26H28F2N9O5+
[1-[(2R,3R)-2-(2,4-difluorophenyl)-2-hydroxy-3-[2-oxo-3-[4-(tetrazol-1-yl)phenyl]imidazolidin-1-yl]butyl]-1,2,4-triazol-4-ium-4-yl]methyl ethyl carbonate
—— 2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]acetamide —— C20H20F3N3O3
2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]acetamide
—— 1-(3-bromophenyl)-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-4,5,6,7-tetrahydroindazole-3-carboxamide —— C20H20BrN3O3
1-(3-bromophenyl)-N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-4,5,6,7-tetrahydroindazole-3-carboxamide
—— N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-5-(4-methoxyphenyl)-1-phenylpyrazole-3-carboxamide —— C23H21N3O4
N-[(2R)-2-(furan-2-yl)-2-hydroxyethyl]-5-(4-methoxyphenyl)-1-phenylpyrazole-3-carboxamide
—— (1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-ethyl-1-(3-methoxyphenyl)ethanamine —— C21H23F2N3O3
(1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-ethyl-1-(3-methoxyphenyl)ethanamine
—— 5-chloro-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-methoxy-4-(tetrazol-1-yl)benzamide —— C17H15ClFN5O3
5-chloro-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-methoxy-4-(tetrazol-1-yl)benzamide
—— 2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C21H20Cl2FN3O2
2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 1-(4-bromophenyl)-5-ethyl-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]pyrazole-4-carboxamide —— C20H19BrFN3O2
1-(4-bromophenyl)-5-ethyl-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]pyrazole-4-carboxamide
—— 2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C21H20Cl2FN3O2
2-[1-(2,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 2-[1-(3-chloro-4-methylphenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C22H23ClFN3O2
2-[1-(3-chloro-4-methylphenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 5-chloro-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-methoxy-4-(tetrazol-1-yl)benzamide —— C17H15ClFN5O3
5-chloro-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-methoxy-4-(tetrazol-1-yl)benzamide
—— N-[(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]methanesulfonamide —— C17H23FN4O3S
N-[(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]methanesulfonamide
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-(4-pyridin-3-ylsulfonylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole —— C20H22FN5O3S
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-(4-pyridin-3-ylsulfonylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole
—— 1-(3-bromophenyl)-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-4,5,6,7-tetrahydroindazole-3-carboxamide —— C20H20BrN3O3
1-(3-bromophenyl)-N-[(2S)-2-(furan-2-yl)-2-hydroxyethyl]-4,5,6,7-tetrahydroindazole-3-carboxamide
—— N-[3-{2-[(5-bromo-2-pyrimidinyl)oxy]ethoxy}-1-methyl-4-(4-methylphenyl)-1H-pyrazol-5-yl]4-(tert-pentyl)benzenesulfonamide —— C28H32BrN5O4S
N-[3-{2-[(5-bromo-2-pyrimidinyl)oxy]ethoxy}-1-methyl-4-(4-methylphenyl)-1H-pyrazol-5-yl]4-(tert-pentyl)benzenesulfonamide
—— 5-[3-[4-[2-(4-Fluorophenyl)-2-(4-propan-2-ylpiperazin-1-yl)ethyl]piperazin-1-yl]propyl]-2,4-diphenyl-1,3-thiazole —— C37H46FN5S
5-[3-[4-[2-(4-Fluorophenyl)-2-(4-propan-2-ylpiperazin-1-yl)ethyl]piperazin-1-yl]propyl]-2,4-diphenyl-1,3-thiazole
—— (3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-1H-indol-2-one;4-[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide —— C32H28F3N5O3S
(3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-1H-indol-2-one;4-[5-(4-methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide
—— 2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C21H21ClFN3O2
2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 6-butyl-8-[5-[4-(1-hydroxy-2-methylpropan-2-yl)piperazin-1-yl]sulfonyl-2-propoxyphenyl]-1H-[1,2,4]triazolo[3,4-f]purin-5-one —— C27H38N8O5S
6-butyl-8-[5-[4-(1-hydroxy-2-methylpropan-2-yl)piperazin-1-yl]sulfonyl-2-propoxyphenyl]-1H-[1,2,4]triazolo[3,4-f]purin-5-one
—— N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-pyrazol-1-ylbenzamide —— C18H16FN3O2
N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-pyrazol-1-ylbenzamide
—— 2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C22H21F4N3O2
2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C21H20Cl2FN3O2
2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C21H20Cl2FN3O2
2-[1-(3,4-dichlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C22H21F4N3O2
2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— 1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(2-methoxyphenyl)piperidine-4-carboxamide —— C24H27FN4O3
1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(2-methoxyphenyl)piperidine-4-carboxamide