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中文名称 英文名称 CAS号 化学式 结构式图片
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-fluorophenyl)methanone —— C22H22F2N4O2
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-fluorophenyl)methanone
—— 1-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-morpholin-4-ylethanone —— C21H28FN5O3
1-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-morpholin-4-ylethanone
—— 1-[(2S)-6-methylheptan-2-yl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C15H27N3OS
1-[(2S)-6-methylheptan-2-yl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 1-[(2R)-6-methylheptan-2-yl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C15H27N3OS
1-[(2R)-6-methylheptan-2-yl]-3-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(2R)-2-(diethylamino)-2-(furan-2-yl)ethyl]acetamide —— C19H23ClN6O2
2-[5-(4-chlorophenyl)tetrazol-2-yl]-N-[(2R)-2-(diethylamino)-2-(furan-2-yl)ethyl]acetamide
—— 4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N,N-dimethylpiperazine-1-carboxamide —— C18H24FN5O2
4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N,N-dimethylpiperazine-1-carboxamide
—— (4-chlorophenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H22ClFN4O2
(4-chlorophenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 1,3-benzodioxol-5-yl-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C23H23FN4O4
1,3-benzodioxol-5-yl-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-heptan-2-yl]urea —— C16H30N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-heptan-2-yl]urea
—— (3-chlorophenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H22ClFN4O2
(3-chlorophenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-fluorophenyl)methanone —— C22H22F2N4O2
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-fluorophenyl)methanone
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-5-methylhexan-2-yl]urea —— C16H30N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2S)-5-methylhexan-2-yl]urea
—— 1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-octan-2-yl]urea —— C17H32N4O
1-[3-(3,5-dimethylpyrazol-1-yl)propyl]-3-[(2R)-octan-2-yl]urea
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(3-methoxyphenyl)methanone —— C23H25FN4O3
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(3-methoxyphenyl)methanone
—— 2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-morpholin-4-ylethanone —— C21H28FN5O3
2-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-1-morpholin-4-ylethanone
—— 2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]ethanone —— C20H23ClN8O
2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]ethanone
—— 2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]ethanone —— C21H22ClN5O2
2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-[(R)-hydroxy(phenyl)methyl]piperidin-1-yl]ethanone
—— 2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-[(S)-hydroxy(phenyl)methyl]piperidin-1-yl]ethanone —— C21H22ClN5O2
2-[5-(4-chlorophenyl)tetrazol-2-yl]-1-[4-[(S)-hydroxy(phenyl)methyl]piperidin-1-yl]ethanone
—— 2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]-N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]acetamide —— C20H28N4O4
2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]-N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]acetamide
—— N-benzyl-N-[(1R)-1-cyclopropylethyl]-2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetamide —— C23H25N3O3
N-benzyl-N-[(1R)-1-cyclopropylethyl]-2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetamide
—— N-[4-[(2S)-butan-2-yl]phenyl]-2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetamide —— C21H23N3O3
N-[4-[(2S)-butan-2-yl]phenyl]-2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetamide
—— N-[4-[(2R)-butan-2-yl]phenyl]-2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetamide —— C21H23N3O3
N-[4-[(2R)-butan-2-yl]phenyl]-2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetamide
—— (3S)-1-[2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetyl]piperidine-3-carboxamide —— C17H20N4O4
(3S)-1-[2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]acetyl]piperidine-3-carboxamide
—— 3-(2,4-dichlorophenyl)-4-[(E)-(2,4-dimethylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C17H14Cl2N4S
3-(2,4-dichlorophenyl)-4-[(E)-(2,4-dimethylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]-N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]acetamide —— C20H28N4O4
2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenoxy]-N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]acetamide
