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—— 6-fluoro-5-methyl-2-[(2S)-1-[2-(4-methylsulfonylphenyl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23FN4O4S
6-fluoro-5-methyl-2-[(2S)-1-[2-(4-methylsulfonylphenyl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(2R)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H21N5O4S
6-[(2R)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one —— C19H23ClN4O4S
6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one
—— 6-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20N4O5S
6-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20ClN5O4S
6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one —— C20H25N3O5S
6-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one
—— 6-[(1-Benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N6O3S
6-[(1-Benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[2-(4-Bromophenyl)-2-oxoethoxy]-2-[(2,3,4-trimethoxyphenyl)methylidene]-1-benzofuran-3-one —— C26H21BrO7
6-[2-(4-Bromophenyl)-2-oxoethoxy]-2-[(2,3,4-trimethoxyphenyl)methylidene]-1-benzofuran-3-one
—— 6-[(2,6-Dichlorophenyl)methoxy]-2-[(2-methylphenyl)methylidene]-1-benzofuran-3-one —— C23H16Cl2O3
6-[(2,6-Dichlorophenyl)methoxy]-2-[(2-methylphenyl)methylidene]-1-benzofuran-3-one
—— 6-Amino-1-benzyl-3-methyl-5-[2-[4-(3-phenylprop-2-enyl)piperazin-1-yl]acetyl]pyrimidine-2,4-dione —— C27H31N5O3
6-Amino-1-benzyl-3-methyl-5-[2-[4-(3-phenylprop-2-enyl)piperazin-1-yl]acetyl]pyrimidine-2,4-dione
—— 6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one —— C18H21ClN4O3S2
6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one
—— 6-[[3-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C41H46N4O8
6-[[3-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[[4-(4-nitrophenyl)piperazin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-(4-Benzhydrylpiperazine-1-carbonyl)-2-(4-chlorophenyl)-4,5-dihydropyridazin-3-one —— C28H27ClN4O2
6-(4-Benzhydrylpiperazine-1-carbonyl)-2-(4-chlorophenyl)-4,5-dihydropyridazin-3-one
—— 6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one —— C19H23ClN4O3S
6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one
—— 6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one —— C19H23ClN4O4S
6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one
—— 6-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one —— C20H25N3O5S
6-[(2S)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one
—— 6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one —— C19H23ClN4O4S
6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one
—— 6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one —— C18H21ClN4O3S2
6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one
—— 6-[(2S)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H21N5O4S
6-[(2S)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-Amino-1-benzyl-3-methyl-5-[2-(2-methyl-2,3-dihydroindol-1-yl)acetyl]pyrimidine-2,4-dione —— C23H24N4O3
6-Amino-1-benzyl-3-methyl-5-[2-(2-methyl-2,3-dihydroindol-1-yl)acetyl]pyrimidine-2,4-dione
—— 6-[(2R)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one —— C20H26N4O4S
6-[(2R)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one
—— 6-[[5-(3,4-Dichlorophenyl)furan-2-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H18Cl2N4O2S
6-[[5-(3,4-Dichlorophenyl)furan-2-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one —— C19H23ClN4O3S
6-[(2R)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one
—— 6-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C44H50N4O7
6-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[(2S)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one —— C20H26N4O4S
6-[(2S)-2-(1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one
—— 6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one —— C18H21ClN4O3S2
6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one
—— 6-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C25H25N5O3
6-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— 6-ethyl-5-methyl-2-[(2R)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H32N4O4
6-ethyl-5-methyl-2-[(2R)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one —— C18H21ClN4O3S2
