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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(3R)-1-[2-(2-methylphenyl)acetyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C22H23N5O2
6-[(3R)-1-[2-(2-methylphenyl)acetyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-methyl-1-[[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C21H19F3N2O2S
6-methyl-1-[[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-Methyl-12-[3-(3-methylpyrazol-1-yl)propanoyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C18H21N5O2S
6-Methyl-12-[3-(3-methylpyrazol-1-yl)propanoyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 6-fluoro-2-[(3S)-1-[(2S)-2-(5-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C22H24FN5O2
6-fluoro-2-[(3S)-1-[(2S)-2-(5-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[(2-Methylphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H28N4O
6-[(2-Methylphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(4-Fluorophenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H18FN5O2
6-[2-(4-Fluorophenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3S)-1-[3-(6-methylpyridin-2-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C24H25FN4O2
6-fluoro-2-[(3S)-1-[3-(6-methylpyridin-2-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3S)-1-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C23H26FN5O2
6-fluoro-2-[(3S)-1-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3R)-1-[(2R)-2-(5-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C22H24FN5O2
6-fluoro-2-[(3R)-1-[(2R)-2-(5-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-(Dimethylsulfamoyl)-2-(3-fluoro-4-methoxyphenyl)quinoline-4-carboxylic acid —— C19H17FN2O5S
6-(Dimethylsulfamoyl)-2-(3-fluoro-4-methoxyphenyl)quinoline-4-carboxylic acid
—— 6-fluoro-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O2
6-fluoro-2-[(3R)-1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-[2-(3-Methylphenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H21N5O2
6-[2-(3-Methylphenyl)acetyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[3-(6-Methylpyridin-2-yl)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H20N6O2
6-[3-(6-Methylpyridin-2-yl)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C20H20N6O2
6-[(3R)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-methyl-1-[[(2R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C22H21F3N2O2S
6-methyl-1-[[(2R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-[(3S)-1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C22H23N5O2
6-[(3S)-1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-[(dimethylamino)methyl]octahydro-5H-4,7-methanoinden-5-one —— C13H21NO
6-[(dimethylamino)methyl]octahydro-5H-4,7-methanoinden-5-one
—— 6-Fluoro-2-[1-[2-(3-methylphenyl)acetyl]piperidin-4-yl]quinoline-3-carboxamide —— C24H24FN3O2
6-Fluoro-2-[1-[2-(3-methylphenyl)acetyl]piperidin-4-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]quinoline-3-carboxamide —— C25H26FN3O2
6-fluoro-2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]quinoline-3-carboxamide
—— (6-methylpyridin-3-yl)-[(3R)-3-(2-methylpyrido[2,3-d]pyrimidin-4-yl)piperidin-1-yl]methanone —— C20H21N5O
(6-methylpyridin-3-yl)-[(3R)-3-(2-methylpyrido[2,3-d]pyrimidin-4-yl)piperidin-1-yl]methanone
—— 6-[(3S)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C20H20N6O2
6-[(3S)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-Methyl-12-(6-methylpyridine-3-carbonyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C18H18N4O2S
6-Methyl-12-(6-methylpyridine-3-carbonyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 6-(6-Methylpyridine-3-carbonyl)-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H16N6O2
6-(6-Methylpyridine-3-carbonyl)-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3R)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O2
6-fluoro-2-[(3R)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3S)-1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O2
6-fluoro-2-[(3S)-1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3R)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]quinoline-3-carboxamide —— C22H21FN4O2
6-fluoro-2-[(3R)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-[(2R)-2-(3,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2R)-2-(3,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2S)-2-(3,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2S)-2-(3,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C22H23N5O2
6-[(3R)-1-[2-(4-methylphenyl)acetyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-Fluoro-2-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]quinoline-3-carboxamide —— C22H21FN4O2
6-Fluoro-2-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]quinoline-3-carboxamide
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxylate —— C20H17N3O7
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxylate
—— (6-Bromonaphthalen-2-yl) 4-chloro-3-pyrrolidin-1-ylsulfonylbenzoate —— C21H17BrClNO4S
(6-Bromonaphthalen-2-yl) 4-chloro-3-pyrrolidin-1-ylsulfonylbenzoate
—— 6'-amino-3'-ethyl-1'H-spiro[fluorene-9,4'-pyrano[2,3-c]pyrazole]-5'-carbonitrile —— C21H16N4O
6'-amino-3'-ethyl-1'H-spiro[fluorene-9,4'-pyrano[2,3-c]pyrazole]-5'-carbonitrile
—— 6-[(2R)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2R)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[4-(2,4-Dimethylphenoxy)butanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O3
6-[4-(2,4-Dimethylphenoxy)butanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2S)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H23N5O3
6-[(2S)-2-(2,4-dimethylphenoxy)propanoyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Imino-11-methyl-5-(4-methylpiperazine-1-carbonyl)-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-2-one —— C24H32N6O3
6-Imino-11-methyl-5-(4-methylpiperazine-1-carbonyl)-7-(3-propan-2-yloxypropyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaen-2-one
—— 6-amino-N-[[4-(5-chloro-2-methylphenyl)-5-[(3-methylphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]hexanamide —— C24H30ClN5OS
6-amino-N-[[4-(5-chloro-2-methylphenyl)-5-[(3-methylphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]hexanamide
—— 6-(Furan-2-carbonyl)-2,2,7-trimethyl-4-(2-oxo-2-piperidin-1-ylethyl)-1,4-benzoxazin-3-one —— C23H26N2O5
6-(Furan-2-carbonyl)-2,2,7-trimethyl-4-(2-oxo-2-piperidin-1-ylethyl)-1,4-benzoxazin-3-one
—— 6-(Furan-2-yl)-2-[(3-methoxyphenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)pyridazin-3-one —— C20H17N3O4
6-(Furan-2-yl)-2-[(3-methoxyphenyl)methyl]-5-(3-methyl-1,2-oxazol-5-yl)pyridazin-3-one
—— 6-fluoro-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O2
6-fluoro-2-[(3S)-1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-(Furan-2-yl)-5-(3-methyl-1,2-oxazol-5-yl)-2-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]pyridazin-3-one —— C23H20N4O4
6-(Furan-2-yl)-5-(3-methyl-1,2-oxazol-5-yl)-2-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]pyridazin-3-one
—— 6-(Furan-2-yl)-2-[2-(4-methoxyphenyl)-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)pyridazin-3-one —— C21H17N3O5
6-(Furan-2-yl)-2-[2-(4-methoxyphenyl)-2-oxoethyl]-5-(3-methyl-1,2-oxazol-5-yl)pyridazin-3-one
—— 6-Chloro-2-{3-[(4-methylpiperidin-1-yl)sulfonyl]phenyl}imidazo[1,2-a]pyridine —— C19H20ClN3O2S
6-Chloro-2-{3-[(4-methylpiperidin-1-yl)sulfonyl]phenyl}imidazo[1,2-a]pyridine
—— 6-Fluoro-2-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]quinoline-3-carboxamide —— C20H19FN4O3
6-Fluoro-2-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]quinoline-3-carboxamide
—— 6-(Furan-2-yl)-5-(3-methyl-1,2-oxazol-5-yl)-2-(2-oxo-2-piperidin-1-ylethyl)pyridazin-3-one —— C19H20N4O4
6-(Furan-2-yl)-5-(3-methyl-1,2-oxazol-5-yl)-2-(2-oxo-2-piperidin-1-ylethyl)pyridazin-3-one
—— (6S)-6-(4-methoxyphenyl)-5-methyl-2-(6-methylpyridin-2-yl)-3,6-dihydrooxazine —— C18H20N2O2
(6S)-6-(4-methoxyphenyl)-5-methyl-2-(6-methylpyridin-2-yl)-3,6-dihydrooxazine
—— (6S)-5-ethyl-2-(4-methylpyridin-2-yl)-6-phenyl-3,6-dihydrooxazine —— C18H20N2O
(6S)-5-ethyl-2-(4-methylpyridin-2-yl)-6-phenyl-3,6-dihydrooxazine
—— 6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C14H12F3N7O
6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— (6S)-5-methyl-6-phenyl-2-pyridin-2-yl-3,6-dihydrooxazine —— C16H16N2O
(6S)-5-methyl-6-phenyl-2-pyridin-2-yl-3,6-dihydrooxazine