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—— (6S)-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C19H21N3O2S2
(6S)-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6S)-2-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C27H29N3O2S2
(6S)-2-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6S)-3-(4-methoxyphenyl)-6-methyl-2-(2-oxo-2-piperidin-1-ylethyl)sulfanyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C21H25N3O3S2
(6S)-3-(4-methoxyphenyl)-6-methyl-2-(2-oxo-2-piperidin-1-ylethyl)sulfanyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6S)-6-methyl-2-(2-oxo-2-piperidin-1-ylethyl)sulfanyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C20H23N3O2S2
(6S)-6-methyl-2-(2-oxo-2-piperidin-1-ylethyl)sulfanyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6R)-6-methyl-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]sulfanyl-3-(2-phenylethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C23H29N3O2S2
(6R)-6-methyl-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]sulfanyl-3-(2-phenylethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6S)-2-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-(2-phenylethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C26H27N3O2S2
(6S)-2-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-(2-phenylethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— 6-ethoxy-3-[[[(1S)-1-[1-(furan-2-ylmethyl)tetrazol-5-yl]propyl]-(2-hydroxyethyl)amino]methyl]-1H-quinolin-2-one —— C23H28N6O4
6-ethoxy-3-[[[(1S)-1-[1-(furan-2-ylmethyl)tetrazol-5-yl]propyl]-(2-hydroxyethyl)amino]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[[[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H32N6OS
6,7-dimethyl-3-[[[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6-methoxy-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one —— C28H36N6O2
6-methoxy-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one
—— 6-ethoxy-3-[[[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H29FN6O2S
6-ethoxy-3-[[[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6,7-dimethoxy-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C24H30N6O3S
6,7-dimethoxy-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6-methoxy-3-[[[(1R)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C25H32N6O2S
6-methoxy-3-[[[(1R)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[[[(1S)-1-[1-(furan-2-ylmethyl)tetrazol-5-yl]propyl]-[(4-methoxyphenyl)methyl]amino]methyl]-1H-quinolin-2-one —— C29H32N6O3
6-ethyl-3-[[[(1S)-1-[1-(furan-2-ylmethyl)tetrazol-5-yl]propyl]-[(4-methoxyphenyl)methyl]amino]methyl]-1H-quinolin-2-one
—— 6-methoxy-3-[[[(1S)-1-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H31N7O3
6-methoxy-3-[[[(1S)-1-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 6-[(1R,2S,6R,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(9-oxofluoren-2-yl)hexanamide —— C28H26N2O4
6-[(1R,2S,6R,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(9-oxofluoren-2-yl)hexanamide
—— (6S)-6-methyl-2-[[2-(4-propanoylpiperazin-1-yl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H28N4O3S
(6S)-6-methyl-2-[[2-(4-propanoylpiperazin-1-yl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-methoxy-1-[(2-methylphenyl)methyl]-3-[[[(2S)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid —— C28H30N2O3
6-methoxy-1-[(2-methylphenyl)methyl]-3-[[[(2S)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid
—— 6-ethoxy-3-[(S)-[4-(4-fluorophenyl)piperazin-1-yl]-[1-(furan-2-ylmethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H28FN7O3
6-ethoxy-3-[(S)-[4-(4-fluorophenyl)piperazin-1-yl]-[1-(furan-2-ylmethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2R)-oxolan-2-yl]methylamino]methyl]indole-2-carboxylic acid —— C24H28N2O4
6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2R)-oxolan-2-yl]methylamino]methyl]indole-2-carboxylic acid
—— 6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2S)-oxolan-2-yl]methylamino]methyl]indole-2-carboxylic acid —— C24H28N2O4
6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2S)-oxolan-2-yl]methylamino]methyl]indole-2-carboxylic acid
—— 6-ethoxy-3-[(R)-[4-(2-fluorophenyl)piperazin-1-yl]-[1-(furan-2-ylmethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H28FN7O3
6-ethoxy-3-[(R)-[4-(2-fluorophenyl)piperazin-1-yl]-[1-(furan-2-ylmethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-methoxy-1-[(2-methylphenyl)methyl]-3-[[[(2R)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid —— C28H30N2O3
6-methoxy-1-[(2-methylphenyl)methyl]-3-[[[(2R)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid
—— 6-ethoxy-3-[(R)-[1-(furan-2-ylmethyl)tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-1H-quinolin-2-one —— C23H27N7O3
6-ethoxy-3-[(R)-[1-(furan-2-ylmethyl)tetrazol-5-yl]-(4-methylpiperazin-1-yl)methyl]-1H-quinolin-2-one
—— 6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2S)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid —— C28H30N2O3
