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—— 6-[(2R)-2-(4,8-dimethyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidin-2-yl)piperidin-1-yl]sulfonyl-3H-1,3-benzoxazol-2-one —— C21H25N5O4S
6-[(2R)-2-(4,8-dimethyl-6,7-dihydro-5H-pyrido[2,3-d]pyrimidin-2-yl)piperidin-1-yl]sulfonyl-3H-1,3-benzoxazol-2-one
—— 6-[(3S)-1-[2-(4-fluorophenyl)-2-methylpropanoyl]piperidin-3-yl]-N-methylpyridine-3-carboxamide —— C22H26FN3O2
6-[(3S)-1-[2-(4-fluorophenyl)-2-methylpropanoyl]piperidin-3-yl]-N-methylpyridine-3-carboxamide
—— 6-[(3S)-1-(3-ethylimidazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C19H25N5O2
6-[(3S)-1-(3-ethylimidazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[(3S)-1-[2-(4-fluorophenyl)-2-methylpropanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C23H28FN3O2
6-[(3S)-1-[2-(4-fluorophenyl)-2-methylpropanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— [6-[1-(2-Ethylpyrazole-3-carbonyl)piperidin-4-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C22H30N6O2
[6-[1-(2-Ethylpyrazole-3-carbonyl)piperidin-4-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— [6-[(3R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C22H29N5O3
[6-[(3R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— [6-[(3S)-1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C25H29FN4O
[6-[(3S)-1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— 6-[(3R)-1-[2-(4-fluorophenoxy)-2-methylpropanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C23H28FN3O3
6-[(3R)-1-[2-(4-fluorophenoxy)-2-methylpropanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[(3R)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C24H31N3O2
6-[(3R)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— [6-[1-(1,3-Dimethylpyrazole-4-carbonyl)piperidin-4-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C22H30N6O2
[6-[1-(1,3-Dimethylpyrazole-4-carbonyl)piperidin-4-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-[(3R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C24H25FN4O3
6-[(3R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-Amino-8-(furan-2-yl)-12-(furan-2-ylmethylidene)-4-thia-2-azatricyclo[7.3.0.03,7]dodeca-1,3(7),5,8-tetraene-5-carboxamide —— C20H15N3O3S
6-Amino-8-(furan-2-yl)-12-(furan-2-ylmethylidene)-4-thia-2-azatricyclo[7.3.0.03,7]dodeca-1,3(7),5,8-tetraene-5-carboxamide
—— 6-[1-(4-methylthiadiazole-5-carbonyl)piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C18H18N6O2S2
6-[1-(4-methylthiadiazole-5-carbonyl)piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-4-yl]-N-(cyclopropylmethyl)pyridine-3-carboxamide —— C22H23N5O2S
6-[1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-4-yl]-N-(cyclopropylmethyl)pyridine-3-carboxamide
—— [6-[(3R)-1-(6-methoxypyridine-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C23H29N5O3
[6-[(3R)-1-(6-methoxypyridine-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-[(3S)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C24H25FN4O3
6-[(3S)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-[(3R)-1-(2-ethylpyrazole-3-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C23H24FN5O2
6-[(3R)-1-(2-ethylpyrazole-3-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-[(4-Bromophenyl)carbamoyl]cyclohex-3-ene-1-carboxylic acid —— C14H14BrNO3
6-[(4-Bromophenyl)carbamoyl]cyclohex-3-ene-1-carboxylic acid
—— 6-[(3S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C24H31N3O2
6-[(3S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[(3R)-1-[[2-(diethylamino)-1,3-thiazol-5-yl]methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C21H31N5OS
6-[(3R)-1-[[2-(diethylamino)-1,3-thiazol-5-yl]methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[1-[2-[(3S)-3-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C22H29N5O2S
6-[1-[2-[(3S)-3-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[(3R)-1-(3-ethylimidazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C19H25N5O2
6-[(3R)-1-(3-ethylimidazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[1-[2-[(3R)-3-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C22H29N5O2S
6-[1-[2-[(3R)-3-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[(3S)-1-(3-ethylimidazole-4-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C23H24FN5O2
6-[(3S)-1-(3-ethylimidazole-4-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— [6-[(3R)-1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C25H29FN4O
