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—— 6-[(2S)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-pyrrolidin-1-ylethyl)-1H-quinoline-4-carboxamide —— C22H30N4O4S
6-[(2S)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-pyrrolidin-1-ylethyl)-1H-quinoline-4-carboxamide
—— 6-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-2-oxo-N-(thiophen-2-ylmethyl)-1H-quinoline-4-carboxamide —— C22H25N3O4S2
6-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-2-oxo-N-(thiophen-2-ylmethyl)-1H-quinoline-4-carboxamide
—— 6-[butyl(ethyl)sulfamoyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-oxo-1H-quinoline-4-carboxamide —— C24H36N4O4S
6-[butyl(ethyl)sulfamoyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-Bromo-3-{[4-(4-fluorophenyl)piperazinyl]carbonyl}-8-methoxychromen-2-one —— C21H18BrFN2O4
6-Bromo-3-{[4-(4-fluorophenyl)piperazinyl]carbonyl}-8-methoxychromen-2-one
—— 6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-N-[2-(4-methylphenyl)ethyl]-2-oxo-1H-quinoline-4-carboxamide —— C26H31N3O4S
6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-N-[2-(4-methylphenyl)ethyl]-2-oxo-1H-quinoline-4-carboxamide
—— (6R)-4-amino-6-(2-fluorophenyl)-11,13-dimethyl-3-oxa-8-thia-10-azatricyclo[7.4.0.02,7]trideca-1(9),2(7),4,10,12-pentaene-5-carbonitrile —— C19H14FN3OS
(6R)-4-amino-6-(2-fluorophenyl)-11,13-dimethyl-3-oxa-8-thia-10-azatricyclo[7.4.0.02,7]trideca-1(9),2(7),4,10,12-pentaene-5-carbonitrile
—— 6-[(2R)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-pyrrolidin-1-ylethyl)-1H-quinoline-4-carboxamide —— C22H30N4O4S
6-[(2R)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-pyrrolidin-1-ylethyl)-1H-quinoline-4-carboxamide
—— 6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-2-oxo-N-(thiophen-2-ylmethyl)-1H-quinoline-4-carboxamide —— C22H25N3O4S2
6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-2-oxo-N-(thiophen-2-ylmethyl)-1H-quinoline-4-carboxamide
—— 6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-N-[(4-fluorophenyl)methyl]-2-oxo-1H-quinoline-4-carboxamide —— C24H26FN3O4S
6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-N-[(4-fluorophenyl)methyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-N-[(4-methylphenyl)methyl]-2-oxo-1H-quinoline-4-carboxamide —— C25H29N3O4S
6-[(2R)-2-ethylpiperidin-1-yl]sulfonyl-N-[(4-methylphenyl)methyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-N-[(4-methylphenyl)methyl]-2-oxo-1H-quinoline-4-carboxamide —— C25H29N3O4S
6-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-N-[(4-methylphenyl)methyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(2S)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-pyrrolidin-1-ylpropyl)-1H-quinoline-4-carboxamide —— C23H32N4O4S
6-[(2S)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-pyrrolidin-1-ylpropyl)-1H-quinoline-4-carboxamide
—— 6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(2S)-4-phenylbutan-2-yl]-1H-quinoline-4-carboxamide —— C26H31N3O4S
6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(2S)-4-phenylbutan-2-yl]-1H-quinoline-4-carboxamide
—— 6-(azepan-1-ylsulfonyl)-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-2-oxo-1H-quinoline-4-carboxamide —— C26H38N4O4S
6-(azepan-1-ylsulfonyl)-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-Bromo-3-[2-(1-methylimidazol-2-yl)sulfanylacetyl]chromen-2-one —— C15H11BrN2O3S
6-Bromo-3-[2-(1-methylimidazol-2-yl)sulfanylacetyl]chromen-2-one
—— (6Z,7S)-7-hydroxy-4,9-dimethoxy-6-[(4-methylanilino)methylidene]-7-(trifluoromethyl)furo[3,2-g]chromen-5-one —— C22H18F3NO6
(6Z,7S)-7-hydroxy-4,9-dimethoxy-6-[(4-methylanilino)methylidene]-7-(trifluoromethyl)furo[3,2-g]chromen-5-one
—— 6-Bromo-4-[(dimethylazaniumyl)methyl]-3-ethoxycarbonyl-1-phenyl-2-(pyrrolidin-1-ylmethyl)indol-5-olate —— C25H30BrN3O3
6-Bromo-4-[(dimethylazaniumyl)methyl]-3-ethoxycarbonyl-1-phenyl-2-(pyrrolidin-1-ylmethyl)indol-5-olate
—— (6Z)-2,6-bis[[4-(dimethylamino)phenyl]methylidene]cyclohexan-1-one —— C24H28N2O
(6Z)-2,6-bis[[4-(dimethylamino)phenyl]methylidene]cyclohexan-1-one
—— (6Z,7R)-7-hydroxy-4,9-dimethoxy-6-[(4-methylanilino)methylidene]-7-(trifluoromethyl)furo[3,2-g]chromen-5-one —— C22H18F3NO6
(6Z,7R)-7-hydroxy-4,9-dimethoxy-6-[(4-methylanilino)methylidene]-7-(trifluoromethyl)furo[3,2-g]chromen-5-one
—— 6-imino-N-[(4-methylphenyl)methyl]-2-oxo-7-(prop-2-en-1-yl)-1,7,9-triazatricyclo[8.4.0.0^{3,8}]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C23H21N5O2
6-imino-N-[(4-methylphenyl)methyl]-2-oxo-7-(prop-2-en-1-yl)-1,7,9-triazatricyclo[8.4.0.0^{3,8}]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6bR,8S,9aS)-8-methyl-9-phenyl-8,9a-dihydro-6bH-acenaphthyleno[1,2-d][1,3]oxazole —— C20H17NO
(6bR,8S,9aS)-8-methyl-9-phenyl-8,9a-dihydro-6bH-acenaphthyleno[1,2-d][1,3]oxazole
—— 6-(3,5-Dimethylphenyl)-3-(3-methylphenyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C18H16N4S
6-(3,5-Dimethylphenyl)-3-(3-methylphenyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6S)-6-tert-butyl-N-(3-methylphenyl)-2-[(2-morpholin-4-ylacetyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H35N3O3S
(6S)-6-tert-butyl-N-(3-methylphenyl)-2-[(2-morpholin-4-ylacetyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— [6-[(5,6-dimethyl-1H-benzimidazol-2-yl)methyl]pyridin-2-yl]methanol —— C16H17N3O
[6-[(5,6-dimethyl-1H-benzimidazol-2-yl)methyl]pyridin-2-yl]methanol
—— 6-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-pyridin-4-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C16H11N5O2S
6-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-pyridin-4-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6‐oxo‐2‐((2‐oxo‐2‐phenylethyl)thio)‐4‐(p‐tolyl)‐1,6‐dihydropyrimidine‐5‐carbonitrile —— C20H15N3O2S
6‐oxo‐2‐((2‐oxo‐2‐phenylethyl)thio)‐4‐(p‐tolyl)‐1,6‐dihydropyrimidine‐5‐carbonitrile
—— (6R)-N-(3,4-dichlorophenyl)-6-(3-methoxyphenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C29H27Cl2N3O3
(6R)-N-(3,4-dichlorophenyl)-6-(3-methoxyphenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6'aS)-2'-chloro-2,2-dimethylspiro[1,3-dioxane-5,6'-6a,7,8,9,10,11-hexahydro-5H-azepino[1,2-a]quinoline]-4,6-dione —— C19H22ClNO4
(6'aS)-2'-chloro-2,2-dimethylspiro[1,3-dioxane-5,6'-6a,7,8,9,10,11-hexahydro-5H-azepino[1,2-a]quinoline]-4,6-dione
—— (6'aR)-2'-chloro-2,2-dimethylspiro[1,3-dioxane-5,6'-6a,7,8,9,10,11-hexahydro-5H-azepino[1,2-a]quinoline]-4,6-dione —— C19H22ClNO4
(6'aR)-2'-chloro-2,2-dimethylspiro[1,3-dioxane-5,6'-6a,7,8,9,10,11-hexahydro-5H-azepino[1,2-a]quinoline]-4,6-dione
—— 6-chloro-N'-cyclooctylidene-2-methylimidazo[1,2-a]pyridine-3-carbohydrazide —— C17H21ClN4O
6-chloro-N'-cyclooctylidene-2-methylimidazo[1,2-a]pyridine-3-carbohydrazide
—— 6-methyl-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]sulfonyl]-1H-pyrimidine-2,4-dione —— C16H18N4O5S
6-methyl-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]sulfonyl]-1H-pyrimidine-2,4-dione
—— 6-chloro-3-[(3R)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C32H33ClN4O3
