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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-imidazol-1-yl-N-[N-[4-imidazol-1-yl-3-(trifluoromethyl)benzoyl]carbamimidoyl]-3-(trifluoromethyl)benzamide —— C23H15F6N7O2
4-imidazol-1-yl-N-[N-[4-imidazol-1-yl-3-(trifluoromethyl)benzoyl]carbamimidoyl]-3-(trifluoromethyl)benzamide
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-methoxyphenyl)methanone —— C23H25FN4O3
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-methoxyphenyl)methanone
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-phenylmethanone —— C23H25FN4O2
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-phenylmethanone
—— (1S)-N-[(2,4-difluorophenyl)methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine —— C19H18F3N3O
(1S)-N-[(2,4-difluorophenyl)methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine
—— 2-[4-(4-fluorophenyl)-5-[2-(3-methoxypropylamino)pyrimidin-4-yl]-1H-imidazol-2-yl]-N-(2-methoxyethyl)-5-methyl-1,3-dioxane-5-carboxamide —— C26H33FN6O5
2-[4-(4-fluorophenyl)-5-[2-(3-methoxypropylamino)pyrimidin-4-yl]-1H-imidazol-2-yl]-N-(2-methoxyethyl)-5-methyl-1,3-dioxane-5-carboxamide
—— (5E)-5-[[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(Z)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C26H17N5O2S
(5E)-5-[[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(Z)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— 2-(2,6-dichlorophenyl)-4-(3-bromophenyl)-5-(2-[3-hydroxypropylamino]pyrimidin-4-yl)-N-H-imidazole —— C22H18BrCl2N5O
2-(2,6-dichlorophenyl)-4-(3-bromophenyl)-5-(2-[3-hydroxypropylamino]pyrimidin-4-yl)-N-H-imidazole
—— (1R)-N-[(2,4-difluorophenyl)methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine —— C19H18F3N3O
(1R)-N-[(2,4-difluorophenyl)methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine
—— 2-[(3-Methoxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid —— C29H28N2O7
2-[(3-Methoxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid
—— 3-cyano-4-(3-dibromomethylenecyclobutyl)-1-(2,6-dichloro-4-trifluoromethylphenyl)pyrazole —— C16H8Br2Cl2F3N3
3-cyano-4-(3-dibromomethylenecyclobutyl)-1-(2,6-dichloro-4-trifluoromethylphenyl)pyrazole
—— Crinecerfont hydrochloride 321839-75-2 C27H29Cl2FN2OS
Crinecerfont hydrochloride
—— N-cyclopentyl-3-[2-(cyclopentylamino)-4-pyrimidinyl]-2-[3-(cyclopropylmethoxy)phenyl]pyrazolo[1,5-a]pyridin-7-amine —— C31H36N6O
N-cyclopentyl-3-[2-(cyclopentylamino)-4-pyrimidinyl]-2-[3-(cyclopropylmethoxy)phenyl]pyrazolo[1,5-a]pyridin-7-amine
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(3-methylphenyl)methanone —— C24H27FN4O2
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(3-methylphenyl)methanone
—— (5Z)-5-[[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(Z)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C26H17N5O2S
(5Z)-5-[[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(Z)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-phenylmethanone —— C23H25FN4O2
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-phenylmethanone
—— N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-isopropyl-piperidin-4-yl)-ethane-1,2-diamine 332178-89-9 C25H34Cl2N6O
N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-isopropyl-piperidin-4-yl)-ethane-1,2-diamine
—— 5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-(5-trifluoromethylsulphenylthien-2-yl)pyrazole —— C16H6Cl2F6N4S2
5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-(5-trifluoromethylsulphenylthien-2-yl)pyrazole
—— methyl 2-butyl-5-chloro-3-[[2-oxo-9-(2H-tetrazol-5-yl)-5-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaenyl]methyl]imidazole-4-carboxylate —— C26H23ClN6O3
methyl 2-butyl-5-chloro-3-[[2-oxo-9-(2H-tetrazol-5-yl)-5-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaenyl]methyl]imidazole-4-carboxylate
—— 3-(3,4-dimethoxyphenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-4-amine —— C19H20N4O2S
3-(3,4-dimethoxyphenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-4-amine
—— N-[[1-[4-[5-(acetamidomethyl)-2-oxo-1,3-oxazolidin-3-yl]-2-fluorophenyl]imidazol-4-yl]methyl]quinoxaline-2-carboxamide —— C25H22FN7O4
N-[[1-[4-[5-(acetamidomethyl)-2-oxo-1,3-oxazolidin-3-yl]-2-fluorophenyl]imidazol-4-yl]methyl]quinoxaline-2-carboxamide
—— 1-[4,5-bis[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]-4-(1H-imidazol-5-yl)piperidine —— C25H21F6N5
1-[4,5-bis[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]-4-(1H-imidazol-5-yl)piperidine
—— N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine —— C19H24N6
N-[(2S)-2-methyl-3-pyrrolidin-1-ylpropyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine
—— 5-bromo-N-pyridin-3-yl-4-[4-[2-(pyridin-3-ylamino)-1,3-thiazol-4-yl]phenyl]-1,3-thiazol-2-amine —— C22H15BrN6S2
5-bromo-N-pyridin-3-yl-4-[4-[2-(pyridin-3-ylamino)-1,3-thiazol-4-yl]phenyl]-1,3-thiazol-2-amine
—— 2-[3,5-Dichloro-4-[2-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]propan-2-yl]phenyl]-3,5-dioxo-1,2,4-triazine-6-carboxylic acid —— C21H14Cl2FN5O5
2-[3,5-Dichloro-4-[2-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]propan-2-yl]phenyl]-3,5-dioxo-1,2,4-triazine-6-carboxylic acid
—— N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine —— C19H24N6
N-[(2R)-2-methyl-3-pyrrolidin-1-ylpropyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine
—— 5-(4-bromophenyl)-N-(2-thiazolyl)-2-(4-trifluoromethylphenyl)imidazole-4-carboxamide 313974-41-3 C20H12BrF3N4OS
5-(4-bromophenyl)-N-(2-thiazolyl)-2-(4-trifluoromethylphenyl)imidazole-4-carboxamide
—— 2-phenyl-4-[[4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,3-thiazole —— C23H25N7S
2-phenyl-4-[[4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,3-thiazole
—— 1-[(4R)-4-[5-[(4R)-3-(3,3-dimethyl-2-oxopentanoyl)-1,3-thiazolidin-4-yl]-1,3,4-oxadiazol-2-yl]-1,3-thiazolidin-3-yl]-3,3-dimethylpentane-1,2-dione —— C22H32N4O5S2
1-[(4R)-4-[5-[(4R)-3-(3,3-dimethyl-2-oxopentanoyl)-1,3-thiazolidin-4-yl]-1,3,4-oxadiazol-2-yl]-1,3-thiazolidin-3-yl]-3,3-dimethylpentane-1,2-dione
—— 2-phenyl-4-[[4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,3-thiazole —— C23H25N7S
2-phenyl-4-[[4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,3-thiazole
—— 1-(4-chlorophenyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide —— C18H16ClN3O2
1-(4-chlorophenyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide
—— 4-[[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]methyl]benzonitrile —— C24H26FN5O
4-[[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]methyl]benzonitrile
—— 2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide —— C21H22ClN3O2
2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide
—— 4-(2-methylsulfanylimidazol-1-yl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide —— C19H19N3O2S
4-(2-methylsulfanylimidazol-1-yl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide
—— N-cyclopropyl-2-[5-[2-(cyclopropylmethylamino)pyrimidin-4-yl]-4-(4-fluorophenyl)-1H-imidazol-2-yl]-5-methyl-1,3-dioxane-5-carboxamide —— C26H29FN6O3
N-cyclopropyl-2-[5-[2-(cyclopropylmethylamino)pyrimidin-4-yl]-4-(4-fluorophenyl)-1H-imidazol-2-yl]-5-methyl-1,3-dioxane-5-carboxamide
—— 1-(4-chlorophenyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide —— C18H16ClN3O2
1-(4-chlorophenyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide
—— N-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzamide —— C23H25FN4O2
N-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzamide
—— N-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzenesulfonamide —— C22H25FN4O3S
N-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzenesulfonamide
—— 2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide —— C21H22ClN3O2
2-[1-(4-chlorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide
—— 5-[[cyclopentyl-[(3,4-dimethyl-1,2-oxazol-5-yl)sulfamoyl]amino]methyl]-N,N-dimethyl-2-(1,3-oxazol-2-yl)benzamide —— C23H29N5O5S
5-[[cyclopentyl-[(3,4-dimethyl-1,2-oxazol-5-yl)sulfamoyl]amino]methyl]-N,N-dimethyl-2-(1,3-oxazol-2-yl)benzamide
—— 2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide —— C22H22F3N3O2
2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide
—— (3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpiperidine-3-carboxamide —— C23H25FN4O2
(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpiperidine-3-carboxamide
—— 2-pyrazol-1-yl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide —— C18H17N3O2
2-pyrazol-1-yl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide
—— N-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzenesulfonamide —— C22H25FN4O3S
N-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzenesulfonamide
—— (3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpiperidine-3-carboxamide —— C23H25FN4O2
(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-phenylpiperidine-3-carboxamide
—— (2,5-dimethylfuran-3-yl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H25FN4O3
(2,5-dimethylfuran-3-yl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 4-[[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]methyl]benzonitrile —— C24H26FN5O
4-[[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]methyl]benzonitrile
—— 6-Fluoro-2-[[3-[[4-(2-methylimidazo[4,5-c]pyridin-1-yl)phenoxy]methyl]phenoxy]methyl]quinoline —— C30H23FN4O2
6-Fluoro-2-[[3-[[4-(2-methylimidazo[4,5-c]pyridin-1-yl)phenoxy]methyl]phenoxy]methyl]quinoline
—— N-[3-(2,4-dimethyl-phenyl)-5-ethyl-2-methyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine 332179-22-3 C28H36N8
N-[3-(2,4-dimethyl-phenyl)-5-ethyl-2-methyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine
—— 2-pyrazol-1-yl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide —— C18H17N3O2
2-pyrazol-1-yl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide
—— 1-(4-bromophenyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide —— C18H16BrN3O2
1-(4-bromophenyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide