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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-propan-2-yl-3-[4-[[[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]carbamoylamino]methyl]phenyl]urea —— C22H27N7O2
1-propan-2-yl-3-[4-[[[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]carbamoylamino]methyl]phenyl]urea
—— (2R)-1-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol —— C21H32N4O3
(2R)-1-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol
—— 1-[(1R)-2-(dimethylamino)-1-phenylethyl]-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]urea —— C23H29N5O
1-[(1R)-2-(dimethylamino)-1-phenylethyl]-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]urea
—— 1-[[4-fluoro-2-(trifluoromethyl)phenyl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C19H17F4N5O
1-[[4-fluoro-2-(trifluoromethyl)phenyl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 1-[(1S)-1-(3-chlorophenyl)propyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C20H22ClN5O
1-[(1S)-1-(3-chlorophenyl)propyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— (1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methyl-1-(4-methylphenyl)ethanamine —— C20H21F2N3O2
(1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methyl-1-(4-methylphenyl)ethanamine
—— 1-[[6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C23H29N7O2
1-[[6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— (3R)-N-(cyclopropylmethyl)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidine-3-carboxamide —— C20H24F2N4O3
(3R)-N-(cyclopropylmethyl)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidine-3-carboxamide
—— 1-[(1R)-1-(3-chlorophenyl)propyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C20H22ClN5O
1-[(1R)-1-(3-chlorophenyl)propyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 1-[[4-(phenoxymethyl)phenyl]methyl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C25H25N5O2
1-[[4-(phenoxymethyl)phenyl]methyl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— N-[(E)-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylideneamino]thiophene-2-carboxamide —— C21H15ClN4OS
N-[(E)-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylideneamino]thiophene-2-carboxamide
—— 1-[(1R)-1-(3-chlorophenyl)propyl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C20H22ClN5O
1-[(1R)-1-(3-chlorophenyl)propyl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 3-(2-ethoxyphenyl)-4-[(E)-(4-methylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C18H18N4OS
3-(2-ethoxyphenyl)-4-[(E)-(4-methylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— (E)-1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine —— C14H13FN6
(E)-1-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine
—— (2R)-1-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol —— C21H32N4O3
(2R)-1-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol
—— 4-[(E)-[4-(dimethylamino)phenyl]methylideneamino]-3-(2-ethoxyphenyl)-1H-1,2,4-triazole-5-thione —— C19H21N5OS
4-[(E)-[4-(dimethylamino)phenyl]methylideneamino]-3-(2-ethoxyphenyl)-1H-1,2,4-triazole-5-thione
—— 3-(4-chlorophenyl)-5-[(1S)-1-[4-[[(3R)-oxolan-3-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H25ClN4O2
3-(4-chlorophenyl)-5-[(1S)-1-[4-[[(3R)-oxolan-3-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-3-(1,3,5-trimethylpyrazol-4-yl)-1H-pyrazole-5-carboxamide —— C20H22N8O
N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-3-(1,3,5-trimethylpyrazol-4-yl)-1H-pyrazole-5-carboxamide
—— 1-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-3-[2-[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]ethyl]urea —— C20H30N4O2S2
1-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-3-[2-[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]ethyl]urea
—— 3-[2-(difluoromethoxy)phenyl]-5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C19H17F2N3O2
3-[2-(difluoromethoxy)phenyl]-5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— [(2R,6R)-2,6-dimethylmorpholin-4-yl]-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone —— C23H31FN4O3
[(2R,6R)-2,6-dimethylmorpholin-4-yl]-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone
—— 3-(4-chlorophenyl)-5-[(1R)-1-[4-[[(3R)-oxolan-3-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C19H25ClN4O2
3-(4-chlorophenyl)-5-[(1R)-1-[4-[[(3R)-oxolan-3-yl]methyl]piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 4-[(E)-(4-chlorophenyl)methylideneamino]-3-(2-ethoxyphenyl)-1H-1,2,4-triazole-5-thione —— C17H15ClN4OS
4-[(E)-(4-chlorophenyl)methylideneamino]-3-(2-ethoxyphenyl)-1H-1,2,4-triazole-5-thione
—— (2S)-1-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol —— C21H32N4O3
(2S)-1-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol
—— 1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-pentylpiperidine-4-carboxamide —— C22H31FN4O2
1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-pentylpiperidine-4-carboxamide
—— (1R)-1-cyclohexyl-N,N-dimethyl-N'-[(4-pyrazol-1-ylphenyl)methyl]ethane-1,2-diamine —— C20H30N4
(1R)-1-cyclohexyl-N,N-dimethyl-N'-[(4-pyrazol-1-ylphenyl)methyl]ethane-1,2-diamine
—— (3S)-N-(cyclopropylmethyl)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidine-3-carboxamide —— C20H24F2N4O3
(3S)-N-(cyclopropylmethyl)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidine-3-carboxamide
—— 1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H24F2N4O3
1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 3-(4-methoxyphenyl)-5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C19H19N3O2
3-(4-methoxyphenyl)-5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C18H17N3O
5-[[(3S)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— [(2R,6S)-2,6-dimethylmorpholin-4-yl]-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone —— C23H31FN4O3
[(2R,6S)-2,6-dimethylmorpholin-4-yl]-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone
—— ethyl N-[(3R)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-3-yl]carbamate —— C18H22F2N4O4
ethyl N-[(3R)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-3-yl]carbamate
—— 1-[(2S)-2-(dimethylamino)-3-phenylpropyl]-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]urea —— C24H31N5O
1-[(2S)-2-(dimethylamino)-3-phenylpropyl]-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]urea
—— (1R)-1-cyclohexyl-N'-[(4-imidazol-1-ylphenyl)methyl]-N,N-dimethylethane-1,2-diamine —— C20H30N4
(1R)-1-cyclohexyl-N'-[(4-imidazol-1-ylphenyl)methyl]-N,N-dimethylethane-1,2-diamine
—— 1-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-3-[2-[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]ethyl]urea —— C20H30N4O2S2
1-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-3-[2-[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]ethyl]urea
—— 3-cyclopentyl-1-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propan-1-one —— C23H31FN4O2
3-cyclopentyl-1-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propan-1-one
—— 1-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H24F2N4O3
1-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-pentylpiperidine-4-carboxamide —— C22H31FN4O2
1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-pentylpiperidine-4-carboxamide
—— 1-[[(2S)-4-benzylmorpholin-2-yl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C23H28N6O2
1-[[(2S)-4-benzylmorpholin-2-yl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 3-(4-methoxyphenyl)-5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C19H19N3O2
3-(4-methoxyphenyl)-5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— 1-[[4-(phenoxymethyl)phenyl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C25H25N5O2
1-[[4-(phenoxymethyl)phenyl]methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— 3-[2-(difluoromethoxy)phenyl]-5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C19H17F2N3O2
3-[2-(difluoromethoxy)phenyl]-5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— 3-cyclopentyl-1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propan-1-one —— C23H31FN4O2
3-cyclopentyl-1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]propan-1-one
—— 2-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-1-pyrrolidin-1-ylethanone —— C22H29FN4O2
2-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-1-pyrrolidin-1-ylethanone
—— 1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(3-propan-2-yloxypropyl)piperidine-4-carboxamide —— C23H33FN4O3
1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(3-propan-2-yloxypropyl)piperidine-4-carboxamide
—— N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-3-(1,3,5-trimethylpyrazol-4-yl)-1H-pyrazole-5-carboxamide —— C21H24N8O
N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-3-(1,3,5-trimethylpyrazol-4-yl)-1H-pyrazole-5-carboxamide
—— [(2R,6R)-2,6-dimethylmorpholin-4-yl]-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone —— C23H31FN4O3
[(2R,6R)-2,6-dimethylmorpholin-4-yl]-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[(3S)-3-methylpiperidin-1-yl]ethyl]-1,2,4-oxadiazole —— C17H22FN3O
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[(3S)-3-methylpiperidin-1-yl]ethyl]-1,2,4-oxadiazole
—— 5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C18H17N3O
5-[[(3R)-3-methyl-2,3-dihydroindol-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— N-[(2S)-butan-2-yl]-3-[[[5-(4-methylphenyl)-1H-pyrazol-4-yl]methylamino]methyl]benzamide —— C23H28N4O
N-[(2S)-butan-2-yl]-3-[[[5-(4-methylphenyl)-1H-pyrazol-4-yl]methylamino]methyl]benzamide