中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C31H31FN4O4S |
|
—— |
(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H32F2N4O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C29H31N5O2S2 |
|
—— |
N,3-dimethyl-5-nitro-N-[(2S)-2-phenylpropyl]imidazole-4-sulfonamide |
—— |
C14H18N4O4S |
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—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C30H33FN4O5S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C34H36N4O6S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C33H37N5O4S |
|
—— |
2-[(4R)-3-tert-butyl-4-(4-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C32H32F2N4O2S |
|
—— |
2-[(4R)-1-(2-methylphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C31H27N5O2S2 |
|
—— |
2-[(4R)-1-(4-fluorophenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C28H27FN4O2S2 |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C33H33FN4O5S |
|
—— |
2-[(4R)-3-tert-butyl-1-(3-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C28H34N4O3S2 |
|
—— |
2-[(4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C31H28ClFN4O3S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C31H28ClFN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(4-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C29H36FN5O2S |
|
—— |
2-[(4R)-4-(3-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C29H26ClFN4O2S |
|
—— |
2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C30H30N4O4S2 |
|
—— |
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C34H32N4O6S |
|
—— |
N-[2-(2,3-dimethylphenyl)-5-methylimidazol-1-yl]-3-methoxy-2-methylbenzamide |
—— |
C21H23N3O2 |
|
—— |
2-[(4S)-1,4-bis(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C33H25F3N4O2S |
|
—— |
2-[(4R)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C30H29FN4O3S |
|
—— |
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C34H36N4O6S |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C31H31FN4O5S |
|
—— |
2-[(4S)-3-tert-butyl-4-(4-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C32H32F2N4O2S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C31H31ClN4O4S |
|
—— |
2-[(4S)-1-(2-methylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C31H27N5O2S2 |
|
—— |
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C31H24Cl2N4O3S |
|
—— |
(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H32F2N4O2S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C31H37FN4O3S |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C33H37N5O4S |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C32H34N4O4S |
|
—— |
2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C32H40N4O5S |
|
—— |
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C34H30FN5O4S |
|
—— |
(4S)-3-tert-butyl-4-(3,4-dimethoxyphenyl)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O5S |
|
—— |
2-[(4R)-4-(3-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C29H26ClFN4O3S |
|
—— |
2-[(4S)-3-tert-butyl-1-(4-fluorophenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C30H31FN4O3S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C29H24Cl2N4O2S |
|
—— |
(4R)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C30H38N4O5S |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C32H25ClFN5O2S |
|
—— |
2-(4-ethoxyphenyl)-7,8-dimethyl-5H-imidazo[1,5-a]quinoxaline-1,3-dione |
—— |
C20H19N3O3 |
|
—— |
2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C32H27FN4O3S |
|
—— |
2-[(4S)-1-(4-fluorophenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C28H27FN4O2S2 |
|
—— |
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C31H24ClFN4O3S |
|
—— |
2-[(4R)-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C29H26F2N4O3S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C34H36N4O6S |
|
—— |
2-[(4R)-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C32H25F2N5O2S |
|
—— |
2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C32H25ClFN5O2S |
|
—— |
(4S)-4-(3-chlorophenyl)-1-(4-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C30H26ClFN4O2S |
|
—— |
[4-(1H-benzo[4,5]thieno[3,2-c]pyrazol-3-yl)benzyl]-pyridin-3-yl-amine |
—— |
C21H16N4S |
|