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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[(E)-(3-chloro-4,5-dimethoxyphenyl)methylideneamino]-3-(4-methylphenyl)-1H-1,2,4-triazole-5-thione —— C18H17ClN4O2S
4-[(E)-(3-chloro-4,5-dimethoxyphenyl)methylideneamino]-3-(4-methylphenyl)-1H-1,2,4-triazole-5-thione
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4,6-dimethylpyrimidin-2-amine —— C18H20FN5
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4,6-dimethylpyrimidin-2-amine
—— 3-(4-chlorophenyl)-5-[(1R)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C20H22ClN5O
3-(4-chlorophenyl)-5-[(1R)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(4-chlorophenyl)-5-[(1R)-1-[4-[[1-(difluoromethyl)imidazol-2-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H21ClF2N6O
3-(4-chlorophenyl)-5-[(1R)-1-[4-[[1-(difluoromethyl)imidazol-2-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— [3-(4-fluorophenyl)-1H-pyrazol-5-yl]-[(3R)-3-hydroxypiperidin-1-yl]methanone —— C15H16FN3O2
[3-(4-fluorophenyl)-1H-pyrazol-5-yl]-[(3R)-3-hydroxypiperidin-1-yl]methanone
—— (3S)-4-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-3-methylmorpholine —— C15H17F2N3O3
(3S)-4-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-3-methylmorpholine
—— (1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-methoxyphenyl)-N-methylethanamine —— C20H21F2N3O3
(1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-methoxyphenyl)-N-methylethanamine
—— (2R)-N-(2-cyanoethyl)-N-methyl-2-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propanamide —— C22H30N6O2
(2R)-N-(2-cyanoethyl)-N-methyl-2-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propanamide
—— 3-(4-chlorophenyl)-5-[(1S)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C20H22ClN5O
3-(4-chlorophenyl)-5-[(1S)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— N-[(E)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-methylfuran-3-carboxamide —— C17H14Cl2N4O2
N-[(E)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-methylfuran-3-carboxamide
—— 4-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione —— C15H14ClFN6S
4-[(E)-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione
—— 3-(4-chlorophenyl)-5-[(1S)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H21ClN4OS
3-(4-chlorophenyl)-5-[(1S)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(2-chlorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-5-carboxamide —— C17H16ClN3O2
3-(2-chlorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-5-carboxamide
—— 3-(4-chlorophenyl)-5-[(1S)-1-[4-[[1-(difluoromethyl)imidazol-2-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H21ClF2N6O
3-(4-chlorophenyl)-5-[(1S)-1-[4-[[1-(difluoromethyl)imidazol-2-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-2-(4-cyanophenoxy)acetamide —— C20H16ClN5O2
N-[(E)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-2-(4-cyanophenoxy)acetamide
—— (2S)-N-(2-cyanoethyl)-N-methyl-2-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propanamide —— C22H30N6O2
(2S)-N-(2-cyanoethyl)-N-methyl-2-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propanamide
—— 3-[2-(difluoromethoxy)phenyl]-5-[[(1R)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-1,2,4-oxadiazole —— C23H20F2N4O2
3-[2-(difluoromethoxy)phenyl]-5-[[(1R)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-1,2,4-oxadiazole
—— (2R)-N-(2-cyanoethyl)-N-methyl-2-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propanamide —— C22H30N6O2
(2R)-N-(2-cyanoethyl)-N-methyl-2-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propanamide
—— (1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-methoxyphenyl)-N-methylethanamine —— C20H21F2N3O3
(1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-methoxyphenyl)-N-methylethanamine
—— 3-[2-(difluoromethoxy)phenyl]-5-[[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-1,2,4-oxadiazole —— C23H20F2N4O2
3-[2-(difluoromethoxy)phenyl]-5-[[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-1,2,4-oxadiazole
—— 5-[[(2R)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C23H24N6O2
5-[[(2R)-2-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 3-(4-chlorophenyl)-5-[(1R)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H21ClN4OS
3-(4-chlorophenyl)-5-[(1R)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 4-[(E)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione —— C15H14Cl2N6S
4-[(E)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione
—— 6-[(1S)-1-[4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]ethyl]-2-N,2-N-dimethyl-1,3,5-triazine-2,4-diamine —— C20H26ClN9O
6-[(1S)-1-[4-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]ethyl]-2-N,2-N-dimethyl-1,3,5-triazine-2,4-diamine
—— 3-(2-chlorophenyl)-N-[(2R)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide —— C13H14ClN3O2
3-(2-chlorophenyl)-N-[(2R)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide
