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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-phenyl-1,3-oxazole —— C19H22N4O
4-[[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-phenyl-1,3-oxazole
—— N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-3-phenyl-1H-pyrazole-5-carboxamide —— C16H20N4O4S
N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-3-phenyl-1H-pyrazole-5-carboxamide
—— 4-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-phenyl-1,3-oxazole —— C19H22N4O
4-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-2-phenyl-1,3-oxazole
—— 3-[2,2-dimethyl-3-oxo-3-(azabicyclo[2.2.1]heptan-7-yl)propyl]-4-[1S-methyl-2-(N-isopropoxycarbonyl-3-pyrid-4-yl-pyrrolidin-1-ylcarboximidamido)ethyl]-5-(3,5-dimethylphenyl)-1H-pyrazole 667466-19-5 C39H53N7O4
3-[2,2-dimethyl-3-oxo-3-(azabicyclo[2.2.1]heptan-7-yl)propyl]-4-[1S-methyl-2-(N-isopropoxycarbonyl-3-pyrid-4-yl-pyrrolidin-1-ylcarboximidamido)ethyl]-5-(3,5-dimethylphenyl)-1H-pyrazole
—— 2-[Bis[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid —— C40H39N3O6
2-[Bis[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid
—— N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-3-phenyl-1H-pyrazole-5-carboxamide —— C16H20N4O4S
N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]-3-phenyl-1H-pyrazole-5-carboxamide
—— thuggacin A —— C35H53NO7S
thuggacin A
—— 4-[2-[[4-[(E)-N-[[2-(4-bromophenyl)-1,3-oxazol-4-yl]methoxy]-C-methylcarbonimidoyl]-3-methylphenoxy]methyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one —— C30H28BrN5O5
4-[2-[[4-[(E)-N-[[2-(4-bromophenyl)-1,3-oxazol-4-yl]methoxy]-C-methylcarbonimidoyl]-3-methylphenoxy]methyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one
—— 4-[5-(4-Methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide;2-[4-(2-methylpropyl)phenyl]propanoic acid —— C30H32F3N3O4S
4-[5-(4-Methylphenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzenesulfonamide;2-[4-(2-methylpropyl)phenyl]propanoic acid
—— (2S)-2-(3-methyl-1,2-oxazol-5-yl)-N-(2-phenyl-5-propan-2-ylpyrazol-3-yl)pyrrolidine-1-carboxamide —— C21H25N5O2
(2S)-2-(3-methyl-1,2-oxazol-5-yl)-N-(2-phenyl-5-propan-2-ylpyrazol-3-yl)pyrrolidine-1-carboxamide
—— 2-[[(3S)-3-(methylsulfonylmethyl)piperidin-1-yl]methyl]-4-phenyl-1,3-thiazole —— C17H22N2O2S2
2-[[(3S)-3-(methylsulfonylmethyl)piperidin-1-yl]methyl]-4-phenyl-1,3-thiazole
—— 1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]urea —— C19H24N6O
1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]urea
—— 2-[[(3R)-3-(methylsulfonylmethyl)piperidin-1-yl]methyl]-4-phenyl-1,3-thiazole —— C17H22N2O2S2
2-[[(3R)-3-(methylsulfonylmethyl)piperidin-1-yl]methyl]-4-phenyl-1,3-thiazole
—— 1-[3-[5-[(3R)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]imidazolidin-2-one —— C15H17N5O2
1-[3-[5-[(3R)-oxolan-3-yl]-1H-1,2,4-triazol-3-yl]phenyl]imidazolidin-2-one
—— 1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]urea —— C19H24N6O
1-(1-ethyl-3,5-dimethylpyrazol-4-yl)-3-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]urea
—— (2R)-2-(3-methyl-1,2-oxazol-5-yl)-N-(2-phenyl-5-propan-2-ylpyrazol-3-yl)pyrrolidine-1-carboxamide —— C21H25N5O2
(2R)-2-(3-methyl-1,2-oxazol-5-yl)-N-(2-phenyl-5-propan-2-ylpyrazol-3-yl)pyrrolidine-1-carboxamide
—— 1,3-dimethyl-4-[(Z)-2-nitroethenyl]pyrazole —— C7H9N3O2
1,3-dimethyl-4-[(Z)-2-nitroethenyl]pyrazole
—— (2S)-4-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]morpholine-2-carboxamide —— C17H22N4O2
(2S)-4-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]morpholine-2-carboxamide
—— 1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]urea —— C16H19FN8O
