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中文名称 英文名称 CAS号 化学式 结构式图片
—— Methyl 2-[2-[4-(trifluoromethyl)pyridin-3-yl]-1,3-oxazol-4-yl]acetate —— C12H9F3N2O3
Methyl 2-[2-[4-(trifluoromethyl)pyridin-3-yl]-1,3-oxazol-4-yl]acetate
—— (4S)-6-amino-3-methyl-4-nonyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C17H26N4O
(4S)-6-amino-3-methyl-4-nonyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (2S)-2,3,3,3-tetrafluoro-2-[(2S)-1,1,2,3,3,3-hexafluoro-2-(1,1,2,2,3,3,3-heptafluoropropoxy)propoxy]-N'-(1,3-thiazol-2-yl)propanimidamide —— C12H4F17N3O2S
(2S)-2,3,3,3-tetrafluoro-2-[(2S)-1,1,2,3,3,3-hexafluoro-2-(1,1,2,2,3,3,3-heptafluoropropoxy)propoxy]-N'-(1,3-thiazol-2-yl)propanimidamide
—— 6-(cyclopropylamino)-9-[4-(dimethylamino)phenyl]-2-(trifluoromethyl)purine —— C17H17F3N6
6-(cyclopropylamino)-9-[4-(dimethylamino)phenyl]-2-(trifluoromethyl)purine
—— 4-N-(furan-2-ylmethyl)-4-N,5-dimethyl-2-N-[4-(1,3-oxazol-5-yl)phenyl]pyrimidine-2,4-diamine —— C20H19N5O2
4-N-(furan-2-ylmethyl)-4-N,5-dimethyl-2-N-[4-(1,3-oxazol-5-yl)phenyl]pyrimidine-2,4-diamine
—— N-[(Z)-(5-chloro-2-phenyl-1,3-oxazol-4-yl)methylideneamino]-4-decoxybenzamide —— C27H32ClN3O3
N-[(Z)-(5-chloro-2-phenyl-1,3-oxazol-4-yl)methylideneamino]-4-decoxybenzamide
—— 3-(4-methylphenyl)-4-[(Z)-(2,4,6-tribromo-3-hydroxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C16H11Br3N4OS
3-(4-methylphenyl)-4-[(Z)-(2,4,6-tribromo-3-hydroxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— N-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-4-decoxybenzamide —— C28H35ClN4O2
N-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-4-decoxybenzamide
—— 8-Phenyl-2,6-di-piperidin-1-yl-7H-purine —— C21H26N6
8-Phenyl-2,6-di-piperidin-1-yl-7H-purine
—— 5-[2-Fluoro-5-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]phenyl]-3-methyl-1,2,4-oxadiazole —— C15H8F4N6O
5-[2-Fluoro-5-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]phenyl]-3-methyl-1,2,4-oxadiazole
—— methyl 4-[2-[(3-chlorophenyl)methyl]-3-sulfanylidene-1H-1,2,4-triazol-5-yl]benzoate —— C17H14ClN3O2S
methyl 4-[2-[(3-chlorophenyl)methyl]-3-sulfanylidene-1H-1,2,4-triazol-5-yl]benzoate
—— 3-(4-Fluoro-3-pyrimidin-2-ylphenyl)-7-(trifluoromethyl)imidazo[1,2-a]pyrimidine —— C17H9F4N5
3-(4-Fluoro-3-pyrimidin-2-ylphenyl)-7-(trifluoromethyl)imidazo[1,2-a]pyrimidine
—— Ethyl 4-[2-[4-(2-methylpyrazol-3-yl)phenoxy]ethyl]piperazine-1-carboxylate —— C19H26N4O3
Ethyl 4-[2-[4-(2-methylpyrazol-3-yl)phenoxy]ethyl]piperazine-1-carboxylate
—— 2-[1-(4-Fluoro-3-methylphenyl)cyclopropyl]-4-(4-methoxyphenyl)-5-methyl-1,3-thiazole —— C21H20FNOS
2-[1-(4-Fluoro-3-methylphenyl)cyclopropyl]-4-(4-methoxyphenyl)-5-methyl-1,3-thiazole
—— ethyl 2-[[(2S)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C31H35N5O6S2
ethyl 2-[[(2S)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— diethyl 5-[[(2R)-2-[[5-[[(3,4-dimethoxybenzoyl)amino]methyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-3-methylthiophene-2,4-dicarboxylate —— C32H34FN5O8S2
diethyl 5-[[(2R)-2-[[5-[[(3,4-dimethoxybenzoyl)amino]methyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-3-methylthiophene-2,4-dicarboxylate
—— 4-[4-[2-[4-(1H-pyrazol-5-yl)phenoxy]ethyl]piperazin-1-yl]butanamide —— C19H27N5O2
4-[4-[2-[4-(1H-pyrazol-5-yl)phenoxy]ethyl]piperazin-1-yl]butanamide
—— [1-[2-(4-Methyl-1,3-thiazol-5-yl)ethyldisulfanyl]-3-nitrooxypropan-2-yl] nitrate —— C9H13N3O6S3
[1-[2-(4-Methyl-1,3-thiazol-5-yl)ethyldisulfanyl]-3-nitrooxypropan-2-yl] nitrate
—— ethyl 2-[[(2R)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C29H31N5O5S2
ethyl 2-[[(2R)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— 1-(4-Methylsulfonylbutyl)-4,5-diphenylimidazole —— C20H22N2O2S
1-(4-Methylsulfonylbutyl)-4,5-diphenylimidazole
—— 7-(Cyclopropylmethoxy)-2-(4-fluorophenyl)-3-pyrimidin-4-ylpyrazolo[1,5-a]pyridine —— C21H17FN4O
7-(Cyclopropylmethoxy)-2-(4-fluorophenyl)-3-pyrimidin-4-ylpyrazolo[1,5-a]pyridine
—— 4-[[4-(3-Methyl-1-phenylpyrazol-4-yl)pyrimidin-2-yl]amino]benzonitrile —— C21H16N6
4-[[4-(3-Methyl-1-phenylpyrazol-4-yl)pyrimidin-2-yl]amino]benzonitrile
—— N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C32H30N6O5S3
N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[4-(4-ethoxyphenyl)-5-[2-[(3R)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C32H30N6O4S3
N-[[4-(4-ethoxyphenyl)-5-[2-[(3R)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— ethyl 2-[[(2R)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C31H35N5O6S2
ethyl 2-[[(2R)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— diethyl 5-[[(2R)-2-[[5-[(furan-2-carbonylamino)methyl]-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-3-methylthiophene-2,4-dicarboxylate —— C29H31N5O8S2
diethyl 5-[[(2R)-2-[[5-[(furan-2-carbonylamino)methyl]-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-3-methylthiophene-2,4-dicarboxylate
—— N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(2,5-dimethylphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C33H32N6O4S3
N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(2,5-dimethylphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(2,3-dimethylphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C33H32N6O4S3
N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(2,3-dimethylphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[5-[2-[(3S)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C33H32N6O5S3
N-[[5-[2-[(3S)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— 8-FLUORO-2-(4-FLUOROPHENYL)-6-[(2S,5S)-5-HYDROXYMETHYL OXOLAN-2-YL]-5,6-DIHYDRO[1,3]-DIAZOLO[1,2-C][1,3]DIAZIN-5-ONE 348597-65-9 C17H15F2N3O3
8-FLUORO-2-(4-FLUOROPHENYL)-6-[(2S,5S)-5-HYDROXYMETHYL OXOLAN-2-YL]-5,6-DIHYDRO[1,3]-DIAZOLO[1,2-C][1,3]DIAZIN-5-ONE
—— N-[[4-(4-bromophenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C30H25BrN6O3S2
N-[[4-(4-bromophenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— 5-fluoro-N-(4-fluoro-3-methylphenyl)-4-imidazo[2,1-b][1,3]thiazol-5-yl-1,3-thiazol-2-amine —— C15H10F2N4S2
5-fluoro-N-(4-fluoro-3-methylphenyl)-4-imidazo[2,1-b][1,3]thiazol-5-yl-1,3-thiazol-2-amine
—— ethyl 2-[[(2S)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C29H31N5O5S2
ethyl 2-[[(2S)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— N-[[4-(4-bromophenyl)-5-[2-[(3R)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C30H25BrN6O2S3
N-[[4-(4-bromophenyl)-5-[2-[(3R)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[4-(2,3-dimethylphenyl)-5-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C31H27FN6O3S2
N-[[4-(2,3-dimethylphenyl)-5-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— N-[[4-(4-fluorophenyl)-5-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C29H22F2N6O3S2
N-[[4-(4-fluorophenyl)-5-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— 2-[4-[2-[4-(Diaminomethylideneamino)phenyl]-1,3-thiazol-4-yl]phenyl]guanidine —— C17H17N7S
2-[4-[2-[4-(Diaminomethylideneamino)phenyl]-1,3-thiazol-4-yl]phenyl]guanidine
—— N-[[4-(2,3-dimethylphenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C32H30N6O2S3
N-[[4-(2,3-dimethylphenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[4-(3-chlorophenyl)-5-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C29H22ClFN6O2S3
N-[[4-(3-chlorophenyl)-5-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[5-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(3-methylphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C30H25FN6O2S3
N-[[5-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(3-methylphenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[4-(4-ethoxyphenyl)-5-[2-[(3R)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C32H30N6O3S3
N-[[4-(4-ethoxyphenyl)-5-[2-[(3R)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[5-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-phenyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C29H23FN6O2S3
N-[[5-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-phenyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[4-(2,5-dimethylphenyl)-5-[2-[(3S)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C32H30N6O4S2
N-[[4-(2,5-dimethylphenyl)-5-[2-[(3S)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C31H27FN6O4S3
N-[[5-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— N-[[4-(2-methoxyphenyl)-5-[2-[(3S)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C31H28N6O5S2
N-[[4-(2-methoxyphenyl)-5-[2-[(3S)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— N-[[4-(4-bromophenyl)-5-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C29H22BrFN6O2S3
N-[[4-(4-bromophenyl)-5-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide
—— 4-[3-[3-(Trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]phenyl]thiadiazole —— C14H7F3N6S
4-[3-[3-(Trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]phenyl]thiadiazole
—— N-[[4-(2,3-dimethylphenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C32H30N6O3S2
N-[[4-(2,3-dimethylphenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— N-[[4-(2,5-dimethylphenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide —— C32H30N6O3S2
N-[[4-(2,5-dimethylphenyl)-5-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]furan-2-carboxamide
—— N-[[4-(4-fluorophenyl)-5-[2-[(3R)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide —— C30H25FN6O3S3
N-[[4-(4-fluorophenyl)-5-[2-[(3R)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]methyl]thiophene-2-carboxamide