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中文名称 英文名称 CAS号 化学式 结构式图片
—— 11-[(3S)-1-(1H-imidazol-5-ylsulfonyl)piperidine-3-carbonyl]-5-phenyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H25N7O4S
11-[(3S)-1-(1H-imidazol-5-ylsulfonyl)piperidine-3-carbonyl]-5-phenyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-thiophen-3-ylethanone —— C18H17N3O2S
1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-thiophen-3-ylethanone
—— 4-[[(2R)-oxolan-2-yl]methyl]-3-undecyl-1H-1,2,4-triazole-5-thione —— C18H33N3OS
4-[[(2R)-oxolan-2-yl]methyl]-3-undecyl-1H-1,2,4-triazole-5-thione
—— 11-[(3R)-1-(1H-imidazol-5-ylsulfonyl)piperidine-3-carbonyl]-5-phenyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H25N7O4S
11-[(3R)-1-(1H-imidazol-5-ylsulfonyl)piperidine-3-carbonyl]-5-phenyl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (3-phenyl-1H-pyrazol-5-yl)-[(3S)-3-(pyridin-3-ylamino)pyrrolidin-1-yl]methanone —— C19H19N5O
(3-phenyl-1H-pyrazol-5-yl)-[(3S)-3-(pyridin-3-ylamino)pyrrolidin-1-yl]methanone
—— ethyl 5-(4-bromophenyl)-1-[4-[[(2R)-4-phenylbutan-2-yl]carbamoyl]phenyl]pyrazole-3-carboxylate —— C29H28BrN3O3
ethyl 5-(4-bromophenyl)-1-[4-[[(2R)-4-phenylbutan-2-yl]carbamoyl]phenyl]pyrazole-3-carboxylate
—— 5-[(3R)-1-cyclopropylsulfonylpyrrolidin-3-yl]-3-phenyl-1,2,4-oxadiazole —— C15H17N3O3S
5-[(3R)-1-cyclopropylsulfonylpyrrolidin-3-yl]-3-phenyl-1,2,4-oxadiazole
—— 1-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-thiophen-2-ylethanone —— C18H17N3O2S
1-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-thiophen-2-ylethanone
—— ethyl 5-(4-bromophenyl)-1-[4-[[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]methylcarbamoyl]phenyl]pyrazole-3-carboxylate —— C25H26BrN3O5
ethyl 5-(4-bromophenyl)-1-[4-[[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]methylcarbamoyl]phenyl]pyrazole-3-carboxylate
—— (2S)-1-[(1-ethylpyrazol-4-yl)methyl]-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine —— C19H24N6
(2S)-1-[(1-ethylpyrazol-4-yl)methyl]-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine
—— furan-2-yl-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C17H15N3O3
furan-2-yl-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— 12-[(3S)-1-(1H-imidazol-5-ylsulfonyl)piperidine-3-carbonyl]-5-phenyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C24H25N7O4S
12-[(3S)-1-(1H-imidazol-5-ylsulfonyl)piperidine-3-carbonyl]-5-phenyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (3R)-N-(2-methoxyethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide —— C16H20N4O3
(3R)-N-(2-methoxyethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
—— 1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-pyridin-3-ylethanone —— C19H18N4O2
1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-pyridin-3-ylethanone
—— 1-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-thiophen-3-ylethanone —— C18H17N3O2S
1-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-thiophen-3-ylethanone
—— (5-methylthiophen-2-yl)-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C18H17N3O2S
(5-methylthiophen-2-yl)-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— [(2R)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]-thiophen-3-ylmethanone —— C18H18N4OS
[(2R)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]-thiophen-3-ylmethanone
—— (2R)-N-tert-butyl-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carboxamide —— C18H25N5O
(2R)-N-tert-butyl-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carboxamide
—— furan-3-yl-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C17H15N3O3
furan-3-yl-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— ethyl 5-(4-bromophenyl)-1-[4-[[(2R)-5-(diethylamino)pentan-2-yl]carbamoyl]phenyl]pyrazole-3-carboxylate —— C28H35BrN4O3
ethyl 5-(4-bromophenyl)-1-[4-[[(2R)-5-(diethylamino)pentan-2-yl]carbamoyl]phenyl]pyrazole-3-carboxylate
—— 2-(3-fluorophenyl)-1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone —— C20H18FN3O2
2-(3-fluorophenyl)-1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone
—— (2S)-N-(2-methylpropyl)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carboxamide —— C18H25N5O
(2S)-N-(2-methylpropyl)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carboxamide
—— 3-nonyl-4-[[(2R)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione —— C16H29N3OS
3-nonyl-4-[[(2R)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione
—— 4-[[(2S)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methyl]pyridine —— C19H21N5
4-[[(2S)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methyl]pyridine