6-chloro-3-[(3R)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— (6S)-3-amino-6-tert-butyl-N-cyclohexyl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxamide —— C22H31N3OS
(6S)-3-amino-6-tert-butyl-N-cyclohexyl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxamide
—— 6-chloro-3-[(3S)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C31H30ClFN4O2
6-chloro-3-[(3S)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— 6-[2-[(5S)-1-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H15ClF3N3O2S
6-[2-[(5S)-1-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— (6R)-3-chloro-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-5,6-dihydrobenzo[b][1]benzothiepin-6-amine —— C21H25ClN2S
(6R)-3-chloro-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-5,6-dihydrobenzo[b][1]benzothiepin-6-amine
—— 6-chloro-3-[(3S)-3-[4-[hydroxy(diphenyl)methyl]piperidine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C39H38ClN3O3
6-chloro-3-[(3S)-3-[4-[hydroxy(diphenyl)methyl]piperidine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— 6-[2-[(5S)-5-hydroxy-1-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C22H18F3N3O2S
6-[2-[(5S)-5-hydroxy-1-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— (6S)-3-amino-6-tert-butyl-N-phenyl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxamide —— C22H25N3OS
(6S)-3-amino-6-tert-butyl-N-phenyl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxamide
—— 6-chloro-3-[(3S)-3-[4-[(2S)-oxolane-2-carbonyl]piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C30H33ClN4O4
6-chloro-3-[(3S)-3-[4-[(2S)-oxolane-2-carbonyl]piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— 6-(Morpholine-4-carbonyl)-2,3-diphenylquinoxaline —— C25H21N3O2
6-(Morpholine-4-carbonyl)-2,3-diphenylquinoxaline
—— 6-[2-[(5R)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H15F4N3O2S
6-[2-[(5R)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-chloro-3-[(3S)-3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C30H29ClN4O4
6-chloro-3-[(3S)-3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— (6R)-2-[(3S)-1-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]sulfanyl-6-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C27H23N3O3S
(6R)-2-[(3S)-1-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]sulfanyl-6-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— 6-[2-[(5S)-5-hydroxy-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C22H18F3N3O3S
6-[2-[(5S)-5-hydroxy-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— (6S)-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-5-(2-methylpropanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C34H37ClN2O4
(6S)-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-5-(2-methylpropanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-N-(3,4-dichlorophenyl)-6-(3-methoxyphenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C29H27Cl2N3O3
(6S)-N-(3,4-dichlorophenyl)-6-(3-methoxyphenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R,9S)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H29F3N2O3
(6R,9S)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[2-[(5R)-5-hydroxy-1-(4-phenyl-1,3-thiazol-2-yl)-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H16F3N3O2S
6-[2-[(5R)-5-hydroxy-1-(4-phenyl-1,3-thiazol-2-yl)-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-[2-[(5S)-1-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H15BrF3N3O2S
6-[2-[(5S)-1-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one