中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H41N5O6S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C33H28ClN5O2S |
|
—— |
(4R)-4-(4-fluorophenyl)-1-(3-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H33FN4O2S |
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—— |
2-[(4S)-1,4-bis(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2S)-butan-2-yl]acetamide |
—— |
C32H34N4O2S |
|
—— |
2-[(4S)-3-tert-butyl-1,4-bis(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C32H35N5O2S |
|
—— |
(4R)-4-(2-methylphenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O3S |
|
—— |
2-[(4R)-1,4-bis(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C35H31FN4O2S |
|
—— |
N-(3-methoxypropyl)-2-[(4R)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H34N4O3S |
|
—— |
2-[(4R)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C32H34N4O2S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4S)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H34N4O3S |
|
—— |
2-[(4R)-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C29H26F2N4O3S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4R)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H34N4O3S |
|
—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2S)-butan-2-yl]acetamide |
—— |
C30H36N4O4S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2R)-butan-2-yl]acetamide |
—— |
C31H29ClN4O4S |
|
—— |
2-[(4S)-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C32H31FN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C29H35FN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-methylphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C31H34N4O3S |
|
—— |
N-(furan-2-ylmethyl)-2-[(4R)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C33H30N4O3S |
|
—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide |
—— |
C33H25ClN4O4S |
|
—— |
2-[(4S)-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C32H25F2N5O2S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C30H28Cl2N4O2S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C30H37ClN4O2S |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4R)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H34N4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-methylphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C33H35FN4O2S |
|
—— |
2-[(4S)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C31H32N4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C31H40N4O6S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C32H33FN4O5S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C29H35FN4O3S |
|
—— |
2-[(4S)-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C32H25F2N5O2S |
|
—— |
2-[(4S)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O3S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C33H36N4O5S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C33H28ClN5O3S |
|
—— |
(4S)-4-(2-methylphenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O3S |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4R)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H34N4O2S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H35FN4O3S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C30H29ClN4O4S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H30ClN5O5S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C33H28ClN5O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C29H36FN5O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C32H40N4O3S |
|
—— |
2-[(4R)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O3S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C31H30N4O5S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
(4S)-4-(2-methylphenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O2S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(3-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H37N5O5S |
|
—— |
2-[[2-(4-chlorophenyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl]-1H-imidazo[4,5-b]pyrazine |
—— |
C20H15ClN6 |
|
—— |
N-cyclopropyl-2-[(4R)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C31H30N4O3S |
|
—— |
(2-butyl-benzofuran-3-yl)-[5-(4-methoxy-phenyl)-oxazol-2-yl]-methanol |
—— |
C23H23NO4 |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C32H27ClN4O3S |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4S)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C32H34N4O2S |
|