[6-[(3R)-1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— 6-[(3S)-1-methylsulfonylpiperidin-3-yl]-N-(3-oxo-3-piperidin-1-ylpropyl)pyridine-3-carboxamide —— C20H30N4O4S
6-[(3S)-1-methylsulfonylpiperidin-3-yl]-N-(3-oxo-3-piperidin-1-ylpropyl)pyridine-3-carboxamide
—— 6-[1-[2-(benzotriazol-1-yl)acetyl]piperidin-4-yl]-N-cyclopentylpyridine-3-carboxamide —— C24H28N6O2
6-[1-[2-(benzotriazol-1-yl)acetyl]piperidin-4-yl]-N-cyclopentylpyridine-3-carboxamide
—— 6-[(3S)-1-(6-methoxypyridine-3-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C20H24N4O3
6-[(3S)-1-(6-methoxypyridine-3-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— [6-[(3R)-1-(2-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C24H31N5O2
[6-[(3R)-1-(2-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— 6-[(3S)-1-[2-(4-fluorophenoxy)-2-methylpropanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C23H28FN3O3
6-[(3S)-1-[2-(4-fluorophenoxy)-2-methylpropanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-4-yl]-N-cyclopentylpyridine-3-carboxamide —— C23H25N5O2S
6-[1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-4-yl]-N-cyclopentylpyridine-3-carboxamide
—— 6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C24H24FN5O2
6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-[1-[2-[[(2S)-oxolan-2-yl]methoxy]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C21H26N4O4S
6-[1-[2-[[(2S)-oxolan-2-yl]methoxy]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— [6-[(3S)-1-(6-methoxypyridine-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C23H29N5O3
[6-[(3S)-1-(6-methoxypyridine-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— [6-[1-(2,4-Dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C22H29N5O2S
[6-[1-(2,4-Dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-[[4-(4-chlorophenyl)-5-prop-2-ynylsulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione —— C16H12ClN5O2S
6-[[4-(4-chlorophenyl)-5-prop-2-ynylsulfanyl-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-[(3R)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C20H21N5O2S
6-[(3R)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[(3S)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-N-methylpyridine-3-carboxamide —— C19H19N5O2S
6-[(3S)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-N-methylpyridine-3-carboxamide
—— 6-[(3S)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-N-(cyclopropylmethyl)pyridine-3-carboxamide —— C22H23N5O2S
6-[(3S)-1-(2,1,3-benzothiadiazole-5-carbonyl)piperidin-3-yl]-N-(cyclopropylmethyl)pyridine-3-carboxamide
—— 6-methyl-2-[2-oxo-2-[(3R)-3-[5-(piperidine-1-carbonyl)pyridin-2-yl]piperidin-1-yl]ethyl]pyridazin-3-one —— C23H29N5O3
6-methyl-2-[2-oxo-2-[(3R)-3-[5-(piperidine-1-carbonyl)pyridin-2-yl]piperidin-1-yl]ethyl]pyridazin-3-one
—— [6-[(3R)-1-(2-ethylpyrazole-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C21H27N5O2
[6-[(3R)-1-(2-ethylpyrazole-3-carbonyl)piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— 6-[(3S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-N-methylpyridine-3-carboxamide —— C18H22N4O3
6-[(3S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-N-methylpyridine-3-carboxamide
—— 6-[(3S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C19H27N5O
6-[(3S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— [6-[(3S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C22H29N5O3
[6-[(3S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— [6-[(3R)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone —— C21H27N5O2
[6-[(3R)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-3-yl]pyridin-3-yl]-pyrrolidin-1-ylmethanone
—— 6-[(3S)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C19H25N5O2
6-[(3S)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[(3R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-N-methylpyridine-3-carboxamide —— C18H22N4O3
6-[(3R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-N-methylpyridine-3-carboxamide
—— (6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C25H31N3O2
(6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-[(3R)-1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C24H26FN5O2
6-[(3R)-1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-[(3R)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C19H25N5O2
6-[(3R)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide