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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-1H-pyrazole-5-carboxylic acid —— C13H16N4O3
4-[[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-1H-pyrazole-5-carboxylic acid
—— N-[(2R)-2-methoxy-2-thiophen-2-ylethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide —— C16H16N4O2S
N-[(2R)-2-methoxy-2-thiophen-2-ylethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
—— N-[(2S)-2-methoxy-2-thiophen-2-ylethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide —— C16H16N4O2S
N-[(2S)-2-methoxy-2-thiophen-2-ylethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
—— 1-(1-propan-2-ylpyrazol-4-yl)-3-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea —— C12H19N7O
1-(1-propan-2-ylpyrazol-4-yl)-3-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea
—— 1-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]azetidin-3-yl]-3,5-dimethylpyrazole —— C15H23N3
1-[1-[[(1R)-cyclohex-3-en-1-yl]methyl]azetidin-3-yl]-3,5-dimethylpyrazole
—— N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-(1H-imidazol-2-yl)benzamide —— C18H20N4OS
N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-(1H-imidazol-2-yl)benzamide
—— [(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone —— C19H23N3O2
[(2R)-2-butyl-2,5-dihydropyrrol-1-yl]-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]methanone
—— 5-phenyl-N-[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide —— C20H20N4O2S
5-phenyl-N-[(3S)-1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
—— 2-(1H-imidazol-2-yl)-N-[(2-methylphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C23H25N3O2
2-(1H-imidazol-2-yl)-N-[(2-methylphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (9S)-9-[2-[2-(1H-imidazol-5-yl)ethyl]-5-phenyl-1,2,4-triazol-3-yl]-6,7,8,9-tetrahydro-5H-tetrazolo[1,5-a]azepine —— C19H21N9
(9S)-9-[2-[2-(1H-imidazol-5-yl)ethyl]-5-phenyl-1,2,4-triazol-3-yl]-6,7,8,9-tetrahydro-5H-tetrazolo[1,5-a]azepine
—— 1-benzyl-5-(imidazol-1-ylmethyl)-3-[(3S)-oxolan-3-yl]-1,2,4-triazole —— C17H19N5O
1-benzyl-5-(imidazol-1-ylmethyl)-3-[(3S)-oxolan-3-yl]-1,2,4-triazole
—— 1-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]-2-[4-(tetrazol-1-yl)phenyl]ethanone —— C16H22N6O2
1-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]-2-[4-(tetrazol-1-yl)phenyl]ethanone
—— N-[(2S)-2-(4-chlorophenyl)-2-piperidin-1-ylethyl]-1-ethyl-5-methylpyrazole-4-carboxamide —— C20H27ClN4O
N-[(2S)-2-(4-chlorophenyl)-2-piperidin-1-ylethyl]-1-ethyl-5-methylpyrazole-4-carboxamide
—— 4-[[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-1H-pyrazole-5-carboxylic acid —— C13H16N4O3
4-[[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl]-1H-pyrazole-5-carboxylic acid
—— 5-[[methyl-[[(3S)-1-methylpiperidin-3-yl]methyl]amino]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid —— C13H22N4O3
5-[[methyl-[[(3S)-1-methylpiperidin-3-yl]methyl]amino]methyl]-2-oxo-1,3-dihydroimidazole-4-carboxylic acid
—— 5-[(2R)-oxolan-2-yl]-N-[(3-pyrazol-1-ylphenyl)methyl]thiophene-2-carboxamide —— C19H19N3O2S
5-[(2R)-oxolan-2-yl]-N-[(3-pyrazol-1-ylphenyl)methyl]thiophene-2-carboxamide
—— 1-(1-propan-2-ylpyrazol-4-yl)-3-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea —— C12H19N7O
1-(1-propan-2-ylpyrazol-4-yl)-3-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]urea
—— 2-ethyl-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide —— C17H22N2O3S
2-ethyl-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide
—— N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C21H21N3O3
N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— 5-[(2S)-oxolan-2-yl]-N-[(3-pyrazol-1-ylphenyl)methyl]thiophene-2-carboxamide —— C19H19N3O2S
5-[(2S)-oxolan-2-yl]-N-[(3-pyrazol-1-ylphenyl)methyl]thiophene-2-carboxamide
—— 5-cyclopropyl-1-[2-(1H-imidazol-5-yl)ethyl]-3-[(3R)-oxolan-3-yl]-1,2,4-triazole —— C14H19N5O
5-cyclopropyl-1-[2-(1H-imidazol-5-yl)ethyl]-3-[(3R)-oxolan-3-yl]-1,2,4-triazole
—— 5-cyclopropyl-1-[2-(1H-imidazol-5-yl)ethyl]-3-[(3S)-oxolan-3-yl]-1,2,4-triazole —— C14H19N5O
5-cyclopropyl-1-[2-(1H-imidazol-5-yl)ethyl]-3-[(3S)-oxolan-3-yl]-1,2,4-triazole
—— N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-(1H-imidazol-2-yl)benzamide —— C18H20N4OS
N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-2-(1H-imidazol-2-yl)benzamide
—— (2R)-N-[[1-(2-methoxyphenyl)pyrazol-4-yl]methyl]-N-methyl-1-pyrazin-2-ylpropan-2-amine —— C19H23N5O
(2R)-N-[[1-(2-methoxyphenyl)pyrazol-4-yl]methyl]-N-methyl-1-pyrazin-2-ylpropan-2-amine
—— N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-(3,4,5-trimethylpyrazol-1-yl)acetamide —— C17H27N5O
N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-(3,4,5-trimethylpyrazol-1-yl)acetamide
—— 3-(4-fluorophenyl)-N-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]-1H-pyrazole-5-carboxamide —— C22H23FN4O
