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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-ethyl-5-[(1S)-1-[(1-phenylpyrazol-4-yl)methylsulfonyl]ethyl]-1,2,4-oxadiazole —— C16H18N4O3S
3-ethyl-5-[(1S)-1-[(1-phenylpyrazol-4-yl)methylsulfonyl]ethyl]-1,2,4-oxadiazole
—— (2R)-2-cycloheptyloxy-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cyclopentyl]propanamide —— C18H29N3O3
(2R)-2-cycloheptyloxy-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cyclopentyl]propanamide
—— 5-tert-butyl-3-[[(S)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole —— C17H20N4O2S
5-tert-butyl-3-[[(S)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole
—— 3-ethyl-5-[(1R)-1-[(1-phenylpyrazol-4-yl)methylsulfonyl]ethyl]-1,2,4-oxadiazole —— C16H18N4O3S
3-ethyl-5-[(1R)-1-[(1-phenylpyrazol-4-yl)methylsulfonyl]ethyl]-1,2,4-oxadiazole
—— 1-[(2S,4S)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea —— C14H19N3O3S
1-[(2S,4S)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea
—— 5-tert-butyl-3-[[(R)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole —— C17H20N4O2S
5-tert-butyl-3-[[(R)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,2,4-oxadiazole
—— 2-(4-fluorophenoxy)-N-[(E)-(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]acetamide —— C23H24FN5O2
2-(4-fluorophenoxy)-N-[(E)-(3-methyl-1-phenyl-5-pyrrolidin-1-ylpyrazol-4-yl)methylideneamino]acetamide
—— 1-[4-[(1R)-1-[(2-cyclobutylideneacetyl)amino]ethyl]phenyl]triazole-4-carboxamide —— C17H19N5O2
1-[4-[(1R)-1-[(2-cyclobutylideneacetyl)amino]ethyl]phenyl]triazole-4-carboxamide
—— 1-[(2R,4S)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea —— C14H19N3O3S
1-[(2R,4S)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea
—— 1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-[(1S,3R)-3-ethylsulfanylcyclohexyl]-2-methylguanidine —— C17H30N4OS
1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-[(1S,3R)-3-ethylsulfanylcyclohexyl]-2-methylguanidine
—— 1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-[(1R,3R)-3-ethylsulfanylcyclohexyl]-2-methylguanidine —— C17H30N4OS
1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-[(1R,3R)-3-ethylsulfanylcyclohexyl]-2-methylguanidine
—— 1-[(2S,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea —— C14H19N3O3S
1-[(2S,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea
—— (1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-N-(ethylsulfamoyl)ethanamine —— C15H22N4O2S
(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]-N-(ethylsulfamoyl)ethanamine
—— 1-[(2R,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea —— C14H19N3O3S
1-[(2R,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-3-[(1S)-1-(1,3-thiazol-2-yl)ethyl]urea
—— 2-methyl-5-[[(S)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,3-thiazole —— C15H15N3OS2
2-methyl-5-[[(S)-(1-phenylpyrazol-4-yl)methylsulfinyl]methyl]-1,3-thiazole
—— (2S)-2-cycloheptyloxy-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cyclopentyl]propanamide —— C18H29N3O3
(2S)-2-cycloheptyloxy-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cyclopentyl]propanamide
—— 3,4-dichloro-N-[2-[2-(4-chlorophenyl)-3-oxo-5-phenyl-1H-pyrazol-4-yl]-2-oxoethyl]-N-propylbenzamide —— C27H22Cl3N3O3
3,4-dichloro-N-[2-[2-(4-chlorophenyl)-3-oxo-5-phenyl-1H-pyrazol-4-yl]-2-oxoethyl]-N-propylbenzamide
—— 1-[4-[1-(difluoromethyl)imidazol-2-yl]phenyl]-3-[(1S,2R,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]urea —— C17H18F2N4O2
1-[4-[1-(difluoromethyl)imidazol-2-yl]phenyl]-3-[(1S,2R,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]urea
—— 1-[4-[1-(difluoromethyl)imidazol-2-yl]phenyl]-3-[(1S,2S,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]urea —— C17H18F2N4O2
1-[4-[1-(difluoromethyl)imidazol-2-yl]phenyl]-3-[(1S,2S,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]urea
—— (1S)-2-[[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]methylamino]-1-(furan-2-yl)ethanol —— C22H20FN3O2
(1S)-2-[[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]methylamino]-1-(furan-2-yl)ethanol
—— (3R)-N-[[2-(3-fluorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine —— C22H23FN2O4S
(3R)-N-[[2-(3-fluorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine
—— [4-[(1S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone —— C19H24ClN5O3
[4-[(1S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone
—— 1-[(4R)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C25H27N7O
1-[(4R)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 1-[(4S)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C25H27N7O
1-[(4S)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— (2S)-N-[(4-methylphenyl)methyl]-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]propanamide —— C20H22N2O2S2
(2S)-N-[(4-methylphenyl)methyl]-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]propanamide
—— (2R)-2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]-N-(2,2,2-trifluoroethyl)propanamide —— C10H13F3N2O2S
(2R)-2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]-N-(2,2,2-trifluoroethyl)propanamide
—— (1R)-2-[[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]methylamino]-1-(furan-2-yl)ethanol —— C22H20FN3O2
(1R)-2-[[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]methylamino]-1-(furan-2-yl)ethanol
—— 1-(4-phenyl-1,3-thiazol-2-yl)-3-[(2R)-1-piperidin-1-ylpropan-2-yl]urea —— C18H24N4OS
1-(4-phenyl-1,3-thiazol-2-yl)-3-[(2R)-1-piperidin-1-ylpropan-2-yl]urea
—— N-[(1R)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-methoxy-3-(2-methoxyethoxy)aniline —— C21H24FN3O4
N-[(1R)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-methoxy-3-(2-methoxyethoxy)aniline
—— (3S)-N-[[2-(3-fluorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine —— C22H23FN2O4S
(3S)-N-[[2-(3-fluorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine
—— 1-[(4S)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C25H27N7O
1-[(4S)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— [4-[(1R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone —— C19H24ClN5O3
[4-[(1R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone
—— (2S)-N-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]-1-thiophen-2-ylpropan-2-amine —— C17H17FN2S2
(2S)-N-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]-1-thiophen-2-ylpropan-2-amine
—— 1-[4-[(1S)-1-[(2-cyclobutylideneacetyl)amino]ethyl]phenyl]triazole-4-carboxamide —— C17H19N5O2
1-[4-[(1S)-1-[(2-cyclobutylideneacetyl)amino]ethyl]phenyl]triazole-4-carboxamide
—— N-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-methoxy-3-(2-methoxyethoxy)aniline —— C21H24FN3O4
N-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-methoxy-3-(2-methoxyethoxy)aniline
—— (2R)-N-[(4-methylphenyl)methyl]-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]propanamide —— C20H22N2O2S2
(2R)-N-[(4-methylphenyl)methyl]-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]propanamide
—— (3R)-4-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-3-methylmorpholine —— C15H17F2N3O3
(3R)-4-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-3-methylmorpholine
—— (3R)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine —— C22H23ClN2O4S
(3R)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine
—— (2S)-2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]-N-(2,2,2-trifluoroethyl)propanamide —— C10H13F3N2O2S
(2S)-2-[(5-methyl-1,2-oxazol-3-yl)methylsulfanyl]-N-(2,2,2-trifluoroethyl)propanamide
—— (2R)-N-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]-1-thiophen-2-ylpropan-2-amine —— C17H17FN2S2
(2R)-N-[[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl]-1-thiophen-2-ylpropan-2-amine
—— 1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-[(1R,3S)-3-ethylsulfanylcyclohexyl]-2-methylguanidine —— C17H30N4OS
1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-[(1R,3S)-3-ethylsulfanylcyclohexyl]-2-methylguanidine
—— 4-[(E)-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione —— C22H18N6OS
4-[(E)-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione
—— (3S)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine —— C22H23ClN2O4S
(3S)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-N-[(4-methoxyphenyl)methyl]-1,1-dioxothiolan-3-amine
—— N-[(E)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-2-(2-fluorophenoxy)acetamide —— C24H19FN4O2
N-[(E)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-2-(2-fluorophenoxy)acetamide
—— 1-[(4R)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C25H27N7O
1-[(4R)-1-benzyl-4,5,6,7-tetrahydroindazol-4-yl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— N-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-methylfuran-3-carboxamide —— C17H14ClFN4O2
N-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-methylfuran-3-carboxamide
—— 1-(4-phenyl-1,3-thiazol-2-yl)-3-[(2S)-1-piperidin-1-ylpropan-2-yl]urea —— C18H24N4OS
1-(4-phenyl-1,3-thiazol-2-yl)-3-[(2S)-1-piperidin-1-ylpropan-2-yl]urea
—— 5-[[(2S)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C23H24N6O2
5-[[(2S)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— N-[(E)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-2-methylfuran-3-carboxamide —— C22H18N4O2
N-[(E)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-2-methylfuran-3-carboxamide
—— 3-(4-fluorophenyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-5-carboxamide —— C18H16FN3O2
3-(4-fluorophenyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-5-carboxamide