1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]urea
—— (2R)-4-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]morpholine-2-carboxamide —— C17H22N4O2
(2R)-4-[(3,5-dimethyl-2-pyrazol-1-ylphenyl)methyl]morpholine-2-carboxamide
—— 3-[[3-Methyl-2-(phenylcarbamoyloxy)butanoyl]amino]-4-oxo-5-[2-phenyl-5-(trifluoromethyl)pyrazol-3-yl]oxypentanoic acid —— C27H27F3N4O7
3-[[3-Methyl-2-(phenylcarbamoyloxy)butanoyl]amino]-4-oxo-5-[2-phenyl-5-(trifluoromethyl)pyrazol-3-yl]oxypentanoic acid
—— 4-[[5-[4-[[6-(Butoxycarbonylamino)indol-1-yl]methyl]-3-methoxyphenyl]tetrazol-2-yl]methyl]benzoic acid —— C30H30N6O5
4-[[5-[4-[[6-(Butoxycarbonylamino)indol-1-yl]methyl]-3-methoxyphenyl]tetrazol-2-yl]methyl]benzoic acid
—— 1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]urea —— C16H19FN8O
1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]urea
—— (3E)-3-[[(3S,3aR)-2-phenyl-3a,4-dihydro-3H-pyrazolo[1,5-a]benzimidazol-3-yl]methylidene]-2-phenylpyrazolo[1,5-a]benzimidazole —— C31H22N6
(3E)-3-[[(3S,3aR)-2-phenyl-3a,4-dihydro-3H-pyrazolo[1,5-a]benzimidazol-3-yl]methylidene]-2-phenylpyrazolo[1,5-a]benzimidazole
—— (3E)-3-[[(3R,3aR)-2-phenyl-3a,4-dihydro-3H-pyrazolo[1,5-a]benzimidazol-3-yl]methylidene]-2-phenylpyrazolo[1,5-a]benzimidazole —— C31H22N6
(3E)-3-[[(3R,3aR)-2-phenyl-3a,4-dihydro-3H-pyrazolo[1,5-a]benzimidazol-3-yl]methylidene]-2-phenylpyrazolo[1,5-a]benzimidazole
—— 1-benzyl-N-[(1S)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-4-carboxamide —— C19H23N5O2
1-benzyl-N-[(1S)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-4-carboxamide
—— 2-[bis(2-cyanoethyl)amino]ethyl N-[[3-[[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]carbamoylamino]phenyl]methyl]carbamate —— C27H29N7O5
2-[bis(2-cyanoethyl)amino]ethyl N-[[3-[[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]carbamoylamino]phenyl]methyl]carbamate
—— N'-{3-[(1,5-Diphenyl-1H-1,2,4-triazol-3-yl)amino]benzoyl}-4-methoxybenzenesulphonohydrazide 301547-66-0 C28H24N6O4S
N'-{3-[(1,5-Diphenyl-1H-1,2,4-triazol-3-yl)amino]benzoyl}-4-methoxybenzenesulphonohydrazide
—— N-[(2S)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide —— C18H20N4O2
N-[(2S)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
—— 1-[(2R)-2-thiophen-2-ylazetidin-1-yl]-2-(3,4,5-trimethylpyrazol-1-yl)ethanone —— C15H19N3OS
1-[(2R)-2-thiophen-2-ylazetidin-1-yl]-2-(3,4,5-trimethylpyrazol-1-yl)ethanone
—— N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazol[1,5-a]pyrimidin-7-yl]-N'-(2-trifluoromethyl-cyclohexyl)-ethane-1,2-diamine 332178-60-6 C24H28Cl2F3N5O
N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazol[1,5-a]pyrimidin-7-yl]-N'-(2-trifluoromethyl-cyclohexyl)-ethane-1,2-diamine
—— 5-(4-chlorophenyl)-2-(4-{2-[2-(2-methoxyethoxy)ethoxy]ethoxy}phenyl)-N-(2-thiazolyl)imidazole-4-carboxamide 313974-49-1 C26H27ClN4O5S
5-(4-chlorophenyl)-2-(4-{2-[2-(2-methoxyethoxy)ethoxy]ethoxy}phenyl)-N-(2-thiazolyl)imidazole-4-carboxamide
—— N-[(2S)-1-(3,4-dihydro-1H-isoquinolin-2-yl)propan-2-yl]-2-[4-(5-methyltetrazol-1-yl)phenyl]acetamide —— C22H26N6O
N-[(2S)-1-(3,4-dihydro-1H-isoquinolin-2-yl)propan-2-yl]-2-[4-(5-methyltetrazol-1-yl)phenyl]acetamide
—— N-[(2R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)propan-2-yl]-2-[4-(5-methyltetrazol-1-yl)phenyl]acetamide —— C22H26N6O
N-[(2R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)propan-2-yl]-2-[4-(5-methyltetrazol-1-yl)phenyl]acetamide
—— 1-[(2S)-2-thiophen-2-ylazetidin-1-yl]-2-(3,4,5-trimethylpyrazol-1-yl)ethanone —— C15H19N3OS