3-(4-fluorophenyl)-N-[2-[(3R)-3-phenylpyrrolidin-1-yl]ethyl]-1H-pyrazole-5-carboxamide
—— 2-(1H-imidazol-2-yl)-N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]benzamide —— C16H20N4O4S
2-(1H-imidazol-2-yl)-N-[[(2R)-4-methylsulfonylmorpholin-2-yl]methyl]benzamide
—— 1-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]azetidin-3-yl]-3,5-dimethylpyrazole —— C15H23N3
1-[1-[[(1S)-cyclohex-3-en-1-yl]methyl]azetidin-3-yl]-3,5-dimethylpyrazole
—— 4-ethyl-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methyl-1,3-thiazole-5-carboxamide —— C16H24N4OS
4-ethyl-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methyl-1,3-thiazole-5-carboxamide
—— N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-(3,4,5-trimethylpyrazol-1-yl)acetamide —— C17H27N5O
N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-(3,4,5-trimethylpyrazol-1-yl)acetamide
—— (6S)-5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C16H15N5O3
(6S)-5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (2S)-N-[(5-fluoro-2-pyrazol-1-ylphenyl)methyl]-N-methyl-1-pyrazin-2-ylpropan-2-amine —— C18H20FN5
(2S)-N-[(5-fluoro-2-pyrazol-1-ylphenyl)methyl]-N-methyl-1-pyrazin-2-ylpropan-2-amine
—— 1-benzyl-5-(imidazol-1-ylmethyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazole —— C17H19N5O
1-benzyl-5-(imidazol-1-ylmethyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazole
—— (6R)-5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C16H15N5O3
(6R)-5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 4-ethyl-N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methyl-1,3-thiazole-5-carboxamide —— C16H24N4OS
4-ethyl-N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-2-methyl-1,3-thiazole-5-carboxamide
—— 2-ethyl-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-N-(thiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide —— C17H22N2O3S
2-ethyl-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-N-(thiophen-3-ylmethyl)-1,3-oxazole-5-carboxamide
—— (6S)-1-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1,4-diazepane-6-carboxylic acid —— C16H26N4O2
(6S)-1-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1,4-diazepane-6-carboxylic acid
—— N-[(2R)-2-(azepan-1-yl)-2-phenylethyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide —— C21H29N3OS
N-[(2R)-2-(azepan-1-yl)-2-phenylethyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
—— 1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1S)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]urea —— C15H18FN9O2
1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1S)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]urea
—— (2R)-N-[(5-fluoro-2-pyrazol-1-ylphenyl)methyl]-N-methyl-1-pyrazin-2-ylpropan-2-amine —— C18H20FN5
(2R)-N-[(5-fluoro-2-pyrazol-1-ylphenyl)methyl]-N-methyl-1-pyrazin-2-ylpropan-2-amine
—— (6R)-1-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1,4-diazepane-6-carboxylic acid —— C16H26N4O2
(6R)-1-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1,4-diazepane-6-carboxylic acid
—— (2S)-2-[5-(oxan-4-yl)-2-phenyl-1,2,4-triazol-3-yl]-6-azaspiro[2.5]octane —— C20H26N4O
(2S)-2-[5-(oxan-4-yl)-2-phenyl-1,2,4-triazol-3-yl]-6-azaspiro[2.5]octane
—— [(2R)-2-[1-(2-methoxyethyl)tetrazol-5-yl]morpholin-4-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C18H21N7O3
[(2R)-2-[1-(2-methoxyethyl)tetrazol-5-yl]morpholin-4-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— (2R)-2-cyclohexyl-2-[2-(2-hydroxyethyl)-5-(5-methylfuran-2-yl)-1,2,4-triazol-3-yl]acetic acid —— C17H23N3O4
(2R)-2-cyclohexyl-2-[2-(2-hydroxyethyl)-5-(5-methylfuran-2-yl)-1,2,4-triazol-3-yl]acetic acid
—— N-[(2S)-2-(azepan-1-yl)-2-phenylethyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide —— C21H29N3OS
N-[(2S)-2-(azepan-1-yl)-2-phenylethyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
—— 1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1R)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]urea —— C15H18FN9O2
1-[2-fluoro-5-(tetrazol-1-yl)phenyl]-3-[(1R)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]urea
—— [(2S)-2-[1-(2-methoxyethyl)tetrazol-5-yl]morpholin-4-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C18H21N7O3
[(2S)-2-[1-(2-methoxyethyl)tetrazol-5-yl]morpholin-4-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— (2R)-2-[5-(oxan-4-yl)-2-phenyl-1,2,4-triazol-3-yl]-6-azaspiro[2.5]octane —— C20H26N4O
(2R)-2-[5-(oxan-4-yl)-2-phenyl-1,2,4-triazol-3-yl]-6-azaspiro[2.5]octane
—— 3-(2-amino-1,3-thiazol-4-yl)-N-[(2R)-1-thiophen-3-ylpropan-2-yl]propanamide —— C13H17N3OS2
3-(2-amino-1,3-thiazol-4-yl)-N-[(2R)-1-thiophen-3-ylpropan-2-yl]propanamide
—— (2S)-2-cyclohexyl-2-[2-(2-hydroxyethyl)-5-(5-methylfuran-2-yl)-1,2,4-triazol-3-yl]acetic acid —— C17H23N3O4
(2S)-2-cyclohexyl-2-[2-(2-hydroxyethyl)-5-(5-methylfuran-2-yl)-1,2,4-triazol-3-yl]acetic acid