—— 1-benzyl-5-ethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide —— C21H30N4O
1-benzyl-5-ethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide
—— (2R,3S)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide —— C21H24N4O
(2R,3S)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide
—— (2R,3R)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide —— C21H24N4O
(2R,3R)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide
—— (2S,3R)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide —— C21H24N4O
(2S,3R)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide
—— (2S,3S)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide —— C21H24N4O
(2S,3S)-3-methyl-2-phenyl-N-[(4-phenyl-1,2,4-triazol-3-yl)methyl]pentanamide
—— 1-benzyl-N-[[6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-5-ethylpyrazole-4-carboxamide —— C25H31N5O2
1-benzyl-N-[[6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-5-ethylpyrazole-4-carboxamide
—— N-[2-(3,5-dimethylpyrazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[(2R)-oxolan-2-yl]methoxy]propanamide —— C20H24F3N3O3
N-[2-(3,5-dimethylpyrazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[(2R)-oxolan-2-yl]methoxy]propanamide
—— 1-benzyl-5-ethyl-N-[(2S)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide —— C23H28N4O
1-benzyl-5-ethyl-N-[(2S)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide —— C21H30N4O
1-benzyl-5-ethyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[[6-[(2R)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]pyrazole-4-carboxamide —— C24H29N5O2
1-benzyl-5-ethyl-N-[[6-[(2R)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]pyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[[6-[(2S)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]pyrazole-4-carboxamide —— C24H29N5O2
1-benzyl-5-ethyl-N-[[6-[(2S)-2-methylmorpholin-4-yl]pyridin-3-yl]methyl]pyrazole-4-carboxamide
—— N-[2-(3,5-dimethylpyrazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[(2S)-oxolan-2-yl]methoxy]propanamide —— C20H24F3N3O3
N-[2-(3,5-dimethylpyrazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[(2S)-oxolan-2-yl]methoxy]propanamide
—— 1-benzyl-N-[[6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-5-ethylpyrazole-4-carboxamide —— C25H31N5O2
1-benzyl-N-[[6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-5-ethylpyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]pyrazole-4-carboxamide —— C22H32N4O
1-benzyl-5-ethyl-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]pyrazole-4-carboxamide
—— 5-chloro-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-1-phenylpyrazole-4-carboxamide —— C22H24ClN3O3
5-chloro-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-1-phenylpyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[2-[(3R)-3-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide —— C21H30N4O
1-benzyl-5-ethyl-N-[2-[(3R)-3-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[(2R)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide —— C23H28N4O
1-benzyl-5-ethyl-N-[(2R)-2-(N-methylanilino)propyl]pyrazole-4-carboxamide
—— 1-benzyl-5-ethyl-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide —— C21H30N4O
1-benzyl-5-ethyl-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]pyrazole-4-carboxamide
—— 5-chloro-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1-(4-fluorophenyl)-3-methylpyrazole-4-carboxamide —— C22H23ClFN3O3
5-chloro-N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1-(4-fluorophenyl)-3-methylpyrazole-4-carboxamide
—— 1-benzyl-N-[[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-5-ethylpyrazole-4-carboxamide —— C25H31N5O2
1-benzyl-N-[[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-5-ethylpyrazole-4-carboxamide
—— 2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]acetamide —— C21H23ClN4O3S
2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]acetamide
—— 5-chloro-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-1-phenylpyrazole-4-carboxamide —— C22H24ClN3O3
5-chloro-N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-methyl-1-phenylpyrazole-4-carboxamide
—— N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C23H28N4O3S
N-[(1S)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1-(4-fluorophenyl)-3,5-dimethylpyrazole-4-carboxamide —— C23H26FN3O3
N-[(1R)-1-(4,5-dimethoxy-2-methylphenyl)ethyl]-1-(4-fluorophenyl)-3,5-dimethylpyrazole-4-carboxamide
—— 3-[[(2S)-oxolan-2-yl]methoxy]-N-(4-pyrazol-1-ylphenyl)propanamide —— C17H21N3O3
3-[[(2S)-oxolan-2-yl]methoxy]-N-(4-pyrazol-1-ylphenyl)propanamide