1-[(2S)-2-thiophen-2-ylazetidin-1-yl]-2-(3,4,5-trimethylpyrazol-1-yl)ethanone
—— 1-benzyl-N-[(1R)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-4-carboxamide —— C19H23N5O2
1-benzyl-N-[(1R)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-4-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide —— C18H20N4O2
N-[(2R)-2-(dimethylamino)-2-(furan-2-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
—— (2Z,5S,9S,12R,13S,14S)-9,13-dihydroxy-2,10,10,12,14-pentamethyl-5-[(E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-6-oxabicyclo[13.3.1]nonadeca-1(18),2,15(19),16-tetraene-7,11-dione —— C30H39NO5S
(2Z,5S,9S,12R,13S,14S)-9,13-dihydroxy-2,10,10,12,14-pentamethyl-5-[(E)-1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-6-oxabicyclo[13.3.1]nonadeca-1(18),2,15(19),16-tetraene-7,11-dione
—— (2R)-2-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl-phenylmethoxycarbonylamino]propanoic acid —— C30H30N2O6
(2R)-2-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl-phenylmethoxycarbonylamino]propanoic acid
—— 3,5-Dichloro-4-[2,5-dimethyl-7-[2-[(1-phenylpyrrolidin-3-yl)amino]ethylamino]pyrazolo[1,5-a]pyrimidin-3-yl]phenol —— C26H28Cl2N6O
3,5-Dichloro-4-[2,5-dimethyl-7-[2-[(1-phenylpyrrolidin-3-yl)amino]ethylamino]pyrazolo[1,5-a]pyrimidin-3-yl]phenol
—— (2S)-2-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl-phenylmethoxycarbonylamino]propanoic acid —— C30H30N2O6
(2S)-2-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl-phenylmethoxycarbonylamino]propanoic acid
—— N-[[7-chloro-1-(2,4-dichlorophenyl)-4,5-dihydrobenzo[g]indazol-3-yl]methyl]-8-azaspiro[4.5]decan-8-amine —— C27H29Cl3N4
N-[[7-chloro-1-(2,4-dichlorophenyl)-4,5-dihydrobenzo[g]indazol-3-yl]methyl]-8-azaspiro[4.5]decan-8-amine
—— 5-[[Cyclopentyl-[[4-(1,3-oxazol-2-yl)-3-[(2-oxopyrrolidin-1-yl)methyl]phenyl]methyl]sulfamoyl]amino]-3,4-dimethyl-1,2-oxazole —— C25H31N5O5S
5-[[Cyclopentyl-[[4-(1,3-oxazol-2-yl)-3-[(2-oxopyrrolidin-1-yl)methyl]phenyl]methyl]sulfamoyl]amino]-3,4-dimethyl-1,2-oxazole
—— N-[3-(2,6-dimethyl-phenyl)-2-methyl-5-propyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine 332179-19-8 C29H38N8
N-[3-(2,6-dimethyl-phenyl)-2-methyl-5-propyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine
—— N-Cyclopentyl-3-[2-(cyclopentylamino)pyrimidin-4-yl]-2-(4-fluorophenyl)-8-methylimidazo[1,2-a]pyridin-6-amine —— C28H31FN6
N-Cyclopentyl-3-[2-(cyclopentylamino)pyrimidin-4-yl]-2-(4-fluorophenyl)-8-methylimidazo[1,2-a]pyridin-6-amine
—— 2-(3-cyclobutyloxypyridin-2-ylmethoxy)-3,7-bis(2-fluorophenyl)pyrazolo[1,5-d][1,2,4]triazine 265643-34-3 C27H21F2N5O2
2-(3-cyclobutyloxypyridin-2-ylmethoxy)-3,7-bis(2-fluorophenyl)pyrazolo[1,5-d][1,2,4]triazine
—— N-[3-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-1-phenylpropyl]cyclobutanecarboxamide —— C28H34N4O3
N-[3-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-1-phenylpropyl]cyclobutanecarboxamide
—— (4Z)-4-[[2-(3,4-dimethylphenyl)-5-ethoxy-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid —— C23H22N4O6S
(4Z)-4-[[2-(3,4-dimethylphenyl)-5-ethoxy-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid
—— N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo [1,5-a]pyrimidin-7-yl]-N'-(2-pyridin4-yl-ethyl)-ethane-1,2-diamine 332179-31-4 C24H26Cl2N6O
N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo [1,5-a]pyrimidin-7-yl]-N'-(2-pyridin4-yl-ethyl)-ethane-1,2-diamine
—— N-[3-(2,4-dimethyl-phenyl)-2-methyl-5-propyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine 332179-23-4 C29H38N8
N-[3-(2,4-dimethyl-phenyl)-2-methyl-5-propyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine