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—— [6-Fluoro-2-(4-fluoro-phenyl)-quinazolin-4-ylsulfanyl]-acetic acid isopropyl ester —— C19H16F2N2O2S
[6-Fluoro-2-(4-fluoro-phenyl)-quinazolin-4-ylsulfanyl]-acetic acid isopropyl ester
—— (6S)-2-benzamido-6-tert-butyl-N,N-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C22H28N2O2S
(6S)-2-benzamido-6-tert-butyl-N,N-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-6-tert-butyl-N-(furan-2-ylmethyl)-2-[(2-methylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H30N2O3S
(6S)-6-tert-butyl-N-(furan-2-ylmethyl)-2-[(2-methylbenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-ethoxy-3-[(R)-[4-(4-hydroxyphenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H33N7O4
6-ethoxy-3-[(R)-[4-(4-hydroxyphenyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-[benzyl(methyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide —— C23H25N3O5S
6-[benzyl(methyl)sulfamoyl]-4-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1H-quinoline-3-carboxamide
—— 6,7-dimethoxy-3-[(S)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-1H-quinolin-2-one —— C28H33N7O4
6,7-dimethoxy-3-[(S)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-1H-quinolin-2-one
—— (6-nitro-1H-benzimidazol-2-yl)methyl 2,4-dichlorobenzoate —— C15H9Cl2N3O4
(6-nitro-1H-benzimidazol-2-yl)methyl 2,4-dichlorobenzoate
—— 6-[(3S)-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C26H32N4O5S
6-[(3S)-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C26H32N4O5S
6-[(3R)-3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3S)-3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C26H32N4O5S
6-[(3S)-3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27FN4O5S
6-[(3R)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3S)-3-[4-(4-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27ClN4O5S
6-[(3S)-3-[4-(4-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3S)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C25H30N4O6S
6-[(3S)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(3-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27ClN4O5S
6-[(3R)-3-[4-(3-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C26H32N4O5S
6-[(3R)-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3S)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27FN4O5S
6-[(3S)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3S)-3-[4-(3-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27ClN4O5S
6-[(3S)-3-[4-(3-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27FN4O5S
6-[(3R)-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C25H30N4O6S
6-[(3R)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3R)-3-[4-(4-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27ClN4O5S
6-[(3R)-3-[4-(4-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-[(3S)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one —— C24H27FN4O5S
6-[(3S)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]sulfonyl-3-methyl-1,3-benzoxazol-2-one
—— 6-(diethylsulfamoyl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide —— C22H32N4O4S
6-(diethylsulfamoyl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-4-oxo-1H-quinoline-3-carboxamide
—— 6-chloro-2-methoxy-N-[(4R)-4-piperidin-1-ylpentyl]acridin-9-amine —— C24H30ClN3O
6-chloro-2-methoxy-N-[(4R)-4-piperidin-1-ylpentyl]acridin-9-amine
—— 6-methoxy-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one —— C22H30N6O2
6-methoxy-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one
—— 6,8-dimethyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-1H-quinolin-2-one —— C22H30N6O
6,8-dimethyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-1H-quinolin-2-one —— C24H34N6O
6,7-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-1H-quinolin-2-one
—— 6-bromo-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]chromene-3-carboxamide —— C15H14BrNO4
6-bromo-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]chromene-3-carboxamide
—— 6-ethoxy-3-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-morpholin-4-ylmethyl]-1H-quinolin-2-one —— C24H25FN6O3
6-ethoxy-3-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-morpholin-4-ylmethyl]-1H-quinolin-2-one
—— 6,7-dimethoxy-3-[(S)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C27H32N6O4
6,7-dimethoxy-3-[(S)-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— 6-ethoxy-3-[(S)-[4-(4-hydroxyphenyl)piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C28H33N7O4
