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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-1-(3-methoxypropanoyl)-6-[[3-(2-methylphenyl)phenyl]methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H32N2O3
(6R)-1-(3-methoxypropanoyl)-6-[[3-(2-methylphenyl)phenyl]methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6S)-1-(cyclopentanecarbonyl)-6-[[3-(2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H30N2O2
(6S)-1-(cyclopentanecarbonyl)-6-[[3-(2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C27H31N3O3
(6S)-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6S)-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C27H31N3O3
(6S)-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6S)-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6S)-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-1,4-diazepan-5-one
—— (6S)-1-(3-methoxypropanoyl)-6-[[3-(2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H28N2O3
(6S)-1-(3-methoxypropanoyl)-6-[[3-(2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-(5-acetyl-4-amino-6-methylpyrimidin-2-yl)-4-[4-(4-fluorophenyl)methylpiperazin-1-yl]-5-methyl-2-phenylthieno[2,3-d]pyrimidine —— C30H28FN7OS
6-(5-acetyl-4-amino-6-methylpyrimidin-2-yl)-4-[4-(4-fluorophenyl)methylpiperazin-1-yl]-5-methyl-2-phenylthieno[2,3-d]pyrimidine
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(2-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H30N4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(2-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Amino-3-(2,5-dimethylthiophen-3-yl)-4-(3-methoxyphenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C20H18N4O2S
6-Amino-3-(2,5-dimethylthiophen-3-yl)-4-(3-methoxyphenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(2-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H30N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(2-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one —— C25H25F2N3O
(6R)-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-methoxyacetyl)-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28N4O4
6-(2-methoxyacetyl)-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-Methylphenyl)-piperazin-1-ylmethyl]isoquinoline —— C21H23N3
6-[(3-Methylphenyl)-piperazin-1-ylmethyl]isoquinoline
—— (6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one —— C26H29N3O2
(6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28N4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butyl-1-methyl-4-(2,4,5-trimethylphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidine-2,5-dione —— C20H27N3O2
6-butyl-1-methyl-4-(2,4,5-trimethylphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidine-2,5-dione
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-methoxyacetyl)-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28N4O4
6-(2-methoxyacetyl)-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-3-[(3S)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-methyl-3-[(3S)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-(4-fluorobenzoyl)-2-[(2R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H26FN5O2
6-(4-fluorobenzoyl)-2-[(2R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one —— C26H29N3O2
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
—— 6-ethoxy-1-(2-iodophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C19H19IN2O
6-ethoxy-1-(2-iodophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-4-one —— C19H25N5O2
6-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-4-one
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one —— C26H29N3O2
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopentanecarbonyl)-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-(cyclopentanecarbonyl)-2-[(2S)-1-(2-methylbenzoyl)piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-4-methyl-1-[(6-methylpyridin-2-yl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6S)-4-methyl-1-[(6-methylpyridin-2-yl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Methyl-3-[1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-Methyl-3-[1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-[[3-[2-(4-Bromophenoxy)ethoxy]phenyl]methylidene]-2-butyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23BrN4O3S
6-[[3-[2-(4-Bromophenoxy)ethoxy]phenyl]methylidene]-2-butyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— [6-(2,4-Dichlorophenyl)-4-(phenoxymethyl)-1,5,2-dioxazinan-2-yl](phenyl)methanone —— C23H19Cl2NO4
[6-(2,4-Dichlorophenyl)-4-(phenoxymethyl)-1,5,2-dioxazinan-2-yl](phenyl)methanone
—— 6-[(3S)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-pyrrolidin-1-yl-1H-pyrimidin-4-one —— C19H25N5O
6-[(3S)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-pyrrolidin-1-yl-1H-pyrimidin-4-one
—— 6'-amino-3'-methyl-2-oxo-1-(propan-2-yl)-1,2-dihydro-1'H-spiro[indole-3,4'-pyrano[2,3-c]pyrazole]-5'-carbonitrile —— C18H17N5O2
6'-amino-3'-methyl-2-oxo-1-(propan-2-yl)-1,2-dihydro-1'H-spiro[indole-3,4'-pyrano[2,3-c]pyrazole]-5'-carbonitrile
—— 6-methyl-2-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-pyrimidin-4-one —— C16H20N4O
6-methyl-2-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-pyrimidin-4-one
—— (6R)-4-methyl-1-[(6-methylpyridin-2-yl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6R)-4-methyl-1-[(6-methylpyridin-2-yl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(4-fluorobenzoyl)-2-[(2S)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H26FN5O2
6-(4-fluorobenzoyl)-2-[(2S)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one —— C26H29N3O2
(6S)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
—— 6-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-pyrrolidin-1-yl-1H-pyrimidin-4-one —— C19H25N5O
6-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-pyrrolidin-1-yl-1H-pyrimidin-4-one
—— (6S)-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one —— C25H25F2N3O
(6S)-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
—— 6-[(6-methylpyridin-2-yl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H23N5
6-[(6-methylpyridin-2-yl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(6-methylpyridin-2-yl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H23N5
6-[(6-methylpyridin-2-yl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-methyl-3-[(3R)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-methyl-3-[(3R)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-[(2-methoxy-3-methylphenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O
6-[(2-methoxy-3-methylphenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(3R)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C24H29N5O
6-[(3R)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[[(2-methoxy-3-methylphenyl)methylamino]methyl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C21H25N5O
6-[[(2-methoxy-3-methylphenyl)methylamino]methyl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-4-ylpyrimidin-4-amine —— C25H31N5O
6-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C24H29N5O
6-[(3S)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[1-[(2-methoxy-3-methylphenyl)methyl]piperidin-4-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C25H31N5O
6-[1-[(2-methoxy-3-methylphenyl)methyl]piperidin-4-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— (6S)-1-(2-methoxy-3-methylbenzoyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H27N3O3
(6S)-1-(2-methoxy-3-methylbenzoyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(3R)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C25H31N5O
6-[(3R)-1-[(2-methoxy-3-methylphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[(2-methoxy-3-methylphenyl)methyl]-2-[(2R)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C22H30N4O
6-[(2-methoxy-3-methylphenyl)methyl]-2-[(2R)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine