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—— (6R)-6-[1-(3-morpholin-4-yl-3-oxopropyl)piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C26H37N3O3
(6R)-6-[1-(3-morpholin-4-yl-3-oxopropyl)piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H29N3O3S
(6S)-1-[(3-methoxyphenyl)methyl]-6-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H32N4O3
(6R)-6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H32N4O3
(6S)-6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[(1-ethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H34N4O2
(6R)-6-[1-[(1-ethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-benzyl-6-[1-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C26H36N4O
(6R)-1-benzyl-6-[1-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C25H32N4O
(6R)-6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C26H33FN4O
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H34N4O2
(6S)-6-[1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-benzyl-6-[1-[2-(3-methoxyphenoxy)ethyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H34N2O3
(6S)-1-benzyl-6-[1-[2-(3-methoxyphenoxy)ethyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H34N4O2
(6R)-6-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-(2-methoxyethyl)-6-[1-[[2-(4-methylphenyl)pyrimidin-5-yl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C26H34N4O2
(6R)-1-(2-methoxyethyl)-6-[1-[[2-(4-methylphenyl)pyrimidin-5-yl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(4-fluorophenyl)methyl]-6-[1-[(1-methylpyrazol-4-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C23H29FN4O
(6S)-1-[(4-fluorophenyl)methyl]-6-[1-[(1-methylpyrazol-4-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-[(1-methylpyrazol-4-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C23H29FN4O
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-[(1-methylpyrazol-4-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-(4-methylphthalazin-1-yl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H29FN4O
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-(4-methylphthalazin-1-yl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H33FN4O
(6R)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(1-ethylimidazol-2-yl)methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C24H31FN4O
(6S)-6-[1-[(1-ethylimidazol-2-yl)methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[3-(4-chlorophenyl)propanoyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C23H31ClN2O3
(6R)-6-[1-[3-(4-chlorophenyl)propanoyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(1-ethylimidazol-2-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C25H34N4O
(6S)-6-[1-[(1-ethylimidazol-2-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(4-fluorophenyl)methyl]-6-[1-(4-methylphthalazin-1-yl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H29FN4O
(6S)-1-[(4-fluorophenyl)methyl]-6-[1-(4-methylphthalazin-1-yl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-(3-bromo-4-hydroxy-5-methoxyphenyl)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H30BrClN4O6S
6-(3-bromo-4-hydroxy-5-methoxyphenyl)-8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6S)-6-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C24H31FN4O
(6S)-6-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-(3-morpholin-4-yl-3-oxopropyl)piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C26H37N3O3
(6S)-6-[1-(3-morpholin-4-yl-3-oxopropyl)piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C28H40N4O
(6R)-6-[1-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— 6-[(2-chloro-6-fluorophenyl)methylsulfanyl]-5-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-one —— C18H12ClFN4OS
6-[(2-chloro-6-fluorophenyl)methylsulfanyl]-5-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-one
—— (6R)-1-benzyl-6-[1-[2-(3-methoxyphenoxy)ethyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H34N2O3
(6R)-1-benzyl-6-[1-[2-(3-methoxyphenoxy)ethyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-(1,5-dimethylpyrazole-4-carbonyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H32N4O3
(6R)-6-[1-(1,5-dimethylpyrazole-4-carbonyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[3-(4-chlorophenyl)propanoyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C23H31ClN2O3
(6S)-6-[1-[3-(4-chlorophenyl)propanoyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-methoxyethyl)-6-[1-[[2-(4-methylphenyl)pyrimidin-5-yl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C26H34N4O2
(6S)-1-(2-methoxyethyl)-6-[1-[[2-(4-methylphenyl)pyrimidin-5-yl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C26H35N5O
(6S)-6-[1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-[(3-methoxyphenyl)methyl]-6-(1-pyrimidin-2-ylpiperidin-4-yl)-5,6-dihydro-2H-azepin-7-one —— C23H28N4O2
(6S)-1-[(3-methoxyphenyl)methyl]-6-(1-pyrimidin-2-ylpiperidin-4-yl)-5,6-dihydro-2H-azepin-7-one
—— 6-(4-iodo-2,5-dimethyl-thiophen-3-yl)-1,6-dihydro-pyrimidine —— C10H11IN2S
6-(4-iodo-2,5-dimethyl-thiophen-3-yl)-1,6-dihydro-pyrimidine
—— (6R)-1-(2-phenylethyl)-6-[1-(quinolin-6-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C29H33N3O
(6R)-1-(2-phenylethyl)-6-[1-(quinolin-6-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H32N4O2
(6S)-6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C28H36N2O3
(6S)-6-[1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H32N4O2
(6R)-6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C27H36N4O
(6S)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-methoxyethyl)-6-[1-[[4-(2-methoxyphenyl)phenyl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C28H36N2O3
(6S)-1-(2-methoxyethyl)-6-[1-[[4-(2-methoxyphenyl)phenyl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-phenylethyl)-6-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H36N4O
(6S)-1-(2-phenylethyl)-6-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C26H35N5O
(6R)-6-[1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C25H32FN5O
(6S)-6-[1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-1-[(4-fluorophenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-(quinolin-6-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C28H30FN3O
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-(quinolin-6-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-[(4-chlorophenyl)methylsulfanyl]-5-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-one —— C18H13ClN4OS
6-[(4-chlorophenyl)methylsulfanyl]-5-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-one
—— (6S)-1-[(4-fluorophenyl)methyl]-6-[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C26H31FN2O2
(6S)-1-[(4-fluorophenyl)methyl]-6-[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-benzyl-6-[1-(quinolin-6-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C28H31N3O
(6S)-1-benzyl-6-[1-(quinolin-6-ylmethyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-(2-Hydroxy-5-methoxyphenyl)-2,8-bis[2-(4-hydroxyphenyl)ethyl]-3a,4,6,6a,9a,10,10a,10b-octahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H36N2O8
6-(2-Hydroxy-5-methoxyphenyl)-2,8-bis[2-(4-hydroxyphenyl)ethyl]-3a,4,6,6a,9a,10,10a,10b-octahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6R)-6-(1-benzoylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one —— C26H30N2O3
(6R)-6-(1-benzoylpiperidin-4-yl)-1-[(3-methoxyphenyl)methyl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(4-fluorophenyl)methyl]-6-[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C26H31FN2O2
(6R)-1-[(4-fluorophenyl)methyl]-6-[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C27H36N4O
(6R)-6-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C28H40N4O
(6S)-6-[1-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one