6-ethoxy-3-[(S)-[4-(4-hydroxyphenyl)piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,8-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3R)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C24H34N6O
6,8-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3R)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— 6-bromo-2-(4-fluorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]imidazo[1,2-a]pyridin-3-amine —— C18H17BrFN3O
6-bromo-2-(4-fluorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]imidazo[1,2-a]pyridin-3-amine
—— 6-bromo-2-(4-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]imidazo[1,2-a]pyridin-3-amine —— C19H20BrN3O
6-bromo-2-(4-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]imidazo[1,2-a]pyridin-3-amine
—— [6-[(2S)-2-methyl-2,3-dihydroindole-1-carbonyl]pyridin-2-yl]-[(2S)-2-methyl-2,3-dihydroindol-1-yl]methanone —— C25H23N3O2
[6-[(2S)-2-methyl-2,3-dihydroindole-1-carbonyl]pyridin-2-yl]-[(2S)-2-methyl-2,3-dihydroindol-1-yl]methanone
—— 6-methyl-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-3-(2-methylpropyl)-4-oxofuro[2,3-d]pyrimidine-5-carboxamide —— C21H32N4O3
6-methyl-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-3-(2-methylpropyl)-4-oxofuro[2,3-d]pyrimidine-5-carboxamide
—— 6-[cyclohexyl(methyl)sulfamoyl]-1-methyl-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide —— C27H40N4O4S
6-[cyclohexyl(methyl)sulfamoyl]-1-methyl-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide
—— 6-[cyclohexyl(methyl)sulfamoyl]-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-1-methyl-4-oxoquinoline-3-carboxamide —— C28H42N4O4S
6-[cyclohexyl(methyl)sulfamoyl]-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-1-methyl-4-oxoquinoline-3-carboxamide
—— 6-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-1-ethyl-4-oxo-N-[(1R)-1-phenylethyl]quinoline-3-carboxamide —— C29H29N3O4S
6-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-1-ethyl-4-oxo-N-[(1R)-1-phenylethyl]quinoline-3-carboxamide
—— 6-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-3-(2-methylpropyl)-4-oxofuro[2,3-d]pyrimidine-5-carboxamide —— C21H32N4O3
6-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-3-(2-methylpropyl)-4-oxofuro[2,3-d]pyrimidine-5-carboxamide
—— 6-bromo-N-cyclopentyl-2-pyridin-4-ylimidazo[1,2-a]pyridin-3-amine —— C17H17BrN4
6-bromo-N-cyclopentyl-2-pyridin-4-ylimidazo[1,2-a]pyridin-3-amine
—— 6-[4-(Furan-2-carbonyl)piperazin-1-yl]-3,3,8-trimethyl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrile —— C21H24N4O3
6-[4-(Furan-2-carbonyl)piperazin-1-yl]-3,3,8-trimethyl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrile
—— 6-ethyl-2-[[(E)-3-phenylprop-2-enoyl]carbamothioylamino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide —— C20H22N4O2S2
6-ethyl-2-[[(E)-3-phenylprop-2-enoyl]carbamothioylamino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide
—— (6R)-2-(2,5-dimethoxyphenyl)imino-N-(2-ethylphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C21H23N3O4S
(6R)-2-(2,5-dimethoxyphenyl)imino-N-(2-ethylphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-fluoro-3-(4-methoxyphenyl)sulfonyl-7-[(3S)-3-methylpiperidin-1-yl]-1-propylquinolin-4-one —— C25H29FN2O4S
6-fluoro-3-(4-methoxyphenyl)sulfonyl-7-[(3S)-3-methylpiperidin-1-yl]-1-propylquinolin-4-one
—— 6-methyl-3-(2-methylpropyl)-4-oxo-N-[(1S)-1-phenylethyl]furo[2,3-d]pyrimidine-5-carboxamide —— C20H23N3O3
6-methyl-3-(2-methylpropyl)-4-oxo-N-[(1S)-1-phenylethyl]furo[2,3-d]pyrimidine-5-carboxamide
—— 6-ethyl-3-[(S)-[4-(furan-2-carbonyl)piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C27H31N7O4
6-ethyl-3-[(S)-[4-(furan-2-carbonyl)piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,8-Dichloro-3-[4-(2-hydroxyethyl)piperazine-1-carbonyl]chromen-2-one —— C16H16Cl2N2O4
6,8-Dichloro-3-[4-(2-hydroxyethyl)piperazine-1-carbonyl]chromen-2-one
—— 6-[cyclohexyl(methyl)sulfamoyl]-1-ethyl-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide —— C29H44N4O4S
6-[cyclohexyl(methyl)sulfamoyl]-1-ethyl-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide
—— 6-[cyclohexyl(methyl)sulfamoyl]-1-ethyl-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide —— C28H42N4O4S
6-[cyclohexyl(methyl)sulfamoyl]-1-ethyl-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-oxoquinoline-3-carboxamide
—— 6-fluoro-3-(4-methoxyphenyl)sulfonyl-7-[(3R)-3-methylpiperidin-1-yl]-1-propylquinolin-4-one —— C25H29FN2O4S
6-fluoro-3-(4-methoxyphenyl)sulfonyl-7-[(3R)-3-methylpiperidin-1-yl]-1-propylquinolin-4-one