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—— (6S,9S)-6-(3-chlorophenyl)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H35ClN2O4
(6S,9S)-6-(3-chlorophenyl)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-[5-(4-bromophenyl)furan-2-yl]-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C25H23BrN2O2
(6S)-6-[5-(4-bromophenyl)furan-2-yl]-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-6-(3-chlorophenyl)-9-(4-methylphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H22ClF3N2O2
(6R,9S)-6-(3-chlorophenyl)-9-(4-methylphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-bromo-N'-[(2-isopropyl-5-methylphenoxy)acetyl]-2-oxo-2H-chromene-3-carbohydrazide —— C22H21BrN2O5
6-bromo-N'-[(2-isopropyl-5-methylphenoxy)acetyl]-2-oxo-2H-chromene-3-carbohydrazide
—— (6S)-5-benzoyl-6-(4-methoxy-3-phenylmethoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C36H34N2O4
(6S)-5-benzoyl-6-(4-methoxy-3-phenylmethoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— [6-Bromo-8-ethyl-2-(4-methoxyphenyl)quinolin-4-yl]-morpholin-4-ylmethanone —— C23H23BrN2O3
[6-Bromo-8-ethyl-2-(4-methoxyphenyl)quinolin-4-yl]-morpholin-4-ylmethanone
—— (6E)-5-imino-2-methyl-6-[[1-[(3-methylphenyl)methyl]indol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H19N5OS
(6E)-5-imino-2-methyl-6-[[1-[(3-methylphenyl)methyl]indol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[5-chloro-3-(9-chloro-5H-chromeno[4,3-b]pyridin-3-yl)-1-benzofuran-2-carbonyl]-4-methyl-1,4-benzoxazin-3-one —— C30H18Cl2N2O5
6-[5-chloro-3-(9-chloro-5H-chromeno[4,3-b]pyridin-3-yl)-1-benzofuran-2-carbonyl]-4-methyl-1,4-benzoxazin-3-one
—— (6R)-9,9-dimethyl-6-[5-(3-nitrophenyl)furan-2-yl]-5-(2-phenylacetyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C33H29N3O5
(6R)-9,9-dimethyl-6-[5-(3-nitrophenyl)furan-2-yl]-5-(2-phenylacetyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-O-ethyl 8-O-methyl (2Z,7S)-5-amino-7-(4-ethoxyphenyl)-2-[(4-ethoxyphenyl)methylidene]-3-oxo-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate —— C29H30N2O7S
6-O-ethyl 8-O-methyl (2Z,7S)-5-amino-7-(4-ethoxyphenyl)-2-[(4-ethoxyphenyl)methylidene]-3-oxo-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate
—— 6-[(2R)-2-(2-chlorophenyl)-2,3-dihydro-1,5-benzothiazepin-4-yl]-4H-1,4-benzoxazin-3-one —— C23H17ClN2O2S
6-[(2R)-2-(2-chlorophenyl)-2,3-dihydro-1,5-benzothiazepin-4-yl]-4H-1,4-benzoxazin-3-one
—— (6S,9R)-6-(4-fluorophenyl)-3-methyl-9-phenyl-5-(thiophene-2-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C31H25FN2O2S
(6S,9R)-6-(4-fluorophenyl)-3-methyl-9-phenyl-5-(thiophene-2-carbonyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-5-benzoyl-9-(4-methoxyphenyl)-6-pyridin-3-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C32H27N3O3
(6R,9S)-5-benzoyl-9-(4-methoxyphenyl)-6-pyridin-3-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[2-[(3S)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C27H22N6O3S2
6-[2-[(3S)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[2-[(3R)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C27H22N6O3S2
6-[2-[(3R)-3-(4-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C26H19FN6O2S2
6-[2-[(3S)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[6-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-7-yl]-N-[(4-methoxyphenyl)methyl]hexanamide —— C29H36N4O6S
6-[6-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-7-yl]-N-[(4-methoxyphenyl)methyl]hexanamide
—— 6-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C26H19FN6O2S2
6-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-imino-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C24H30N6O4
6-imino-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (6S,9R)-6-(3-fluorophenyl)-5-propanoyl-9-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C31H31FN2O5
(6S,9R)-6-(3-fluorophenyl)-5-propanoyl-9-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-2-(3,5-dichlorophenyl)imino-3-ethyl-N-(3-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C20H19Cl2N3O3S
(6S)-2-(3,5-dichlorophenyl)imino-3-ethyl-N-(3-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxylic acid —— C22H21F3N2O5S
(6S)-3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxylic acid
—— (6R)-N-(2,4-dimethoxyphenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C20H21N3O4S
(6R)-N-(2,4-dimethoxyphenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-[(2,6-dichlorophenyl)methylsulfanylmethyl]-1H-pyrimidine-2,4-dione —— C12H10Cl2N2O2S
6-[(2,6-dichlorophenyl)methylsulfanylmethyl]-1H-pyrimidine-2,4-dione
—— 6-O-ethyl 2-O-methyl 3-benzoyl-4-oxo-1H-quinoline-2,6-dicarboxylate —— C21H17NO6
6-O-ethyl 2-O-methyl 3-benzoyl-4-oxo-1H-quinoline-2,6-dicarboxylate
—— [6-Bromo-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-1-benzofuran-3-yl]-(2,5-dimethoxyphenyl)methanone —— C21H22BrNO5
[6-Bromo-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-1-benzofuran-3-yl]-(2,5-dimethoxyphenyl)methanone
—— 6-Morpholin-4-yl-17-thia-2,7,8-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),2,4,6,11(16)-pentaen-9-one —— C17H18N4O2S
6-Morpholin-4-yl-17-thia-2,7,8-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),2,4,6,11(16)-pentaen-9-one
—— 6-Bromo-2-(4-methoxyphenyl)iminochromene-3-carboxamide —— C17H13BrN2O3
6-Bromo-2-(4-methoxyphenyl)iminochromene-3-carboxamide
—— 6-[2-[(3,4-Dimethoxyphenyl)methylideneamino]phenoxy]-1,3-dimethylpyrimidine-2,4-dione —— C21H21N3O5
6-[2-[(3,4-Dimethoxyphenyl)methylideneamino]phenoxy]-1,3-dimethylpyrimidine-2,4-dione
—— 6-(diethylsulfamoyl)-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide —— C22H32N4O4S
6-(diethylsulfamoyl)-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide
—— 6-Ethoxy-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methylsulfanyl]quinoline-3-carbonitrile —— C21H16N4O2S
6-Ethoxy-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methylsulfanyl]quinoline-3-carbonitrile
—— 6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C23H28N6O4
6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-[2-[(2-Chloro-5-nitrophenyl)methylideneamino]phenoxy]-1,3-dimethylpyrimidine-2,4-dione —— C19H15ClN4O5
6-[2-[(2-Chloro-5-nitrophenyl)methylideneamino]phenoxy]-1,3-dimethylpyrimidine-2,4-dione
—— 6-(azepan-1-ylsulfonyl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-oxo-1H-quinoline-4-carboxamide —— C24H34N4O4S
6-(azepan-1-ylsulfonyl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[2-[(4-Bromophenyl)methylamino]phenoxy]-1,3-dimethylpyrimidine-2,4-dione —— C19H18BrN3O3
6-[2-[(4-Bromophenyl)methylamino]phenoxy]-1,3-dimethylpyrimidine-2,4-dione
—— 6-ethoxy-N-[(2R)-2-ethoxy-3,3,4-trimethyl-2-oxo-1,4,2lambda5-diazaphosphol-5-yl]-4,4-bis(trifluoromethyl)-1,3,5-oxadiazin-2-amine —— C14H20F6N5O4P
6-ethoxy-N-[(2R)-2-ethoxy-3,3,4-trimethyl-2-oxo-1,4,2lambda5-diazaphosphol-5-yl]-4,4-bis(trifluoromethyl)-1,3,5-oxadiazin-2-amine
—— (6R)-2-(1,3-benzodioxol-5-ylimino)-3-ethyl-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C21H21N3O5S
(6R)-2-(1,3-benzodioxol-5-ylimino)-3-ethyl-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(pyridin-3-ylmethyl)-1H-quinoline-4-carboxamide —— C22H24N4O4S
6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(pyridin-3-ylmethyl)-1H-quinoline-4-carboxamide
—— (6S)-2-benzamido-6-methyl-N-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H22N2O2S
(6S)-2-benzamido-6-methyl-N-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-piperidin-1-ylpropyl)-1H-quinoline-4-carboxamide —— C24H34N4O4S
6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-piperidin-1-ylpropyl)-1H-quinoline-4-carboxamide
—— 6-(azepan-1-ylsulfonyl)-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-2-oxo-1H-quinoline-4-carboxamide —— C24H34N4O4S
6-(azepan-1-ylsulfonyl)-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-piperidin-1-ylpropyl)-1H-quinoline-4-carboxamide —— C24H34N4O4S
6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-piperidin-1-ylpropyl)-1H-quinoline-4-carboxamide
—— 6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C23H28N6O4
6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(pyridin-3-ylmethyl)-1H-quinoline-4-carboxamide —— C22H24N4O4S
6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(pyridin-3-ylmethyl)-1H-quinoline-4-carboxamide
—— 6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(1S)-1-phenylethyl]-1H-quinoline-4-carboxamide —— C24H27N3O4S
6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(1S)-1-phenylethyl]-1H-quinoline-4-carboxamide
—— 6,8-dibromo-2-oxo-N-[(1S)-1-phenylethyl]chromene-3-carboxamide —— C18H13Br2NO3
6,8-dibromo-2-oxo-N-[(1S)-1-phenylethyl]chromene-3-carboxamide
—— 6-(azepan-1-ylsulfonyl)-N-[(2S)-3-(diethylamino)-2-methylpropyl]-2-oxo-1H-quinoline-4-carboxamide —— C24H36N4O4S
6-(azepan-1-ylsulfonyl)-N-[(2S)-3-(diethylamino)-2-methylpropyl]-2-oxo-1H-quinoline-4-carboxamide
—— (6R)-2-benzamido-6-methyl-N-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H22N2O2S
(6R)-2-benzamido-6-methyl-N-phenyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-6-cyano-6-(2,6-dichlorophenyl)-N-(2,5-dimethoxyphenyl)-5-oxohexanamide —— C21H20Cl2N2O4
(6R)-6-cyano-6-(2,6-dichlorophenyl)-N-(2,5-dimethoxyphenyl)-5-oxohexanamide
—— (6S,9R)-9-phenyl-6-[2-(trifluoromethyl)phenyl]-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H21F3N2O
(6S,9R)-9-phenyl-6-[2-(trifluoromethyl)phenyl]-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one