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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[4-phenyl-5-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-3-yl]morpholine —— C21H21F3N4OS
4-[4-phenyl-5-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-3-yl]morpholine
—— 1-(3-fluorophenyl)-3-[[(3S)-1-[1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carbonyl]piperidin-3-yl]methyl]urea —— C27H32FN5O2
1-(3-fluorophenyl)-3-[[(3S)-1-[1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carbonyl]piperidin-3-yl]methyl]urea
—— 1-(3-fluorophenyl)-3-[[(3S)-1-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperidin-3-yl]methyl]urea —— C23H23F2N5O2
1-(3-fluorophenyl)-3-[[(3S)-1-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperidin-3-yl]methyl]urea
—— N-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfinyl)pyrazol-3-yl]-N'-methylmethanimidamide —— C14H7Cl2F6N5OS
N-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfinyl)pyrazol-3-yl]-N'-methylmethanimidamide
—— 1-[[(3S)-1-[2-[1-(2,3-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea —— C26H30FN5O2S
1-[[(3S)-1-[2-[1-(2,3-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea
—— 1-[[(3S)-1-[2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea —— C26H30FN5O2S
1-[[(3S)-1-[2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea
—— 1-(3-fluorophenyl)-3-[[(3R)-1-[2-[1-(2-methylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]urea —— C25H28FN5O2S
1-(3-fluorophenyl)-3-[[(3R)-1-[2-[1-(2-methylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]urea
—— 3-[4-(difluoromethoxy)-3-methoxyphenyl]-5-[[(2R)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C20H18F2N4O5
3-[4-(difluoromethoxy)-3-methoxyphenyl]-5-[[(2R)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— N-benzyl-2-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]acetamide —— C24H29N3O3S
N-benzyl-2-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]acetamide
—— methyl (3S)-3-[(3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-(4-methylsulfanylphenyl)propanoate —— C22H23N3O3S
methyl (3S)-3-[(3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-(4-methylsulfanylphenyl)propanoate
—— N-benzyl-1-(4-fluorophenyl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]triazole-4-carboxamide —— C23H26FN5O2
N-benzyl-1-(4-fluorophenyl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]triazole-4-carboxamide
—— 3-(4-methoxyphenyl)-5-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-4-amine —— C18H17F3N4OS
3-(4-methoxyphenyl)-5-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-4-amine
—— 1-[[(3R)-1-[5-(4-chlorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea —— C23H23ClFN5O2
1-[[(3R)-1-[5-(4-chlorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea
—— 3-(2,4-dimethoxyphenyl)-5-[[(2S)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C20H20N4O5
3-(2,4-dimethoxyphenyl)-5-[[(2S)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— N-benzyl-2-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]acetamide —— C24H29N3O3S
N-benzyl-2-(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]acetamide
—— N-benzyl-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)acetamide —— C23H27N5O2S
N-benzyl-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)acetamide
—— 1-(3-fluorophenyl)-3-[[(3R)-1-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperidin-3-yl]methyl]urea —— C23H23F2N5O2
1-(3-fluorophenyl)-3-[[(3R)-1-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperidin-3-yl]methyl]urea
—— 3-(4-methoxyphenyl)-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-4-amine —— C18H17F3N4OS
3-(4-methoxyphenyl)-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-4-amine
—— 3-(2-methoxyphenyl)-5-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-4-amine —— C18H17F3N4OS
3-(2-methoxyphenyl)-5-[(1R)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-4-amine
—— (3R)-3-acetyl-N-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C20H18N4O4
(3R)-3-acetyl-N-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— 3-(2-methoxyphenyl)-4-prop-2-enyl-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazole —— C21H20F3N3OS
3-(2-methoxyphenyl)-4-prop-2-enyl-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazole
—— 1-(3-fluorophenyl)-3-[[(3S)-1-[1-(4-fluorophenyl)pyrazole-3-carbonyl]piperidin-3-yl]methyl]urea —— C23H23F2N5O2
1-(3-fluorophenyl)-3-[[(3S)-1-[1-(4-fluorophenyl)pyrazole-3-carbonyl]piperidin-3-yl]methyl]urea
—— N-benzyl-3-methyl-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-1-phenylpyrazole-4-carboxamide —— C25H30N4O2
N-benzyl-3-methyl-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-1-phenylpyrazole-4-carboxamide
—— 3-[4-amino-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide —— C21H24F3N5O2S2
3-[4-amino-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide
—— 5-methoxy-2-methyl-4-[2-[[3-methyl-4-[(E)-C-methyl-N-(thiophen-3-ylmethoxy)carbonimidoyl]phenoxy]methyl]phenyl]-1,2,4-triazol-3-one —— C25H26N4O4S
5-methoxy-2-methyl-4-[2-[[3-methyl-4-[(E)-C-methyl-N-(thiophen-3-ylmethoxy)carbonimidoyl]phenoxy]methyl]phenyl]-1,2,4-triazol-3-one
—— 3-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazole —— C23H24F3N3O2S
3-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazole
—— 2-[2-methyl-3-[(1-phenyltetrazol-5-yl)sulfanylmethyl]phenyl]sulfanylethyl N-phenylcarbamate —— C24H23N5O2S2
2-[2-methyl-3-[(1-phenyltetrazol-5-yl)sulfanylmethyl]phenyl]sulfanylethyl N-phenylcarbamate
—— 1-(3-fluorophenyl)-3-[[(3S)-1-[1-(2-fluorophenyl)-5-methylpyrazole-4-carbonyl]piperidin-3-yl]methyl]urea —— C24H25F2N5O2
1-(3-fluorophenyl)-3-[[(3S)-1-[1-(2-fluorophenyl)-5-methylpyrazole-4-carbonyl]piperidin-3-yl]methyl]urea
—— 4-[3-[4-[3-(Methylamino)propylcarbamoyl]phenyl]-5-nitroindazol-1-yl]benzoic acid —— C25H23N5O5
4-[3-[4-[3-(Methylamino)propylcarbamoyl]phenyl]-5-nitroindazol-1-yl]benzoic acid
—— N-benzyl-2-(2-methylphenyl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-1,3-thiazole-4-carboxamide —— C25H29N3O2S
N-benzyl-2-(2-methylphenyl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-1,3-thiazole-4-carboxamide
—— 3-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazole —— C23H24F3N3O2S
3-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-5-[(1S)-1-[4-(trifluoromethyl)phenyl]ethyl]sulfanyl-1,2,4-triazole
—— N-benzyl-1-(4-fluorophenyl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]triazole-4-carboxamide —— C23H26FN5O2
N-benzyl-1-(4-fluorophenyl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]triazole-4-carboxamide
—— (4Z)-4-[[5-methyl-2-(4-nitrophenyl)-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid —— C20H15N5O7S
(4Z)-4-[[5-methyl-2-(4-nitrophenyl)-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid
—— 1-(3-fluorophenyl)-3-[[(3R)-1-[1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carbonyl]piperidin-3-yl]methyl]urea —— C27H32FN5O2
1-(3-fluorophenyl)-3-[[(3R)-1-[1-(4-methylphenyl)-5-propan-2-ylpyrazole-4-carbonyl]piperidin-3-yl]methyl]urea
—— 1-[[(3S)-1-[2-[1-(3,5-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea —— C26H30FN5O2S
1-[[(3S)-1-[2-[1-(3,5-dimethylphenyl)imidazol-2-yl]sulfanylacetyl]piperidin-3-yl]methyl]-3-(3-fluorophenyl)urea
—— 3-(2,4-dimethoxyphenyl)-5-[[(2R)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C20H20N4O5
3-(2,4-dimethoxyphenyl)-5-[[(2R)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— 3-[4-(difluoromethoxy)-3-methoxyphenyl]-5-[[(2S)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole —— C20H18F2N4O5
3-[4-(difluoromethoxy)-3-methoxyphenyl]-5-[[(2S)-2-methyl-5-nitro-2,3-dihydroindol-1-yl]methyl]-1,2,4-oxadiazole
—— 3-(5-aminopentyl)-1-[(4-methoxyphenyl)methyl]-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1,3-diazinan-4-one —— C26H31N5O2S
3-(5-aminopentyl)-1-[(4-methoxyphenyl)methyl]-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1,3-diazinan-4-one
—— N-benzyl-3-methyl-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-1-phenylpyrazole-4-carboxamide —— C25H30N4O2
N-benzyl-3-methyl-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-1-phenylpyrazole-4-carboxamide
—— methyl (3R)-3-[[1-(2-chlorophenyl)pyrazole-3-carbonyl]amino]-3-(4-methylsulfanylphenyl)propanoate —— C21H20ClN3O3S
methyl (3R)-3-[[1-(2-chlorophenyl)pyrazole-3-carbonyl]amino]-3-(4-methylsulfanylphenyl)propanoate
—— N-benzyl-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)acetamide —— C23H27N5O2S
N-benzyl-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-2-(2-pyrazin-2-yl-1,3-thiazol-4-yl)acetamide
—— 1-[3-ethyl-6-methyl-1-(2,4,6-trichlorophenyl)pyrazolo[3,4-d]pyrimidin-4-yl]-3,6-dihydro-2H-pyridine-4-carboxamide —— C20H19Cl3N6O
1-[3-ethyl-6-methyl-1-(2,4,6-trichlorophenyl)pyrazolo[3,4-d]pyrimidin-4-yl]-3,6-dihydro-2H-pyridine-4-carboxamide
—— 3-(6-aminohexyl)-1-(cyclohexylmethyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1,3-diazinan-4-one —— C26H37N5OS
3-(6-aminohexyl)-1-(cyclohexylmethyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1,3-diazinan-4-one
—— 2-[[5-[4-[[3-Cyclopentylpropanoyl(methyl)amino]methyl]-3-methoxyphenyl]tetrazol-2-yl]methyl]benzoic acid —— C26H31N5O4
2-[[5-[4-[[3-Cyclopentylpropanoyl(methyl)amino]methyl]-3-methoxyphenyl]tetrazol-2-yl]methyl]benzoic acid
—— methyl (3R)-3-[(3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-(4-methylsulfanylphenyl)propanoate —— C22H23N3O3S
methyl (3R)-3-[(3-methyl-1-phenylpyrazole-4-carbonyl)amino]-3-(4-methylsulfanylphenyl)propanoate
—— methyl (3S)-3-[[1-(2-chlorophenyl)pyrazole-3-carbonyl]amino]-3-(4-methylsulfanylphenyl)propanoate —— C21H20ClN3O3S
methyl (3S)-3-[[1-(2-chlorophenyl)pyrazole-3-carbonyl]amino]-3-(4-methylsulfanylphenyl)propanoate
—— N-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfanyl)pyrazol-3-yl]-N'-ethylmethanimidamide —— C15H9Cl2F6N5S
N-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfanyl)pyrazol-3-yl]-N'-ethylmethanimidamide
—— N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-3-ethoxy-N-[[(2R)-oxolan-2-yl]methyl]propanamide —— C19H23BrN2O3S
N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-3-ethoxy-N-[[(2R)-oxolan-2-yl]methyl]propanamide
—— N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-3-ethoxy-N-[[(2S)-oxolan-2-yl]methyl]propanamide —— C19H23BrN2O3S
N-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-3-ethoxy-N-[[(2S)-oxolan-2-yl]methyl]propanamide
—— 3-[2-bromo-4-(dimethylamino)-6-methoxyphenyl]-5-methyl-N,N-dipropyltriazolo[4,5-d]pyrimidin-7-amine —— C20H28BrN7O
3-[2-bromo-4-(dimethylamino)-6-methoxyphenyl]-5-methyl-N,N-dipropyltriazolo[4,5-d]pyrimidin-7-amine