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—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(2-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27FN4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(2-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(cyclobutanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C21H24N2O2S
(6S)-1-(cyclobutanecarbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(2-chlorophenyl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H24ClN3O
(6S)-1-[(2-chlorophenyl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-fluorobenzoyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H22FN3O2
(6S)-1-(3-fluorobenzoyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25FN4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-(2-fluorobenzoyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H18FN3O2
6-[1-(2-fluorobenzoyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[(3R)-1-(2-fluorobenzoyl)piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C20H18FN3O2
6-[(3R)-1-(2-fluorobenzoyl)piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[2-[[(2S)-oxolan-2-yl]methoxy]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H25N3O4
6-[1-[2-[[(2S)-oxolan-2-yl]methoxy]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-cyclopentyl-2-[(3S)-1-(2-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27FN4O2
6-cyclopentyl-2-[(3S)-1-(2-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25FN4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O3
6-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H19N3O4
6-[1-(1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[(3S)-1-(2-fluorobenzoyl)piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C20H18FN3O2
6-[(3S)-1-(2-fluorobenzoyl)piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(imidazo[1,2-a]pyrimidine-2-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H18N6O2
6-[1-(imidazo[1,2-a]pyrimidine-2-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C17H16N4O2S
6-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(2-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-(cyclohexylmethyl)-2-[(2R)-1-(2-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3S)-1-[(2R)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O3
6-[(3S)-1-[(2R)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-cyclopentyl-2-[(3R)-1-(2-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27FN4O2
6-cyclopentyl-2-[(3R)-1-(2-fluorobenzoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[2-[[(2R)-oxolan-2-yl]methoxy]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H25N3O4
6-[1-[2-[[(2R)-oxolan-2-yl]methoxy]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[3-[(2R)-oxolan-2-yl]propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H25N3O3
6-[1-[3-[(2R)-oxolan-2-yl]propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[(3R)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C21H20FN3O2
6-[(3R)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(1,2-oxazole-5-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C17H16N4O3
6-[1-(1,2-oxazole-5-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H25N3O3
6-[1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[(3R)-1-[(2R)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O3
6-[(3R)-1-[(2R)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C23H22N6O3
6-[1-[3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6R)-8-[(2,4-dichlorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one —— C17H15Cl2N3O
(6R)-8-[(2,4-dichlorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one
—— 6-[1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H19F2N3O2
6-[1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O3
6-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(2-cyclohexylacetyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H27N3O2
6-[1-(2-cyclohexylacetyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[(3S)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C21H20FN3O2
6-[(3S)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-fluoro-N-[2-[3-[(3S)-pyrrolidin-3-yl]pyrazolo[3,4-b]pyridin-1-yl]ethyl]-1H-indole-2-carboxamide —— C21H21FN6O
6-fluoro-N-[2-[3-[(3S)-pyrrolidin-3-yl]pyrazolo[3,4-b]pyridin-1-yl]ethyl]-1H-indole-2-carboxamide
—— 6-[1-[3-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C23H22N6O3
6-[1-[3-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(thiophene-2-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C18H17N3O2S
6-[1-(thiophene-2-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[(1S)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H23N3O2
6-[1-[(1S)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H23N3O2
6-[1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[(1R)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H23N3O2
6-[1-[(1R)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H20FN3O2
6-[1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-Fluoro-2-piperidin-4-ylquinolin-3-amine —— C14H16FN3
6-Fluoro-2-piperidin-4-ylquinolin-3-amine
—— 6-[(3S)-1-[(2S)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O3
6-[(3S)-1-[(2S)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H24N4O2
6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-Fluoro-2-piperidin-4-ylquinoline-3-carboxamide —— C15H16FN3O
6-Fluoro-2-piperidin-4-ylquinoline-3-carboxamide
—— (6-amino-2,3-dihydro-1,4-benzodioxin-7-yl)-[(3S)-3-(5-fluorobenzimidazol-1-yl)piperidin-1-yl]methanone —— C21H21FN4O3
(6-amino-2,3-dihydro-1,4-benzodioxin-7-yl)-[(3S)-3-(5-fluorobenzimidazol-1-yl)piperidin-1-yl]methanone
—— 6-[(R)-[1-(4,5-dichloro-1,2-thiazole-3-carbonyl)piperidin-4-yl]-hydroxymethyl]-4H-1,4-benzoxazin-3-one —— C18H17Cl2N3O4S
6-[(R)-[1-(4,5-dichloro-1,2-thiazole-3-carbonyl)piperidin-4-yl]-hydroxymethyl]-4H-1,4-benzoxazin-3-one
—— 6-Ethyl-2-(5-methyl-2-furyl)quinoline-4-carboxylic acid —— C17H15NO3
6-Ethyl-2-(5-methyl-2-furyl)quinoline-4-carboxylic acid
—— 6-Fluoro-4-(3-methyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)-2-{5-[4-(propan-2-yl)phenyl]furan-2-yl}quinoline —— C26H20FN5OS
6-Fluoro-4-(3-methyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)-2-{5-[4-(propan-2-yl)phenyl]furan-2-yl}quinoline
—— 6-Bromo-2-[2-(4-ethoxyphenyl)ethenyl]-3,1-benzoxazin-4-one —— C18H14BrNO3
6-Bromo-2-[2-(4-ethoxyphenyl)ethenyl]-3,1-benzoxazin-4-one
—— 6-Methoxy-1-naphthalen-1-yl-1,2,3,4-tetrahydroisoquinoline —— C20H19NO
6-Methoxy-1-naphthalen-1-yl-1,2,3,4-tetrahydroisoquinoline
—— 6-(3-fluoropropylsulfanyl)-7H-purine —— C8H9FN4S
6-(3-fluoropropylsulfanyl)-7H-purine
—— 6-chloro-2-(3-chlorophenyl)-7-methyl-2,3-dihydro-1H-indole —— C15H13Cl2N
6-chloro-2-(3-chlorophenyl)-7-methyl-2,3-dihydro-1H-indole
—— 6-fluoro-N-[2-[3-[(3R)-pyrrolidin-3-yl]pyrazolo[3,4-b]pyridin-1-yl]ethyl]-1H-indole-2-carboxamide —— C21H21FN6O
6-fluoro-N-[2-[3-[(3R)-pyrrolidin-3-yl]pyrazolo[3,4-b]pyridin-1-yl]ethyl]-1H-indole-2-carboxamide