6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2S)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid
—— 6,7-dimethyl-3-[(S)-morpholin-4-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C25H28N6O2
6,7-dimethyl-3-[(S)-morpholin-4-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-Methoxy-2-[2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl]sulfanylquinoline-3-carbonitrile —— C21H16N4O3S
6-Methoxy-2-[2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl]sulfanylquinoline-3-carbonitrile
—— (6aS)-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C23H27N3O4
(6aS)-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aS)-N-[(3-fluorophenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C21H22FN3O2
(6aS)-N-[(3-fluorophenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— 6-Amino-7-chloro-3-[(4-fluorophenyl)methyl]-2-methylquinazolin-4-one —— C16H13ClFN3O
6-Amino-7-chloro-3-[(4-fluorophenyl)methyl]-2-methylquinazolin-4-one
—— 6-(4-Methylpiperidin-1-yl)-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrile —— C17H17N3O2
6-(4-Methylpiperidin-1-yl)-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrile
—— (6aS)-5-methyl-6-oxo-N-(3-propan-2-yloxypropyl)-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C20H29N3O3
(6aS)-5-methyl-6-oxo-N-(3-propan-2-yloxypropyl)-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aS)-N-[(5-bromo-2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C22H24BrN3O3
(6aS)-N-[(5-bromo-2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— 6-methyl-N-[(1R)-1-phenylethyl]thieno[2,3-b]quinoline-2-carboxamide —— C21H18N2OS
6-methyl-N-[(1R)-1-phenylethyl]thieno[2,3-b]quinoline-2-carboxamide
—— (6aS)-N-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C29H39N5O2
(6aS)-N-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— 6-[4-(2-Methylbenzoyl)-1,4-diazepan-1-yl]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrile —— C24H22N4O3
6-[4-(2-Methylbenzoyl)-1,4-diazepan-1-yl]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrile
—— 6-[4-(Cyclopropanecarbonyl)-1,4-diazepan-1-yl]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrile —— C20H20N4O3
6-[4-(Cyclopropanecarbonyl)-1,4-diazepan-1-yl]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrile
—— (6aR)-N-[2-(3,4-diethoxyphenyl)ethyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C26H33N3O4
(6aR)-N-[2-(3,4-diethoxyphenyl)ethyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[(2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C22H25N3O3
(6aR)-N-[(2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C29H39N5O2
(6aR)-N-[3-[4-(2,5-dimethylphenyl)piperazin-1-yl]propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aS)-N-[3-(azepan-1-yl)propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C23H34N4O2
(6aS)-N-[3-(azepan-1-yl)propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-5-methyl-N-[(2-methylphenyl)methyl]-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C22H25N3O2
(6aR)-5-methyl-N-[(2-methylphenyl)methyl]-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aS)-N-[2-(3,4-diethoxyphenyl)ethyl]-6-oxo-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxaline-3-carboxamide —— C25H31N3O4
(6aS)-N-[2-(3,4-diethoxyphenyl)ethyl]-6-oxo-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[(5-bromo-2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C22H24BrN3O3
(6aR)-N-[(5-bromo-2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[(3-fluorophenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C21H22FN3O2
(6aR)-N-[(3-fluorophenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— 6-Ethyl-2-[4-(4-fluorobenzoyl)-1,4-diazepan-1-yl]quinoline-3-carbonitrile —— C24H23FN4O
6-Ethyl-2-[4-(4-fluorobenzoyl)-1,4-diazepan-1-yl]quinoline-3-carbonitrile
—— (6aR)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-methyl-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxalin-6-one —— C21H27N3O4
(6aR)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-methyl-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxalin-6-one
—— (6aS)-N-[3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]propyl]-6-oxo-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxaline-3-carboxamide —— C27H34ClN5O2
(6aS)-N-[3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]propyl]-6-oxo-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxaline-3-carboxamide
—— 6-(1,3-benzodioxol-5-ylamino)-N-(2-phenylethyl)pyridine-3-carboxamide —— C21H19N3O3
6-(1,3-benzodioxol-5-ylamino)-N-(2-phenylethyl)pyridine-3-carboxamide
—— (6aS)-N-(3-methoxypropyl)-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C18H25N3O3
(6aS)-N-(3-methoxypropyl)-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aS)-5-ethyl-N-(2-methoxyethyl)-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C18H25N3O3
(6aS)-5-ethyl-N-(2-methoxyethyl)-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide