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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(3R,5R)-1-azabicyclo[3.2.1]octan-3-yl]-4-(3-methylphenyl)pyrazole-1-carboxamide —— C18H22N4O
N-[(3R,5R)-1-azabicyclo[3.2.1]octan-3-yl]-4-(3-methylphenyl)pyrazole-1-carboxamide
—— (1-benzylpyrazol-4-yl)-[(3S)-3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]methanone —— C16H16F3N3O2
(1-benzylpyrazol-4-yl)-[(3S)-3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]methanone
—— 6,8-difluoro-2-(2-fluorophenyl)-1H-pyrazolo[4,3-c]quinolin-3-one —— C16H8F3N3O
6,8-difluoro-2-(2-fluorophenyl)-1H-pyrazolo[4,3-c]quinolin-3-one
—— 1-[[5-[2-(Diaminomethylideneamino)-1,3-thiazol-4-yl]furan-2-yl]methyl]-3-methylthiourea —— C11H14N6OS2
1-[[5-[2-(Diaminomethylideneamino)-1,3-thiazol-4-yl]furan-2-yl]methyl]-3-methylthiourea
—— (E)-N-[4-methoxy-3-(tetrazol-1-yl)phenyl]-2-methylpent-2-enamide —— C14H17N5O2
(E)-N-[4-methoxy-3-(tetrazol-1-yl)phenyl]-2-methylpent-2-enamide
—— Thiazolyl derivative, 3 —— C18H22N2OS
Thiazolyl derivative, 3
—— 1,3-Dimethyl-4-(5-methylfuran-2-yl)imidazol-1-ium;iodide —— C10H13IN2O
1,3-Dimethyl-4-(5-methylfuran-2-yl)imidazol-1-ium;iodide
—— Ethyl 8-chloro-2-methyl-5-oxidopyrazolo[5,1-c][1,2,4]benzotriazin-5-ium-3-carboxylate —— C13H11ClN4O3
Ethyl 8-chloro-2-methyl-5-oxidopyrazolo[5,1-c][1,2,4]benzotriazin-5-ium-3-carboxylate
—— 1,3-Dimethyl-4-(5-methylfuran-2-yl)imidazol-1-ium —— C10H13N2O+
1,3-Dimethyl-4-(5-methylfuran-2-yl)imidazol-1-ium
—— 1-<5-(2-hydroxyethylamino)-3-p-chlorophenyl-1H-pyrazol-4-yl>-1,2,4-triazole —— C13H13ClN6O
1-<5-(2-hydroxyethylamino)-3-p-chlorophenyl-1H-pyrazol-4-yl>-1,2,4-triazole
—— 3-methoxy-2-(3'-methoxyphenyl)-6-methylthioimidazo<1,2-b>pyridazine —— C15H15N3O2S
3-methoxy-2-(3'-methoxyphenyl)-6-methylthioimidazo<1,2-b>pyridazine
—— 5-[(3-fluorophenyl)methyl]-2-phenyl-5H-imidazo[4,5-c]pyridine —— C19H14FN3
5-[(3-fluorophenyl)methyl]-2-phenyl-5H-imidazo[4,5-c]pyridine
—— (1-tert-butylpyrazol-4-yl)-[(3S)-3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]methanone —— C13H18F3N3O2
(1-tert-butylpyrazol-4-yl)-[(3S)-3-hydroxy-3-(trifluoromethyl)pyrrolidin-1-yl]methanone
—— [5-(4-Chloro-phenyl)-4-nitroso-2H-pyrazol-3-yl]-phenyl-amine —— C15H11ClN4O
[5-(4-Chloro-phenyl)-4-nitroso-2H-pyrazol-3-yl]-phenyl-amine
—— (Z)-4-[1-cyclohexyl-2-(imidazol-1-yl)ethylidene]aminoxybutanoic acid —— C15H23N3O3
(Z)-4-[1-cyclohexyl-2-(imidazol-1-yl)ethylidene]aminoxybutanoic acid
—— [(3R,5S)-3,5-dimethylmorpholin-4-yl]-[4-(1,3-oxazol-5-yl)phenyl]methanone —— C16H18N2O3
[(3R,5S)-3,5-dimethylmorpholin-4-yl]-[4-(1,3-oxazol-5-yl)phenyl]methanone
—— 2-(4-Chloro-phenyl)-imidazo[1,2-a]quinoxalin-4-ylamine —— C16H11ClN4
2-(4-Chloro-phenyl)-imidazo[1,2-a]quinoxalin-4-ylamine
—— (1R)-1-(3-fluoro-4-methoxyphenyl)-2-(2-phenylimidazol-1-yl)ethanol —— C18H17FN2O2
(1R)-1-(3-fluoro-4-methoxyphenyl)-2-(2-phenylimidazol-1-yl)ethanol
—— [(3S,5S)-3,5-dimethylmorpholin-4-yl]-[4-(1,3-oxazol-5-yl)phenyl]methanone —— C16H18N2O3
[(3S,5S)-3,5-dimethylmorpholin-4-yl]-[4-(1,3-oxazol-5-yl)phenyl]methanone
—— [(3R,5R)-3,5-dimethylmorpholin-4-yl]-(4-imidazol-1-ylphenyl)methanone —— C16H19N3O2
[(3R,5R)-3,5-dimethylmorpholin-4-yl]-(4-imidazol-1-ylphenyl)methanone
—— (1S)-1-(3-fluoro-4-methoxyphenyl)-2-(2-phenylimidazol-1-yl)ethanol —— C18H17FN2O2
(1S)-1-(3-fluoro-4-methoxyphenyl)-2-(2-phenylimidazol-1-yl)ethanol
—— [(3R,5S)-3,5-dimethylmorpholin-4-yl]-(4-imidazol-1-ylphenyl)methanone —— C16H19N3O2
[(3R,5S)-3,5-dimethylmorpholin-4-yl]-(4-imidazol-1-ylphenyl)methanone
—— 1-[(Z)-(4-chlorophenyl)methylideneamino]-4-pyridin-2-ylimidazol-2-amine —— C15H12ClN5
1-[(Z)-(4-chlorophenyl)methylideneamino]-4-pyridin-2-ylimidazol-2-amine
—— [(3S,5S)-3,5-dimethylmorpholin-4-yl]-(4-imidazol-1-ylphenyl)methanone —— C16H19N3O2
[(3S,5S)-3,5-dimethylmorpholin-4-yl]-(4-imidazol-1-ylphenyl)methanone
—— N-[(1S,2R,4R)-7-azabicyclo[2.2.1]heptan-2-yl]-4-(4-methylphenyl)pyrazole-1-carboxamide —— C17H20N4O
N-[(1S,2R,4R)-7-azabicyclo[2.2.1]heptan-2-yl]-4-(4-methylphenyl)pyrazole-1-carboxamide
—— [(3R,5R)-3,5-dimethylmorpholin-4-yl]-[4-(1,3-oxazol-5-yl)phenyl]methanone —— C16H18N2O3
[(3R,5R)-3,5-dimethylmorpholin-4-yl]-[4-(1,3-oxazol-5-yl)phenyl]methanone
—— 2-[(Z)-2-(2-tert-butyl-1,3-thiazol-5-yl)ethenyl]-N-methyl-1,3-thiazole-5-carboxamide —— C14H17N3OS2
2-[(Z)-2-(2-tert-butyl-1,3-thiazol-5-yl)ethenyl]-N-methyl-1,3-thiazole-5-carboxamide
—— (Z)-N-[3-(1-ethyltetrazol-5-yl)phenyl]-3-pyridin-3-ylprop-2-enamide —— C17H16N6O
(Z)-N-[3-(1-ethyltetrazol-5-yl)phenyl]-3-pyridin-3-ylprop-2-enamide
—— N-[(1R)-1-(2-chloro-4-fluorophenyl)ethyl]-1-methylpyrazole-4-carboxamide —— C13H13ClFN3O
N-[(1R)-1-(2-chloro-4-fluorophenyl)ethyl]-1-methylpyrazole-4-carboxamide
—— 2-[(4R)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C30H28ClFN4O2S
2-[(4R)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H32N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2S)-butan-2-yl]acetamide —— C32H32N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(2S)-butan-2-yl]acetamide
—— N-[(1R)-cyclohex-3-en-1-yl]-2-(4-methylpyrazol-1-yl)acetamide —— C12H17N3O
N-[(1R)-cyclohex-3-en-1-yl]-2-(4-methylpyrazol-1-yl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C32H32N4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— N-[(1S)-1-(2-chloro-4-fluorophenyl)ethyl]-1-methylpyrazole-4-carboxamide —— C13H13ClFN3O
N-[(1S)-1-(2-chloro-4-fluorophenyl)ethyl]-1-methylpyrazole-4-carboxamide
—— 2-[(4R)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H26ClFN4O3S
2-[(4R)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— methyl (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-2-pyridin-4-ylprop-2-enoate —— C16H18N2O2S
methyl (Z)-3-(2-tert-butyl-1,3-thiazol-5-yl)-2-pyridin-4-ylprop-2-enoate
—— 2-[(4S)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C30H28ClFN4O2S
2-[(4S)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— (4-pyrazol-1-ylphenyl) (Z)-2-(2-chlorophenyl)ethenesulfonate —— C17H13ClN2O3S
(4-pyrazol-1-ylphenyl) (Z)-2-(2-chlorophenyl)ethenesulfonate
—— 2-[(4S)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H26ClFN4O3S
2-[(4S)-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— (4S)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H34N4O3S
(4S)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H36N4O3S
2-[(4R)-3-tert-butyl-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-1-(4-fluorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C32H31FN4O3S
2-[(4S)-1-(4-fluorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H32N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C35H33N5O3S
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C31H38N4O5S
2-[(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C32H40N4O4S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-4-(2-chlorophenyl)-1-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C29H32ClFN4O3S
2-[(4S)-3-tert-butyl-4-(2-chlorophenyl)-1-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C27H30ClFN4O3S
2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— N-cyclopropyl-2-[(4S)-4-(2-methoxyphenyl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H30N4O3S
N-cyclopropyl-2-[(4S)-4-(2-methoxyphenyl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide