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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-5-one —— C25H29FN2O3
(6R)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O3S
(6S)-4-ethyl-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N4O3
(6S)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H34N4O2
(6R)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(1S)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C28H34N2O3
(6S)-1-[(1S)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-[(5-tert-butyl-1H-pyrazol-4-yl)methyl]-4-ethyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H35N5O
(6S)-1-[(5-tert-butyl-1H-pyrazol-4-yl)methyl]-4-ethyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(5-hydroxypyridine-3-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6R)-4-ethyl-1-(5-hydroxypyridine-3-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C25H29N5O3
(6R)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-fluorobenzoyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H26FN3O2
(6R)-4-ethyl-1-(3-fluorobenzoyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-methoxypropanoyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H29N3O3
(6R)-4-ethyl-1-(3-methoxypropanoyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[2-(3-fluorophenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H28FN3O2
(6R)-4-ethyl-1-[2-(3-fluorophenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-phenylpropanoyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H31N3O2
(6R)-4-ethyl-1-(3-phenylpropanoyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one —— C28H31N3O2
(6S)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O2
(6R)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(pyridine-2-carbonyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N4O2
(6S)-4-ethyl-1-(pyridine-2-carbonyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(pyridine-2-carbonyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N4O2
(6R)-4-ethyl-1-(pyridine-2-carbonyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(2S)-oxolane-2-carbonyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O3
(6S)-4-ethyl-1-[(2S)-oxolane-2-carbonyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(1,5-dimethylpyrazole-4-carbonyl)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H32N4O2
(6R)-1-(1,5-dimethylpyrazole-4-carbonyl)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O3
(6R)-4-ethyl-1-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopropylmethyl)-4-ethyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H29N3O
(6S)-1-(cyclopropylmethyl)-4-ethyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(2-methoxyacetyl)-1,4-diazepan-5-one —— C23H27FN2O3
(6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(2-methoxyacetyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-methylpyrazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(2-methylpyrazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one —— C27H29N3O2
(6S)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[2-(4-methylphenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H31N3O2
(6R)-4-ethyl-1-[2-(4-methylphenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-5-one —— C25H29FN2O3
(6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-5-one
—— (6S)-1-(1,5-dimethylpyrazole-4-carbonyl)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29FN4O2
(6S)-1-(1,5-dimethylpyrazole-4-carbonyl)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N3O3
(6R)-4-ethyl-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6R)-4-ethyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-ethyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H31N3O2
(6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-ethyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2
(6R)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one —— C28H36N2O3
(6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H30N4O2
(6R)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one —— C26H30N4O2
(6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[2-(3-methylphenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H31N3O2
(6S)-4-ethyl-1-[2-(3-methylphenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C27H29N3O2
(6S)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2R)-oxolane-2-carbonyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H30N2O3
(6R)-4-ethyl-1-[(2R)-oxolane-2-carbonyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6R)-4-ethyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C26H26FN3O2
(6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[3-[(2R)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one —— C28H36N2O3
(6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[3-[(2R)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclopentanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H34N2O3
(6R)-1-(cyclopentanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2
(6R)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(1R)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C28H34N2O3
(6R)-1-[(1R)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-phenoxyacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6S)-4-ethyl-1-(2-phenoxyacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[2-(2-oxopyrimidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H28N4O3
(6S)-4-ethyl-1-[2-(2-oxopyrimidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Chloro-3-(4,5-dihydro-1,3-thiazol-2-ylsulfanyl)-4-phenylquinolin-2-ol —— C18H13ClN2OS2
6-Chloro-3-(4,5-dihydro-1,3-thiazol-2-ylsulfanyl)-4-phenylquinolin-2-ol
—— (6S)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6S)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one