—— [(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C18H16N4O2
[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— (2R)-1-methylsulfonyl-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine —— C14H18N4O2S
(2R)-1-methylsulfonyl-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine
—— 5-(4-methoxyphenyl)-11-[(2S)-2-methyl-3-piperidin-1-ylpropanoyl]-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C25H31N5O3
5-(4-methoxyphenyl)-11-[(2S)-2-methyl-3-piperidin-1-ylpropanoyl]-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 4-methyl-5-[[(2R)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methyl]-1,3-thiazole —— C18H21N5S
4-methyl-5-[[(2R)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methyl]-1,3-thiazole
—— (2R)-1-(furan-2-ylmethyl)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine —— C18H20N4O
(2R)-1-(furan-2-ylmethyl)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine
—— 3-octyl-4-[[(2R)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione —— C15H27N3OS
3-octyl-4-[[(2R)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione
—— 12-[(3R)-1-(3-chloro-4-fluorophenyl)-5-oxopyrrolidine-3-carbonyl]-5-phenyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C26H21ClFN5O3
12-[(3R)-1-(3-chloro-4-fluorophenyl)-5-oxopyrrolidine-3-carbonyl]-5-phenyl-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (3S)-N-(furan-2-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide —— C18H18N4O3
(3S)-N-(furan-2-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
—— 2-(2-fluorophenyl)-1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone —— C20H18FN3O2
2-(2-fluorophenyl)-1-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethanone
—— 3-octyl-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione —— C15H27N3OS
3-octyl-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione
—— ethyl 5-(4-bromophenyl)-1-[4-[[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]methylcarbamoyl]phenyl]pyrazole-3-carboxylate —— C25H26BrN3O5
ethyl 5-(4-bromophenyl)-1-[4-[[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]methylcarbamoyl]phenyl]pyrazole-3-carboxylate
—— 3-nonyl-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione —— C16H29N3OS
3-nonyl-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione
—— ethyl 5-(4-bromophenyl)-1-[4-[[(2S)-5-(diethylamino)pentan-2-yl]carbamoyl]phenyl]pyrazole-3-carboxylate —— C28H35BrN4O3
ethyl 5-(4-bromophenyl)-1-[4-[[(2S)-5-(diethylamino)pentan-2-yl]carbamoyl]phenyl]pyrazole-3-carboxylate
—— (2-methylpyrazol-3-yl)-[(2S)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C18H20N6O
(2-methylpyrazol-3-yl)-[(2S)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— 3-(2,4-difluorophenyl)-5-thiophen-2-yl-1H-pyrazole —— C13H8F2N2S
3-(2,4-difluorophenyl)-5-thiophen-2-yl-1H-pyrazole
—— (2-fluorophenyl)-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C19H16FN3O2
(2-fluorophenyl)-[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (3R)-N-cyclopentyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide —— C18H22N4O2
(3R)-N-cyclopentyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
—— (3R)-N-benzyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide —— C20H20N4O2
(3R)-N-benzyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
—— 4-[[(2S)-oxolan-2-yl]methyl]-3-undecyl-1H-1,2,4-triazole-5-thione —— C18H33N3OS
4-[[(2S)-oxolan-2-yl]methyl]-3-undecyl-1H-1,2,4-triazole-5-thione
—— (2S)-N-tert-butyl-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carboxamide —— C18H25N5O
(2S)-N-tert-butyl-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine-1-carboxamide
—— (2R)-1-[(1-ethylpyrazol-4-yl)methyl]-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine —— C19H24N6
(2R)-1-[(1-ethylpyrazol-4-yl)methyl]-2-(4-phenyl-1,2,4-triazol-3-yl)piperidine
—— [(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C18H16N4O2
[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— furan-3-yl-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C17H15N3O3
furan-3-yl-[(3S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (5-methyl-1H-pyrazol-3-yl)-[(2S)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C18H20N6O
(5-methyl-1H-pyrazol-3-yl)-[(2S)-2-(4-phenyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— [(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-pyridin-4-ylmethanone —— C18H16N4O2
[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-pyridin-4-ylmethanone
—— 3-decyl-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione —— C17H31N3OS
3-decyl-4-[[(2S)-oxolan-2-yl]methyl]-1H-1,2,4-triazole-5-thione