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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(4-bromophenyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide —— C18H16BrN3O2
1-(4-bromophenyl)-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrazole-4-carboxamide
—— N-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzamide —— C23H25FN4O2
N-[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]benzamide
—— methyl 4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazine-1-carboxylate —— C17H21FN4O3
methyl 4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazine-1-carboxylate
—— methyl 4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazine-1-carboxylate —— C17H21FN4O3
methyl 4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazine-1-carboxylate
—— 4-(2-methylsulfanylimidazol-1-yl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide —— C19H19N3O2S
4-(2-methylsulfanylimidazol-1-yl)-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]benzamide
—— (2,5-dimethylfuran-3-yl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C22H25FN4O3
(2,5-dimethylfuran-3-yl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— (1R)-1-(2-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine —— C19H18ClF2N3O2
(1R)-1-(2-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine
—— 2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide —— C22H22F3N3O2
2-[3,5-dimethyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]acetamide
—— N-butyl-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-methylpiperidine-4-carboxamide —— C22H31FN4O2
N-butyl-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-methylpiperidine-4-carboxamide
—— (3-fluoro-4-methylphenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C23H24F2N4O2
(3-fluoro-4-methylphenyl)-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— N-butyl-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-methylpiperidine-4-carboxamide —— C22H31FN4O2
N-butyl-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-methylpiperidine-4-carboxamide
—— (1S)-1-(3-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine —— C19H18ClF2N3O2
(1S)-1-(3-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine
—— 1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-(1H-indol-3-yl)ethanone —— C25H26FN5O2
1-[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-2-(1H-indol-3-yl)ethanone
—— (3S)-3-benzyl-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one —— C21H20N4O2
(3S)-3-benzyl-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one
—— 2-[(2R)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]ethanol —— C18H24FN3O
2-[(2R)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]ethanol
—— [1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-(4-methylpiperidin-1-yl)methanone —— C23H31FN4O2
[1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-(4-methylpiperidin-1-yl)methanone
—— 3-[2-(difluoromethoxy)phenyl]-5-[[(2R)-2-(2-phenylethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C22H23F2N3O2
3-[2-(difluoromethoxy)phenyl]-5-[[(2R)-2-(2-phenylethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methyl-1-[(2S)-oxolan-2-yl]methanamine —— C16H19F2N3O3
N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methyl-1-[(2S)-oxolan-2-yl]methanamine
—— (1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-fluorophenyl)-N-methylethanamine —— C19H18F3N3O2
(1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-fluorophenyl)-N-methylethanamine
—— 3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-[5-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-1-yl]ethyl]-1,2,4-oxadiazole —— C22H23F4N5O
3-(4-fluoro-3-methylphenyl)-5-[(1R)-1-[4-[5-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-1-yl]ethyl]-1,2,4-oxadiazole
—— [1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-(4-methylpiperidin-1-yl)methanone —— C23H31FN4O2
[1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-4-yl]-(4-methylpiperidin-1-yl)methanone
—— 3-(β-D-glucopyranosyloxy)-4-[(4-isopropoxyphenyl)methyl]-5-methyl-1-phenyl-1H-pyrazole —— C26H32N2O7
3-(β-D-glucopyranosyloxy)-4-[(4-isopropoxyphenyl)methyl]-5-methyl-1-phenyl-1H-pyrazole
—— (1R)-1-(3-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine —— C19H18ClF2N3O2
(1R)-1-(3-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine
—— (3-fluoro-4-methylphenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone —— C23H24F2N4O2
(3-fluoro-4-methylphenyl)-[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]methanone
—— N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methyl-1-[(2R)-oxolan-2-yl]methanamine —— C16H19F2N3O3
N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methyl-1-[(2R)-oxolan-2-yl]methanamine
—— N-[(1S)-1-(4-chlorophenyl)ethyl]-N-methyl-2-[methyl-[(1-phenylpyrazol-4-yl)methyl]amino]acetamide —— C22H25ClN4O
N-[(1S)-1-(4-chlorophenyl)ethyl]-N-methyl-2-[methyl-[(1-phenylpyrazol-4-yl)methyl]amino]acetamide
—— N-[2-[(2R)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]ethyl]methanesulfonamide —— C18H24F2N4O4S
N-[2-[(2R)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]ethyl]methanesulfonamide
—— (1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2,5-difluorophenyl)-N-methylethanamine —— C19H17F4N3O2
(1R)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2,5-difluorophenyl)-N-methylethanamine
—— (1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-fluorophenyl)-N-methylethanamine —— C19H18F3N3O2
(1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2-fluorophenyl)-N-methylethanamine
—— 1,5-dimethyl-4-[[methyl-[(2S)-1-pyrazin-2-ylpropan-2-yl]amino]methyl]-2-phenylpyrazol-3-one —— C20H25N5O
1,5-dimethyl-4-[[methyl-[(2S)-1-pyrazin-2-ylpropan-2-yl]amino]methyl]-2-phenylpyrazol-3-one
—— 3-[2-(difluoromethoxy)phenyl]-5-[[(2S)-2-(2-phenylethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C22H23F2N3O2
3-[2-(difluoromethoxy)phenyl]-5-[[(2S)-2-(2-phenylethyl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— N-ethyl-N-[(2R)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide —— C19H25N3O3S
N-ethyl-N-[(2R)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
—— N-ethyl-N-[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide —— C19H25N3O3S
N-ethyl-N-[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
—— 3-(4-chlorophenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-4-amine —— C17H15ClN4S
3-(4-chlorophenyl)-5-[(Z)-3-phenylprop-2-enyl]sulfanyl-1,2,4-triazol-4-amine
—— N-[(1R)-1-(4-chlorophenyl)ethyl]-N-methyl-2-[methyl-[(1-phenylpyrazol-4-yl)methyl]amino]acetamide —— C22H25ClN4O
N-[(1R)-1-(4-chlorophenyl)ethyl]-N-methyl-2-[methyl-[(1-phenylpyrazol-4-yl)methyl]amino]acetamide
—— N-methyl-N-[(1R)-1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide —— C16H17N5OS
N-methyl-N-[(1R)-1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
—— (3R)-3-benzyl-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one —— C21H20N4O2
(3R)-3-benzyl-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one
—— (3S)-8-[[1-(2-fluorophenyl)pyrazol-4-yl]methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol —— C18H22FN3O2
(3S)-8-[[1-(2-fluorophenyl)pyrazol-4-yl]methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
—— 2-[(2S)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]ethanol —— C18H24FN3O
2-[(2S)-1-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]pyrrolidin-2-yl]ethanol
—— N-[[1-(2,4-dichlorophenyl)-7-fluoro-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]azepan-1-amine —— C23H23Cl2FN4S
N-[[1-(2,4-dichlorophenyl)-7-fluoro-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]azepan-1-amine
—— N-methyl-N-[(1R)-1-(3-phenyl-1H-pyrazol-5-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide —— C19H18N6O
N-methyl-N-[(1R)-1-(3-phenyl-1H-pyrazol-5-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
—— 5-[1-(imidazol-1-ylmethyl)cyclopropyl]-3-[(3S)-oxolan-3-yl]-1-phenyl-1,2,4-triazole —— C19H21N5O
5-[1-(imidazol-1-ylmethyl)cyclopropyl]-3-[(3S)-oxolan-3-yl]-1-phenyl-1,2,4-triazole
—— N-(2-morpholin-4-ylethyl)-3-phenyl-1,4-dihydroindeno[1,2-c]pyrazol-6-amine;trihydrochloride —— C22H27Cl3N4O
N-(2-morpholin-4-ylethyl)-3-phenyl-1,4-dihydroindeno[1,2-c]pyrazol-6-amine;trihydrochloride
—— 5-[1-(imidazol-1-ylmethyl)cyclopropyl]-3-[(3R)-oxolan-3-yl]-1-phenyl-1,2,4-triazole —— C19H21N5O
5-[1-(imidazol-1-ylmethyl)cyclopropyl]-3-[(3R)-oxolan-3-yl]-1-phenyl-1,2,4-triazole
—— tert-butyl N-[2-[4-(6-methoxynaphthalen-2-yl)-5-phenyl-1H-imidazol-2-yl]-2-methylpropyl]carbamate —— C29H33N3O3
tert-butyl N-[2-[4-(6-methoxynaphthalen-2-yl)-5-phenyl-1H-imidazol-2-yl]-2-methylpropyl]carbamate
—— N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-[[(3S)-oxolan-3-yl]methyl]ethanamine —— C23H27N3O
N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-[[(3S)-oxolan-3-yl]methyl]ethanamine
—— N-[2-[[4-(1,3-benzoxazol-2-yl)phenyl]methoxy]ethyl]-2-[3-(4-methylphenyl)prop-2-ynoxy]ethanamine —— C28H28N2O3
N-[2-[[4-(1,3-benzoxazol-2-yl)phenyl]methoxy]ethyl]-2-[3-(4-methylphenyl)prop-2-ynoxy]ethanamine
—— (1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2,5-difluorophenyl)-N-methylethanamine —— C19H17F4N3O2
(1S)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1-(2,5-difluorophenyl)-N-methylethanamine
—— (1S)-1-(2-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine —— C19H18ClF2N3O2
(1S)-1-(2-chlorophenyl)-N-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylethanamine
—— ethyl (Z)-4-[(4R,7R)-4-methyl-3-phenyl-7-propan-2-yl-4,5,6,7-tetrahydroindazol-1-yl]-4-oxobut-2-enoate —— C23H28N2O3
ethyl (Z)-4-[(4R,7R)-4-methyl-3-phenyl-7-propan-2-yl-4,5,6,7-tetrahydroindazol-1-yl]-4-oxobut-2-enoate