6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-methyl-1,3-benzothiazol-2-one
—— 6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20ClN5O4S
6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20N4O5S
6-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]pyridine-3-carboxamide —— C25H25N5O2
6-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]pyridine-3-carboxamide
—— 6-(furan-2-yl)-2-[[1-[(1R,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one —— C22H29N3O4
6-(furan-2-yl)-2-[[1-[(1R,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one
—— 6-Ethoxy-3-[(2-ethylpiperidin-1-yl)methyl]-1,3-benzothiazole-2-thione —— C17H24N2OS2
6-Ethoxy-3-[(2-ethylpiperidin-1-yl)methyl]-1,3-benzothiazole-2-thione
—— 6-(furan-2-yl)-2-[[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one —— C22H29N3O4
6-(furan-2-yl)-2-[[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one
—— 6-[4-(2-hydroxyethoxy)phenyl]-5'-(5-methoxy-4-methoxycarbonyl-5-oxopent-1-ynyl)-1'-[(1-methoxy-3-methyl-1-oxobutan-2-yl)carbamoyl]-1,2'-dioxo-3,4-diphenylspiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-8-carboxylic acid —— C50H49N3O14
6-[4-(2-hydroxyethoxy)phenyl]-5'-(5-methoxy-4-methoxycarbonyl-5-oxopent-1-ynyl)-1'-[(1-methoxy-3-methyl-1-oxobutan-2-yl)carbamoyl]-1,2'-dioxo-3,4-diphenylspiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-8-carboxylic acid
—— 6-phenylmethoxy-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-2-ium —— C27H29N2O4+
6-phenylmethoxy-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-2-ium
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-(3-methoxyphenyl)prop-2-enoate —— C19H17NO7
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-(3-methoxyphenyl)prop-2-enoate
—— 6-(furan-2-yl)-2-[1-[(2R)-2-phenylpropanoyl]piperidin-4-yl]pyridazin-3-one —— C22H23N3O3
6-(furan-2-yl)-2-[1-[(2R)-2-phenylpropanoyl]piperidin-4-yl]pyridazin-3-one
—— 6-(furan-2-yl)-2-[[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]methyl]pyridazin-3-one —— C19H23N3O4
6-(furan-2-yl)-2-[[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]methyl]pyridazin-3-one
—— 6-(furan-2-yl)-2-[[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one —— C22H29N3O4
6-(furan-2-yl)-2-[[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one
—— 6-(furan-2-yl)-2-[[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one —— C22H29N3O4
6-(furan-2-yl)-2-[[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]methyl]pyridazin-3-one
—— 6-(furan-2-yl)-2-[1-[(2S)-2-phenylpropanoyl]piperidin-4-yl]pyridazin-3-one —— C22H23N3O3
6-(furan-2-yl)-2-[1-[(2S)-2-phenylpropanoyl]piperidin-4-yl]pyridazin-3-one
—— 6-(furan-2-yl)-2-[[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]methyl]pyridazin-3-one —— C19H23N3O4
6-(furan-2-yl)-2-[[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]methyl]pyridazin-3-one
—— 6-Chloro-2-(2,4-dichlorophenyl)-8-methylquinoline-4-carboxylic acid —— C17H10Cl3NO2
6-Chloro-2-(2,4-dichlorophenyl)-8-methylquinoline-4-carboxylic acid
—— 6-bromo-3-[2-[3-(4-fluorophenyl)-7-[(4-fluorophenyl)methylidene]-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-1,3-thiazol-5-yl]chromen-2-one —— C32H22BrF2N3O2S
6-bromo-3-[2-[3-(4-fluorophenyl)-7-[(4-fluorophenyl)methylidene]-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-1,3-thiazol-5-yl]chromen-2-one
—— 6-Amino-3-ethyl-4-(4-methoxyphenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C16H16N4O2
6-Amino-3-ethyl-4-(4-methoxyphenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-ethyl-5-methyl-2-(oxan-4-yl)-N-[(1-propylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C23H37N5O
6-ethyl-5-methyl-2-(oxan-4-yl)-N-[(1-propylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 6-ethyl-N-[(1S)-1-(2-methoxyphenyl)ethyl]-5-methyl-2-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine —— C23H30N4O2
6-ethyl-N-[(1S)-1-(2-methoxyphenyl)ethyl]-5-methyl-2-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 6-bromo-2-[(2-chlorobenzyl)sulfanyl]-3H-imidazo[4,5-b]pyridine —— C13H9BrClN3S
6-bromo-2-[(2-chlorobenzyl)sulfanyl]-3H-imidazo[4,5-b]pyridine