—— 4-chloro-5-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-phenylpyridazin-3-one —— C22H19ClFN5O
4-chloro-5-[[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-phenylpyridazin-3-one
—— 3-(2-chlorophenyl)-N-[(R)-(4-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-1H-pyrazole-5-carboxamide —— C22H20ClN5O2
3-(2-chlorophenyl)-N-[(R)-(4-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
—— [3-(2-chlorophenyl)-1H-pyrazol-5-yl]-[(3S)-3-hydroxypiperidin-1-yl]methanone —— C15H16ClN3O2
[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-[(3S)-3-hydroxypiperidin-1-yl]methanone
—— 3-(4-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]-1H-pyrazole-5-carboxamide —— C13H14FN3O2
3-(4-fluorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]-1H-pyrazole-5-carboxamide
—— N-[(E)-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]methylideneamino]cyclopropanecarboxamide —— C22H18N4O2
N-[(E)-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]methylideneamino]cyclopropanecarboxamide
—— (2R)-2-[4-[3-(2-chlorophenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl]-2-(4-methoxyphenyl)acetonitrile —— C23H22ClN5O2
(2R)-2-[4-[3-(2-chlorophenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl]-2-(4-methoxyphenyl)acetonitrile
—— N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-8-nitroisoquinolin-5-amine —— C21H18FN5O2
N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-8-nitroisoquinolin-5-amine
—— N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-3,4-dimethoxybenzamide —— C21H22N4O3
N-[(E)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-3,4-dimethoxybenzamide
—— 4-chloro-5-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-phenylpyridazin-3-one —— C22H19ClFN5O
4-chloro-5-[[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]amino]-2-phenylpyridazin-3-one
—— 3-(4-fluorophenyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-5-carboxamide —— C18H16FN3O2
3-(4-fluorophenyl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-1H-pyrazole-5-carboxamide
—— [3-(2-chlorophenyl)-1H-pyrazol-5-yl]-[(2S)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]methanone —— C22H22ClN3O3
[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-[(2S)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]methanone
—— 4-ethyl-2-[[(3S)-3-methylmorpholin-4-yl]methyl]-5-(3-methylphenyl)-1,2,4-triazole-3-thione —— C17H24N4OS
4-ethyl-2-[[(3S)-3-methylmorpholin-4-yl]methyl]-5-(3-methylphenyl)-1,2,4-triazole-3-thione
—— 3-(4-fluorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-1H-pyrazole-5-carboxamide —— C13H14FN3O2
3-(4-fluorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-1H-pyrazole-5-carboxamide
—— 3-(4-fluorophenyl)-N-[(2R)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide —— C13H14FN3O2
3-(4-fluorophenyl)-N-[(2R)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide
—— 3-(2-chlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]-1H-pyrazole-5-carboxamide —— C13H14ClN3O2
3-(2-chlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]-1H-pyrazole-5-carboxamide
—— methyl (3R)-3-[[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]amino]-3-thiophen-2-ylpropanoate —— C18H16FN3O3S
methyl (3R)-3-[[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]amino]-3-thiophen-2-ylpropanoate
—— [(2R)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]methanone —— C22H22FN3O3
[(2R)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]methanone
—— methyl (3R)-3-[[3-(2-chlorophenyl)-1H-pyrazole-5-carbonyl]amino]-3-(4-methoxyphenyl)propanoate —— C21H20ClN3O4
methyl (3R)-3-[[3-(2-chlorophenyl)-1H-pyrazole-5-carbonyl]amino]-3-(4-methoxyphenyl)propanoate
—— 3-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide —— C13H14ClN3O2
3-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide
—— 3-(4-fluorophenyl)-N-[(2S)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide —— C13H14FN3O2
3-(4-fluorophenyl)-N-[(2S)-2-hydroxypropyl]-1H-pyrazole-5-carboxamide
—— [3-(2-chlorophenyl)-1H-pyrazol-5-yl]-[(2R)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]methanone —— C22H22ClN3O3
[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-[(2R)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]methanone
—— methyl (3S)-3-[[3-(2-chlorophenyl)-1H-pyrazole-5-carbonyl]amino]-3-(4-methoxyphenyl)propanoate —— C21H20ClN3O4
methyl (3S)-3-[[3-(2-chlorophenyl)-1H-pyrazole-5-carbonyl]amino]-3-(4-methoxyphenyl)propanoate
—— 3-(4-fluorophenyl)-N-[(1S)-1-pyridin-4-ylethyl]-1H-pyrazole-5-carboxamide —— C17H15FN4O
3-(4-fluorophenyl)-N-[(1S)-1-pyridin-4-ylethyl]-1H-pyrazole-5-carboxamide
—— N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methoxypyrimidin-2-amine —— C17H18FN5O
N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-4-methoxypyrimidin-2-amine
—— [(2S)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]methanone —— C22H22FN3O3
[(2S)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]methanone