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—— (6R)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-(2-piperidin-1-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H38N6O3
(6R)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-(2-piperidin-1-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-[(4-chlorophenyl)methyl]-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O3
(6R)-5-[(4-chlorophenyl)methyl]-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-5-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3
(6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-5-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-6-N-cycloheptyl-5,6-dimethyl-2-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H35N5O3
(6S)-6-N-cycloheptyl-5,6-dimethyl-2-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-cyclohexyl-6-methyl-8-oxo-2-phenyl-7-(2-phenylethyl)-5H-[1,3]thiazolo[5,4-f][1,4]oxazepine-6-carboxamide —— C28H31N3O3S
(6R)-N-cyclohexyl-6-methyl-8-oxo-2-phenyl-7-(2-phenylethyl)-5H-[1,3]thiazolo[5,4-f][1,4]oxazepine-6-carboxamide
—— (6S)-5-[(4-ethylphenyl)methyl]-2-(furan-2-yl)-6-methyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H32N4O3
(6S)-5-[(4-ethylphenyl)methyl]-2-(furan-2-yl)-6-methyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-benzyl-2-tert-butyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3
(6S)-N-benzyl-2-tert-butyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-benzyl-2-tert-butyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3
(6R)-N-benzyl-2-tert-butyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-5,6-dimethyl-2-(morpholine-4-carbonyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C21H31N5O4
(6R)-N-cycloheptyl-5,6-dimethyl-2-(morpholine-4-carbonyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-6-methyl-8-oxo-2-phenyl-7-(2-phenylethyl)-5H-[1,3]thiazolo[5,4-f][1,4]oxazepine-6-carboxamide —— C28H31N3O3S
(6S)-N-cyclohexyl-6-methyl-8-oxo-2-phenyl-7-(2-phenylethyl)-5H-[1,3]thiazolo[5,4-f][1,4]oxazepine-6-carboxamide
—— (6S,9R)-6-(4-methoxyphenyl)-9-pyridin-3-yl-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one —— C20H18N6O2
(6S,9R)-6-(4-methoxyphenyl)-9-pyridin-3-yl-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one —— C22H21N5O2
(6S,9R)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-6-(4-methoxyphenyl)-9-pyridin-3-yl-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one —— C20H18N6O2
(6S,9S)-6-(4-methoxyphenyl)-9-pyridin-3-yl-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one —— C22H21N5O2
(6R,9R)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one —— C22H21N5O2
(6S,9S)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one
—— 6-[2-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-ylidene]-4-fluorocyclohexa-2,4-dien-1-one —— C18H11ClFN3O
6-[2-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-ylidene]-4-fluorocyclohexa-2,4-dien-1-one
—— 6-(4-Hydroxynaphthalen-1-yl)-9-methyl-2-(4-nitrophenyl)-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C33H24N2O7
6-(4-Hydroxynaphthalen-1-yl)-9-methyl-2-(4-nitrophenyl)-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— 6-(3-Bromo-4-hydroxy-5-methoxyphenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-9-methyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C32H27BrN4O10
6-(3-Bromo-4-hydroxy-5-methoxyphenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-9-methyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— 6-(2-Hydroxy-6-methoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindole-2-carboxamide —— C25H22N2O7
6-(2-Hydroxy-6-methoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindole-2-carboxamide
—— 6-Ethyl-2-[3-(4-methylphenyl)prop-2-enoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H24N2O2S
6-Ethyl-2-[3-(4-methylphenyl)prop-2-enoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-Bromo-2-(4-tert-butylphenyl)-4-[(3-methyl-1-piperidinyl)carbonyl]quinoline —— C26H29BrN2O
6-Bromo-2-(4-tert-butylphenyl)-4-[(3-methyl-1-piperidinyl)carbonyl]quinoline
—— 6-(3-bromo-4-hydroxy-5-methoxyphenyl)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2,6a-dimethyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H32BrClN4O6S
6-(3-bromo-4-hydroxy-5-methoxyphenyl)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2,6a-dimethyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-chloro-N-(4-fluorophenyl)-2-(furan-2-yl)imidazo[1,2-a]pyridin-3-amine —— C17H11ClFN3O
6-chloro-N-(4-fluorophenyl)-2-(furan-2-yl)imidazo[1,2-a]pyridin-3-amine
—— (6R,9S)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one —— C22H21N5O2
(6R,9S)-6-(4-methoxyphenyl)-9-(4-methylphenyl)-5,6,7,9-tetrahydro-4H-tetrazolo[5,1-b]quinazolin-8-one
—— (6S)-9,9-dimethyl-6-(4-methylphenyl)-7-oxo-N-propyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C26H31N3O2
(6S)-9,9-dimethyl-6-(4-methylphenyl)-7-oxo-N-propyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— 6-acetyl-2-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one —— C33H29N3O3S
