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中文名称 英文名称 CAS号 化学式 结构式图片
—— [1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-piperidin-1-ylmethanone —— C22H29FN4O2
[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-piperidin-1-ylmethanone
—— 1-[[(2S)-4-benzylmorpholin-2-yl]methyl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea —— C23H28N6O2
1-[[(2S)-4-benzylmorpholin-2-yl]methyl]-3-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]urea
—— (2S)-1-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol —— C21H32N4O3
(2S)-1-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-3-propan-2-yloxypropan-2-ol
—— 1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(3-propan-2-yloxypropyl)piperidine-4-carboxamide —— C23H33FN4O3
1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(3-propan-2-yloxypropyl)piperidine-4-carboxamide
—— [(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-morpholin-4-ylmethanone —— C21H27FN4O3
[(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-morpholin-4-ylmethanone
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C20H23FN4OS
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-(4-methylpiperidin-1-yl)ethyl]-1,2,4-oxadiazole —— C17H22FN3O
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-(4-methylpiperidin-1-yl)ethyl]-1,2,4-oxadiazole
—— (4-ethylphenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C24H27FN4O2
(4-ethylphenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 5-[(1S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C18H18FN3OS
5-[(1S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— N-[(2R)-butan-2-yl]-3-[[[5-(4-methylphenyl)-1H-pyrazol-4-yl]methylamino]methyl]benzamide —— C23H28N4O
N-[(2R)-butan-2-yl]-3-[[[5-(4-methylphenyl)-1H-pyrazol-4-yl]methylamino]methyl]benzamide
—— 5-[(1R)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H27FN4O
5-[(1R)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1S)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C22H24FN3O3
5-[(1S)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone —— C20H26FN5O3
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone
—— [(2R,6S)-2,6-dimethylmorpholin-4-yl]-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone —— C23H31FN4O3
[(2R,6S)-2,6-dimethylmorpholin-4-yl]-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone
—— [(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-morpholin-4-ylmethanone —— C21H27FN4O3
[(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-morpholin-4-ylmethanone
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone —— C20H26FN5O3
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-morpholin-4-ylmethanone
—— 1-[(2R)-2-(dimethylamino)-3-phenylpropyl]-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]urea —— C24H31N5O
1-[(2R)-2-(dimethylamino)-3-phenylpropyl]-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]urea
—— 2-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-1-pyrrolidin-1-ylethanone —— C22H29FN4O2
2-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-1-pyrrolidin-1-ylethanone
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(imidazo[1,2-a]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C23H25FN6O
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(imidazo[1,2-a]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C20H23FN4OS
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[(3S)-3-methylpiperidin-1-yl]ethyl]-1,2,4-oxadiazole —— C17H22FN3O
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[(3S)-3-methylpiperidin-1-yl]ethyl]-1,2,4-oxadiazole
—— 5-[(1S)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C20H27FN4O
5-[(1S)-1-(4-cyclopentylpiperazin-1-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C18H18FN3OS
5-[(1R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole —— C22H24FN3O3
5-[(1R)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(imidazo[1,2-a]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C23H25FN6O
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(imidazo[1,2-a]pyridin-2-ylmethyl)piperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 1-(azepan-1-yl)-2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethanone —— C23H32FN5O2
1-(azepan-1-yl)-2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethanone
—— [1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-piperidin-1-ylmethanone —— C22H29FN4O2
[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-piperidin-1-ylmethanone
—— 1-(3-chlorophenyl)-5-methyl-3-[(3S)-oxolan-3-yl]-1,2,4-triazole —— C13H14ClN3O
1-(3-chlorophenyl)-5-methyl-3-[(3S)-oxolan-3-yl]-1,2,4-triazole
—— N,N-diethyl-2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]acetamide —— C21H30FN5O2
N,N-diethyl-2-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]acetamide
—— N-benzyl-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidine-4-carboxamide —— C24H27FN4O2
N-benzyl-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidine-4-carboxamide
—— (3,4-difluorophenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H21F3N4O2
(3,4-difluorophenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 4-[(2S)-1-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole —— C21H25FN4O
4-[(2S)-1-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
—— 3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(2S)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]propan-1-one —— C15H23N3O
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(2S)-2-propan-2-yl-2,5-dihydropyrrol-1-yl]propan-1-one
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(2-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C21H22F2N4O3S
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(2-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(2-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C21H22F2N4O3S
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(2-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— N-benzyl-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidine-4-carboxamide —— C24H27FN4O2
N-benzyl-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidine-4-carboxamide
—— (3,4-difluorophenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H21F3N4O2
(3,4-difluorophenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— N,N-diethyl-2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]acetamide —— C21H30FN5O2
N,N-diethyl-2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]acetamide
—— 3-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-1H-benzimidazol-2-one —— C23H24FN5O2
3-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-1H-benzimidazol-2-one
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C21H22F2N4O3S
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 4-[(2R)-1-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole —— C21H25FN4O
4-[(2R)-1-[[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]methyl]pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
—— (4-ethylphenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C24H27FN4O2
(4-ethylphenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 1-(3-chlorophenyl)-5-methyl-3-[(3R)-oxolan-3-yl]-1,2,4-triazole —— C13H14ClN3O
1-(3-chlorophenyl)-5-methyl-3-[(3R)-oxolan-3-yl]-1,2,4-triazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C21H22F2N4O3S
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— azepan-1-yl-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone —— C23H31FN4O2
azepan-1-yl-[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C21H22F2N4O3S
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-(4-phenylmethoxypiperidin-1-yl)ethyl]-1,2,4-oxadiazole —— C23H26FN3O2
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-(4-phenylmethoxypiperidin-1-yl)ethyl]-1,2,4-oxadiazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole —— C21H22F2N4O3S
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]ethyl]-1,2,4-oxadiazole
—— azepan-1-yl-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone —— C23H31FN4O2
azepan-1-yl-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]methanone
—— N-[[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-3-[(2S)-oxolan-2-yl]propan-1-amine —— C19H27N3O2
N-[[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl]-N-methyl-3-[(2S)-oxolan-2-yl]propan-1-amine