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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C28H36N2O3
(6S)-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6S)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopropylmethyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H31N3O
(6S)-1-(cyclopropylmethyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C26H30N4O3
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C25H28N4O2
(6S)-6-[(3-phenylphenyl)methyl]-4-propyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N5O
(6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-ethylimidazole-4-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C27H32N4O2
(6S)-1-(3-ethylimidazole-4-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-ethylimidazole-4-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6R)-1-(3-ethylimidazole-4-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1-[(2S)-2-pyrrolidin-1-ylpropanoyl]-1,4-diazepan-5-one —— C27H36N4O2
(6R)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1-[(2S)-2-pyrrolidin-1-ylpropanoyl]-1,4-diazepan-5-one
—— (6R)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6R)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(1-methylimidazole-2-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C27H32N4O2
(6R)-1-(1-methylimidazole-2-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N5O
(6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6R)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-1-(2-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Benzyl-5-methyl-2-(oxan-4-yl)-7-propoxypyrazolo[1,5-a]pyrimidine —— C22H27N3O2
6-Benzyl-5-methyl-2-(oxan-4-yl)-7-propoxypyrazolo[1,5-a]pyrimidine
—— (6R)-1-(1-methylpyrazole-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6R)-1-(1-methylpyrazole-3-carbonyl)-6-[(3-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(3-ethylimidazole-4-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-1-(3-ethylimidazole-4-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-ethylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C27H32N4O2
(6R)-1-(3-ethylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C28H36N2O3
(6S)-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(5-methylthiophene-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6S)-1-(5-methylthiophene-3-carbonyl)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C23H27N5O2S
(6S)-4-propyl-6-[(3-thiophen-2-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1-[(2S)-2-pyrrolidin-1-ylpropanoyl]-1,4-diazepan-5-one —— C27H36N4O2
(6S)-4-propyl-6-[(4-pyridin-3-ylphenyl)methyl]-1-[(2S)-2-pyrrolidin-1-ylpropanoyl]-1,4-diazepan-5-one
—— (6S)-1-[2-(4-methyltriazol-1-yl)acetyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H31N5O2
(6S)-1-[2-(4-methyltriazol-1-yl)acetyl]-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-1-(1-methylpyrazole-3-carbonyl)-4-propyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclopropylmethyl)-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H31N3O
(6R)-1-(cyclopropylmethyl)-4-propyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C24H27N5O3
(6S)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-propyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclobutanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C27H34N2O3
(6R)-1-(cyclobutanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(1-methylimidazole-4-carbonyl)-6-[[3-(3-methylphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C27H32N4O2
(6S)-1-(1-methylimidazole-4-carbonyl)-6-[[3-(3-methylphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(2-phenylacetyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H31N3O2
(6S)-1-(2-phenylacetyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-methoxypropanoyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C25H32N2O3
(6R)-1-(3-methoxypropanoyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O3
(6S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-propyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[(2-phenylphenyl)methyl]-1-propanoyl-4-propyl-1,4-diazepan-5-one —— C24H30N2O2
(6S)-6-[(2-phenylphenyl)methyl]-1-propanoyl-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(2-methylpyrazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C26H30N4O2
(6S)-1-(2-methylpyrazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6S)-1-(cyclobutanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one —— C27H34N2O3
(6S)-1-(cyclobutanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one —— C24H27N5O3
(6R)-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-6-[(2-phenylphenyl)methyl]-4-propyl-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6R)-4-propyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6S)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N5O
(6S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-propyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one —— C26H29FN4O2
(6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-4-propyl-1,4-diazepan-5-one
—— (6S)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C24H28N6O2
(6S)-4-propyl-6-[(4-pyridin-4-ylphenyl)methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-6-[[3-(2-fluorophenyl)phenyl]methyl]-4-propyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one —— C26H27FN4O2
(6R)-6-[[3-(2-fluorophenyl)phenyl]methyl]-4-propyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-4-propyl-1-(2-pyrazol-1-ylacetyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one