6-acetyl-2-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one
—— 6-(3-chloro-4-hydroxy-5-methoxyphenyl)-2-(4-chlorophenyl)-8-(4-methylanilino)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H33Cl2N3O6
6-(3-chloro-4-hydroxy-5-methoxyphenyl)-2-(4-chlorophenyl)-8-(4-methylanilino)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6,7-Diethoxy-3-[(3-methoxyphenyl)methyl]-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one —— C20H22N2O4S
6,7-Diethoxy-3-[(3-methoxyphenyl)methyl]-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one
—— 6-(2-hydroxy-3-methylphenyl)-8-(4-methylanilino)-6a-phenyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H37N3O5
6-(2-hydroxy-3-methylphenyl)-8-(4-methylanilino)-6a-phenyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6,7-diethoxy-3-[2-(4-methylpiperidin-1-ium-1-yl)ethyl]-2-sulfanylidene-1H-quinazolin-4-one —— C20H30N3O3S+
6,7-diethoxy-3-[2-(4-methylpiperidin-1-ium-1-yl)ethyl]-2-sulfanylidene-1H-quinazolin-4-one
—— 6-tert-butyl-2-[(4-chlorobenzoyl)amino]-N-[2-(trifluoromethyl)phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C27H26ClF3N2O2S
6-tert-butyl-2-[(4-chlorobenzoyl)amino]-N-[2-(trifluoromethyl)phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[2-(2-hydroxyethoxy)phenyl]-2-[2-(4-hydroxyphenyl)ethyl]-8-(4-methylanilino)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C43H41N3O7
6-[2-(2-hydroxyethoxy)phenyl]-2-[2-(4-hydroxyphenyl)ethyl]-8-(4-methylanilino)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6S)-N-(3-ethoxypropyl)-6-(furan-2-yl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C23H27N3O4
(6S)-N-(3-ethoxypropyl)-6-(furan-2-yl)-7-oxo-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— 6,7-Diethoxy-3-[3-(pyrrolidin-1-YL)propyl]-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one —— C19H27N3O3S
6,7-Diethoxy-3-[3-(pyrrolidin-1-YL)propyl]-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one
—— 6,7-Diethoxy-3-[2-(4-methylphenyl)ethyl]-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one —— C21H24N2O3S
6,7-Diethoxy-3-[2-(4-methylphenyl)ethyl]-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one
—— 6-[3-(adamantane-1-carbonylamino)phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C33H38N4O3S
6-[3-(adamantane-1-carbonylamino)phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6R)-9,9-dimethyl-5-methylsulfonyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C20H22N2O3S2
(6R)-9,9-dimethyl-5-methylsulfonyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6,7-Diethoxy-3-(2-ethylhexyl)-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one —— C20H30N2O3S
6,7-Diethoxy-3-(2-ethylhexyl)-2-sulfanylidene-1,2,3,4-tetrahydroquinazolin-4-one
—— (6S)-5-(4-ethylphenyl)sulfonyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H24N2O4S
(6S)-5-(4-ethylphenyl)sulfonyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-N-(2-ethoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C26H25N3O3S
(6S)-N-(2-ethoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-9,9-dimethyl-7-oxo-N-propyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C23H27N3O2S
(6R)-9,9-dimethyl-7-oxo-N-propyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-6-(4-methoxyphenyl)-9,9-dimethyl-N-(2-methylphenyl)-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C30H31N3O3
(6R)-6-(4-methoxyphenyl)-9,9-dimethyl-N-(2-methylphenyl)-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-5-(benzenesulfonyl)-6-(furan-2-yl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H24N2O4S
(6R)-5-(benzenesulfonyl)-6-(furan-2-yl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-N-(3-ethoxypropyl)-9,9-dimethyl-7-oxo-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C25H31N3O3S
(6R)-N-(3-ethoxypropyl)-9,9-dimethyl-7-oxo-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R,9R)-9-(furan-2-yl)-6-(4-methoxyphenyl)-7-oxo-N-propyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C28H29N3O4
(6R,9R)-9-(furan-2-yl)-6-(4-methoxyphenyl)-7-oxo-N-propyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— 6-[2-(4-bromophenyl)-2-oxoethyl]sulfanyl-5-(2-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-one —— C20H15BrN4O2S
6-[2-(4-bromophenyl)-2-oxoethyl]sulfanyl-5-(2-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-one
—— (6S)-5-(benzenesulfonyl)-6-(furan-2-yl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H24N2O4S
(6S)-5-(benzenesulfonyl)-6-(furan-2-yl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-(3,4-dimethylphenyl)sulfonyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H24N2O4S
(6S)-5-(3,4-dimethylphenyl)sulfonyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-9,9-dimethyl-5-methylsulfonyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C20H22N2O3S2
(6S)-9,9-dimethyl-5-methylsulfonyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-(furan-2-yl)-5-(4-propan-2-ylphenyl)sulfonyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C26H26N2O4S
(6R)-6-(furan-2-yl)-5-(4-propan-2-ylphenyl)sulfonyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one