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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-1-[2-(1-phenylethylamino)pyrimidin-4-yl]-2-(3-trifluoromethylphenyl)-1H-imidazole-4-carboxylic acid (2-dimethylaminoethyl)amide 306297-59-6 C27H28F3N7O
(S)-1-[2-(1-phenylethylamino)pyrimidin-4-yl]-2-(3-trifluoromethylphenyl)-1H-imidazole-4-carboxylic acid (2-dimethylaminoethyl)amide
—— 2-[[4-[(2S)-butan-2-yl]-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[3-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)phenyl]acetamide —— C30H39N7O6S3
2-[[4-[(2S)-butan-2-yl]-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[3-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)phenyl]acetamide
—— ethyl (4R)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H24ClFN4O5
ethyl (4R)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[(3S,3aR,7E)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-2-[[5-(2-chlorophenyl)-4-(2,5-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C34H30ClN5OS3
1-[(3S,3aR,7E)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-2-[[5-(2-chlorophenyl)-4-(2,5-dimethylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— ethyl (4S)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H24ClFN4O5
ethyl (4S)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 4-[[5-[2-[2-(2-Methoxyphenyl)-4,10-dihydroimidazo[2,1-c][1,4]benzodiazepin-5-yl]-2-oxoethyl]imidazol-1-yl]methyl]benzonitrile —— C31H26N6O2
4-[[5-[2-[2-(2-Methoxyphenyl)-4,10-dihydroimidazo[2,1-c][1,4]benzodiazepin-5-yl]-2-oxoethyl]imidazol-1-yl]methyl]benzonitrile
—— N'-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfonyl)pyrazol-3-yl]-N-prop-1-en-2-ylmethanimidamide —— C16H9Cl2F6N5O2S
N'-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfonyl)pyrazol-3-yl]-N-prop-1-en-2-ylmethanimidamide
—— N-[3-(2,6-dichloro-4-methoxy-phenyl)2,5-dimethyl-pyrazolo [1,5-a]pyrimidin-7-yl]-N'-(2,2,6,6-tetramethyl-piperidin-4-yl)ethane-1,2-diamine 332178-90-2 C26H36Cl2N6O
N-[3-(2,6-dichloro-4-methoxy-phenyl)2,5-dimethyl-pyrazolo [1,5-a]pyrimidin-7-yl]-N'-(2,2,6,6-tetramethyl-piperidin-4-yl)ethane-1,2-diamine
—— 3-[2-Methyl-5-[2-methyl-5-(2-sulfamoylphenyl)benzimidazole-1-carbonyl]imidazol-1-yl]benzenecarboximidamide —— C26H23N7O3S
3-[2-Methyl-5-[2-methyl-5-(2-sulfamoylphenyl)benzimidazole-1-carbonyl]imidazol-1-yl]benzenecarboximidamide
—— N-[3-(2,6-dichloro-phenyl)-5-ethyl-2-methyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine 332179-02-9 C26H30Cl2N8
N-[3-(2,6-dichloro-phenyl)-5-ethyl-2-methyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)-ethane-1,2-diamine
—— 3-[3-Methyl-5-[2-methyl-5-(2-sulfamoylphenyl)benzimidazole-1-carbonyl]pyrazol-1-yl]benzenecarboximidamide —— C26H23N7O3S
3-[3-Methyl-5-[2-methyl-5-(2-sulfamoylphenyl)benzimidazole-1-carbonyl]pyrazol-1-yl]benzenecarboximidamide
—— 3-Chloro4-(2,2-dibromocyclopropyl)-1-(2,6-dichloro-4-trifluoromethylphenyl)pyrazole —— C13H6Br2Cl3F3N2
3-Chloro4-(2,2-dibromocyclopropyl)-1-(2,6-dichloro-4-trifluoromethylphenyl)pyrazole
—— 3-[5-(4-chlorophenyl)-1-[4-(quinolin-2-ylmethoxy)phenyl]pyrazol-3-yl]-N-hydroxy-N-methylpropanamide —— C29H25ClN4O3
3-[5-(4-chlorophenyl)-1-[4-(quinolin-2-ylmethoxy)phenyl]pyrazol-3-yl]-N-hydroxy-N-methylpropanamide
—— 1-(2,4,6-trichlorophenyl)-3-isopropyl-6-(3-aminoindazol-5-ylmethyl)pyrazolo[3,4-d]pyrimidin-4-one —— C22H18Cl3N7O
1-(2,4,6-trichlorophenyl)-3-isopropyl-6-(3-aminoindazol-5-ylmethyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 2-[(3-Hydroxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid —— C28H26N2O7
2-[(3-Hydroxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid
—— 2-[[4-(cyclopropylmethoxy)phenyl]sulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]-N-hydroxyacetamide;hydrochloride —— C21H24ClN5O5S
2-[[4-(cyclopropylmethoxy)phenyl]sulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]-N-hydroxyacetamide;hydrochloride
—— N-[4-(2-(phenyloxazol-4yl)ethoxy)phenyl]-N-phenylmethyl sulfonylglycine 328248-02-8 C26H24N2O6S
N-[4-(2-(phenyloxazol-4yl)ethoxy)phenyl]-N-phenylmethyl sulfonylglycine
—— N-[(1R)-1-phenylethyl]-4-[2-piperidin-1-yl-4-[3-(trifluoromethyl)phenyl]-1H-imidazol-5-yl]pyridin-2-amine —— C28H28F3N5
N-[(1R)-1-phenylethyl]-4-[2-piperidin-1-yl-4-[3-(trifluoromethyl)phenyl]-1H-imidazol-5-yl]pyridin-2-amine
—— L 368935 —— C27H26N8O2
L 368935
—— N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5 dimethyl-pyrazolo [1,5-a]pyrimidin-7-yl]-N'-(1-ethyl-piperidin-4-yl)-ethane-1,2-di amine 332178-88-8 C24H32Cl2N6O
N-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5 dimethyl-pyrazolo [1,5-a]pyrimidin-7-yl]-N'-(1-ethyl-piperidin-4-yl)-ethane-1,2-di amine
—— 2-[[4-(cyclopropylmethoxy)phenyl]sulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]-N-hydroxyacetamide —— C21H23N5O5S
2-[[4-(cyclopropylmethoxy)phenyl]sulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]-N-hydroxyacetamide
—— (4Z)-4-[[5-methyl-2-(3-nitrophenyl)-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid —— C20H15N5O7S
(4Z)-4-[[5-methyl-2-(3-nitrophenyl)-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid
—— 8-(2,6-difluorobenzyl)-5,8-dihydro-3-(hydroxymethyl)-2-(4-nitrophenyl)-5-oxoimidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester 229484-75-7 C23H18F2N4O6
8-(2,6-difluorobenzyl)-5,8-dihydro-3-(hydroxymethyl)-2-(4-nitrophenyl)-5-oxoimidazo[1,2-a]pyrimidine-6-carboxylic acid ethyl ester
—— 2-(2-fluorophenyl)-4-(trifluoromethyl)-N-[1-[3-(trifluoromethoxy)phenyl]ethyl]-5-thiazolecarboxamide 725247-76-7 C20H13F7N2O2S
2-(2-fluorophenyl)-4-(trifluoromethyl)-N-[1-[3-(trifluoromethoxy)phenyl]ethyl]-5-thiazolecarboxamide
—— (Z)-1-[2-[[1-(2,4-dichlorophenyl)-4-methylpyrazol-3-yl]oxymethyl]phenyl]-1-(5,6-dihydro-1,4,2-dioxazin-3-yl)-N-methoxymethanimine —— C22H20Cl2N4O4
(Z)-1-[2-[[1-(2,4-dichlorophenyl)-4-methylpyrazol-3-yl]oxymethyl]phenyl]-1-(5,6-dihydro-1,4,2-dioxazin-3-yl)-N-methoxymethanimine
—— [(2R)-2-[(1-benzyl-5-chloro-3-methylpyrazole-4-carbonyl)amino]propyl] 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylate —— C27H27Cl2N5O3
[(2R)-2-[(1-benzyl-5-chloro-3-methylpyrazole-4-carbonyl)amino]propyl] 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylate
—— (2R)-N-[(Z)-1-(4-bromophenyl)ethylideneamino]-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C27H26BrClN6OS
(2R)-N-[(Z)-1-(4-bromophenyl)ethylideneamino]-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N'-Benzoyl-4-[(1,5-diphenyl-1H-1,2,4-triazol-3-yl)amino]benzohydrazide 301547-52-4 C28H22N6O2
N'-Benzoyl-4-[(1,5-diphenyl-1H-1,2,4-triazol-3-yl)amino]benzohydrazide
—— (2S)-N-[(Z)-1-(4-bromophenyl)ethylideneamino]-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C27H26BrClN6OS
(2S)-N-[(Z)-1-(4-bromophenyl)ethylideneamino]-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N'-[3-(2,6-dichloro-4-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-piperidin-4-ylethane-1,2-diamine —— C22H28Cl2N6O
N'-[3-(2,6-dichloro-4-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-piperidin-4-ylethane-1,2-diamine
—— 1-(2,4,6-trichlorophenyl)-3-isopropyl-6-(3-hydroxybenzyl)pyrazolo[3,4-d]pyrimidin-4-one —— C21H17Cl3N4O2
1-(2,4,6-trichlorophenyl)-3-isopropyl-6-(3-hydroxybenzyl)pyrazolo[3,4-d]pyrimidin-4-one
—— 4-[2-[[(E)-1-[4-[(E)-N-[(E)-but-2-enoxy]-C-methylcarbonimidoyl]phenyl]ethylideneamino]oxymethyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one —— C25H29N5O4
4-[2-[[(E)-1-[4-[(E)-N-[(E)-but-2-enoxy]-C-methylcarbonimidoyl]phenyl]ethylideneamino]oxymethyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one
—— [2-Bromo-4-(3-methyl-pyrazol-1-yl)-phenyl]-(11H-5-oxa-4,10-diaza-dibenzo[a,d]cyclohepten-10-yl)-methanone —— C23H17BrN4O2
[2-Bromo-4-(3-methyl-pyrazol-1-yl)-phenyl]-(11H-5-oxa-4,10-diaza-dibenzo[a,d]cyclohepten-10-yl)-methanone
—— 3-(2-bromo-6-methoxy-4-methylsulfanylphenyl)-N-butyl-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine —— C19H25BrN6OS
3-(2-bromo-6-methoxy-4-methylsulfanylphenyl)-N-butyl-N-ethyl-5-methyltriazolo[4,5-d]pyrimidin-7-amine
—— 2-[[5-[4-[(2-Butylimidazo[4,5-b]pyridin-3-yl)methyl]phenyl]tetrazol-2-yl]methyl]benzoic acid —— C26H25N7O2
2-[[5-[4-[(2-Butylimidazo[4,5-b]pyridin-3-yl)methyl]phenyl]tetrazol-2-yl]methyl]benzoic acid
—— [(3aS,6aR)-1-[(1-methylpyrazol-4-yl)methyl]-2,3,3a,5,6,6a-hexahydropyrrolo[3,2-b]pyrrol-4-yl]-(1,3-thiazol-4-yl)methanone —— C15H19N5OS
[(3aS,6aR)-1-[(1-methylpyrazol-4-yl)methyl]-2,3,3a,5,6,6a-hexahydropyrrolo[3,2-b]pyrrol-4-yl]-(1,3-thiazol-4-yl)methanone
—— (4Z)-4-[[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid —— C20H15ClN4O5S
(4Z)-4-[[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid
—— 1-(1-Adamantyl)-3-[1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]urea —— C34H35FN6O3S
1-(1-Adamantyl)-3-[1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]urea
—— 4-[[[5-[(2,6-Difluorophenyl)methyl]-4-(2-hydroxyphenyl)-1,3-thiazol-2-yl]amino]methyl]cyclohexane-1-carboxylic acid —— C24H24F2N2O3S
4-[[[5-[(2,6-Difluorophenyl)methyl]-4-(2-hydroxyphenyl)-1,3-thiazol-2-yl]amino]methyl]cyclohexane-1-carboxylic acid
—— 4-[4-(4-fluorophenyl)-2-(1-methylpiperidin-4-yl)-1,3-oxazol-5-yl]-N-[(1S)-1-phenylethyl]pyrimidin-2-amine —— C27H28FN5O
4-[4-(4-fluorophenyl)-2-(1-methylpiperidin-4-yl)-1,3-oxazol-5-yl]-N-[(1S)-1-phenylethyl]pyrimidin-2-amine
—— (3aR,6aS)-4-[(6-methylpyridin-2-yl)methyl]-1-(1,3-thiazole-4-carbonyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one —— C17H18N4O2S
(3aR,6aS)-4-[(6-methylpyridin-2-yl)methyl]-1-(1,3-thiazole-4-carbonyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one
—— (3aS,6aR)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(1,3-thiazol-2-ylmethyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one —— C15H18N4OS2
(3aS,6aR)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(1,3-thiazol-2-ylmethyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one
—— (3aS,6aR)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one —— C17H20N4OS
(3aS,6aR)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one
—— (3aR,6aR)-4-[(6-methylpyridin-2-yl)methyl]-1-(1,3-thiazole-4-carbonyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one —— C17H18N4O2S
(3aR,6aR)-4-[(6-methylpyridin-2-yl)methyl]-1-(1,3-thiazole-4-carbonyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one
—— 3,4-dimethoxy-N-[[4-(3-phenyl-1,2,4-oxadiazol-5-yl)phenyl]methyl]benzenesulfonamide —— C23H21N3O5S
3,4-dimethoxy-N-[[4-(3-phenyl-1,2,4-oxadiazol-5-yl)phenyl]methyl]benzenesulfonamide
—— (3aS,6aS)-4-[(6-methylpyridin-2-yl)methyl]-1-(1,3-thiazole-4-carbonyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one —— C17H18N4O2S
(3aS,6aS)-4-[(6-methylpyridin-2-yl)methyl]-1-(1,3-thiazole-4-carbonyl)-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrol-5-one
—— [2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl] (E)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C32H25N3O5
[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl] (E)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— 1,3-diethyl-5-[5-(3-methylphenyl)-3-[(3R)-pyrrolidin-3-yl]imidazol-4-yl]benzimidazol-2-one;hydrochloride —— C25H30ClN5O
1,3-diethyl-5-[5-(3-methylphenyl)-3-[(3R)-pyrrolidin-3-yl]imidazol-4-yl]benzimidazol-2-one;hydrochloride
—— [(2S)-2-[(1-benzyl-5-chloro-3-methylpyrazole-4-carbonyl)amino]propyl] 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylate —— C27H27Cl2N5O3
[(2S)-2-[(1-benzyl-5-chloro-3-methylpyrazole-4-carbonyl)amino]propyl] 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylate
—— [2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl] (E)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C32H25N3O5
[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl] (E)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate