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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-ethylsulfonyl-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(4-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2S)-1-(4-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-ethylsulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C21H26N2O4S
(6R)-1-ethylsulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1-ethylsulfonyl-1,4-diazepan-5-one —— C20H22F2N2O3S
(6R)-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1-ethylsulfonyl-1,4-diazepan-5-one
—— (6S)-1-ethylsulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C21H26N2O4S
(6S)-1-ethylsulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-ethylsulfonyl-2-[(2S)-1-(2-pyridin-3-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H27N5O4S
6-ethylsulfonyl-2-[(2S)-1-(2-pyridin-3-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H25FN4O4S
6-ethylsulfonyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(2-ethoxybenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N2O3S
(6R)-1-(2-ethoxybenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1-ethylsulfonyl-1,4-diazepan-5-one —— C22H28N2O3S
(6S)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1-ethylsulfonyl-1,4-diazepan-5-one
—— 6-ethylsulfonyl-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H25FN4O4S
6-ethylsulfonyl-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H25FN4O4S
6-ethylsulfonyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1-ethylsulfonyl-1,4-diazepan-5-one —— C22H28N2O3S
(6R)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1-ethylsulfonyl-1,4-diazepan-5-one
—— 6-(cyclohexanecarbonyl)-2-[(2S)-1-ethylsulfonylpiperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H32N4O4S
6-(cyclohexanecarbonyl)-2-[(2S)-1-ethylsulfonylpiperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-[(6-methylpyridin-2-yl)methyl]-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H32N4O
(6R)-1-[(6-methylpyridin-2-yl)methyl]-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N3O2
(6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(pyridin-4-ylmethyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6R)-4-propyl-1-(pyridin-4-ylmethyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1-methylimidazole-2-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(1-methylimidazole-2-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6S)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N3O2
(6S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N3O2
(6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[[3-[(2,4-Dichlorophenyl)methoxy]phenyl]methylidene]-5-imino-2-(4-methylphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H18Cl2N4O2S
6-[[3-[(2,4-Dichlorophenyl)methoxy]phenyl]methylidene]-5-imino-2-(4-methylphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[2-[2-(3-Methylbutyl)benzimidazol-1-yl]ethyl]indolo[3,2-b]quinoxaline —— C28H27N5
6-[2-[2-(3-Methylbutyl)benzimidazol-1-yl]ethyl]indolo[3,2-b]quinoxaline
—— 6-bromo-N-cyclohexyl-2-(2-methylphenyl)imidazo[1,2-a]pyridin-3-amine —— C20H22BrN3
6-bromo-N-cyclohexyl-2-(2-methylphenyl)imidazo[1,2-a]pyridin-3-amine
—— (6S)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— 6-[[3-Bromo-4-[2-(3,4-dimethylphenoxy)ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H27BrN4O4S
6-[[3-Bromo-4-[2-(3,4-dimethylphenoxy)ethoxy]-5-ethoxyphenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-6-[[3-(2-fluorophenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one —— C26H29FN4O2
(6S)-6-[[3-(2-fluorophenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6S)-4-propyl-1-(1H-pyrazole-5-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(1-methylimidazole-4-carbonyl)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(1-methylimidazole-4-carbonyl)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C25H30N6O2
(6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H28N4O3
(6S)-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-6-[[3-(2-fluorophenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one —— C26H29FN4O2
(6R)-6-[[3-(2-fluorophenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H28N4O3
(6S)-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(1-methylimidazole-2-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(1-methylimidazole-2-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-phenylacetyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H31N3O2
(6R)-1-(2-phenylacetyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-methylpyrazole-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6R)-1-(2-methylpyrazole-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C28H36N2O3
(6S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C28H33N3O2
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N3O2
(6S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6R)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C28H36N2O3
(6R)-1-[3-[(2S)-oxolan-2-yl]propanoyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6R)-4-propyl-6-[(2-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(4-methylphenyl)phenyl]methyl]-4-propyl-1-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-5-one —— C25H29N5O2
(6R)-6-[[2-(4-methylphenyl)phenyl]methyl]-4-propyl-1-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-(3-methoxypropanoyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C25H32N2O3
(6S)-1-(3-methoxypropanoyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O
(6R)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O
(6S)-1-[(1-ethylimidazol-2-yl)methyl]-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one