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—— 6-amino-8-(3-chlorophenyl)-8,8a-dihydro-1H-isothiochromene-5,7,7(3H)-tricarbonitrile —— C18H13ClN4S
6-amino-8-(3-chlorophenyl)-8,8a-dihydro-1H-isothiochromene-5,7,7(3H)-tricarbonitrile
—— 6-amino-N-[3-[N-[(4-chlorophenyl)carbamoyl]anilino]propyl]hexanamide —— C22H29ClN4O2
6-amino-N-[3-[N-[(4-chlorophenyl)carbamoyl]anilino]propyl]hexanamide
—— 6-Amino-4-[1-[2-(2,6-dimethylpiperidin-1-yl)-2-oxoethyl]indol-3-yl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H28N6O2
6-Amino-4-[1-[2-(2,6-dimethylpiperidin-1-yl)-2-oxoethyl]indol-3-yl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (6S)-5-[2-(4-chlorophenyl)ethyl]-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H37ClN4O2
(6S)-5-[2-(4-chlorophenyl)ethyl]-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-5-(4-methoxyphenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H36N4O3
(6S)-N-cyclooctyl-5-(4-methoxyphenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-6-methyl-5-(2-methylphenyl)-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H36N4O2
(6S)-N-cyclooctyl-6-methyl-5-(2-methylphenyl)-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-5-(2,4-dimethylphenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H38N4O2
(6S)-N-cyclooctyl-5-(2,4-dimethylphenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(3,4-dimethylphenyl)-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H36N4O2
(6R)-N-cyclohexyl-5-(3,4-dimethylphenyl)-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cycloheptyl-6-methyl-4-oxo-5-[(4-propan-2-yloxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H42N4O3
(6S)-2-tert-butyl-N-cycloheptyl-6-methyl-4-oxo-5-[(4-propan-2-yloxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(4-ethylphenyl)-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H33FN4O2
(6R)-N-cyclohexyl-2-(4-ethylphenyl)-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-6-methyl-5-[(4-methylphenyl)methyl]-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H38N4O2
(6S)-N-cyclooctyl-6-methyl-5-[(4-methylphenyl)methyl]-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-(3,4-dimethylphenyl)-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H36N4O2
(6S)-N-cyclohexyl-5-(3,4-dimethylphenyl)-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-2-(4-ethylphenyl)-5-(2-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H31FN4O2
(6S)-N-cyclohexyl-2-(4-ethylphenyl)-5-(2-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-benzyl-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H36N4O2
(6R)-5-benzyl-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclooctyl-5-(2,5-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O2
(6S)-2-tert-butyl-N-cyclooctyl-5-(2,5-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-5-(3-propylsulfanylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H42N4O2S
(6S)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-5-(3-propylsulfanylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-(4-chlorophenyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H33ClN4O2
(6R)-5-(4-chlorophenyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-tert-butyl-N-cyclooctyl-6-methyl-5-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H38N4O2
(6R)-2-tert-butyl-N-cyclooctyl-6-methyl-5-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-5-(4-ethylphenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H38N4O2
(6S)-N-cyclooctyl-5-(4-ethylphenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-6-methyl-5-(4-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O2S
(6R)-N-cyclooctyl-6-methyl-5-(4-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(4-ethylphenyl)-5-[(3-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H33FN4O2
(6R)-N-cyclohexyl-2-(4-ethylphenyl)-5-[(3-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(1,3-benzodioxol-5-ylmethyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N4O4
(6S)-5-(1,3-benzodioxol-5-ylmethyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H36N4O2S
(6S)-N-cyclooctyl-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-[(4-chlorophenyl)methyl]-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H35ClN4O2
(6S)-5-[(4-chlorophenyl)methyl]-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(3-chlorophenyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H33ClN4O2
(6S)-5-(3-chlorophenyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-(2,4-dimethylphenyl)-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H36N4O2
(6S)-N-cyclohexyl-5-(2,4-dimethylphenyl)-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-5-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H35N5O2
(6R)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-5-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclooctyl-5-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O3
(6S)-2-tert-butyl-N-cyclooctyl-5-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-5-[(2-ethoxyphenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O3
(6R)-N-cyclooctyl-5-[(2-ethoxyphenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclooctyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H35FN4O2
(6S)-2-tert-butyl-N-cyclooctyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H35FN4O2
(6R)-N-cyclooctyl-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-(Dimethylsulfamoyl)-2-(4-methylsulfanylphenyl)quinoline-4-carboxylic acid —— C19H18N2O4S2
6-(Dimethylsulfamoyl)-2-(4-methylsulfanylphenyl)quinoline-4-carboxylic acid
—— (6S)-5-(5-chloro-2-methylphenyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H35ClN4O2
(6S)-5-(5-chloro-2-methylphenyl)-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-tert-butyl-N-cyclooctyl-5-(3,5-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O2
(6R)-2-tert-butyl-N-cyclooctyl-5-(3,5-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-5-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H34N4O2
(6S)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-5-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-5-[(4-ethoxyphenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O3
(6R)-N-cyclooctyl-5-[(4-ethoxyphenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O2
(6R)-N-cyclooctyl-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-2-cyclopropyl-5-(3-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H34N4O3
(6R)-N-cyclooctyl-2-cyclopropyl-5-(3-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-cyclohexyl-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H40N4O2
(6R)-5-cyclohexyl-N-cyclooctyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cycloheptyl-5-(2,4-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H38N4O2
(6S)-2-tert-butyl-N-cycloheptyl-5-(2,4-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C31H38N4O2
(6S)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-5-(2,4-difluorophenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H32F2N4O2
(6S)-N-cyclooctyl-5-(2,4-difluorophenyl)-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclooctyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-propylsulfanylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H38N4O3S
(6R)-N-cyclooctyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-propylsulfanylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclooctyl-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H37FN4O2
(6S)-2-tert-butyl-N-cyclooctyl-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-2-(furan-2-yl)-5-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H34N4O4
(6S)-N-cyclooctyl-2-(furan-2-yl)-5-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2,5-bis(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H36N4O2
(6R)-N-cyclohexyl-2,5-bis(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-5-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H38N4O3
(6S)-N-cyclooctyl-5-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclooctyl-6-methyl-4-oxo-5-[(2S)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H42N4O2
(6S)-2-tert-butyl-N-cyclooctyl-6-methyl-4-oxo-5-[(2S)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-tert-butyl-N-cyclooctyl-6-methyl-4-oxo-5-[(2S)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H42N4O2
(6R)-2-tert-butyl-N-cyclooctyl-6-methyl-4-oxo-5-[(2S)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclooctyl-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H40N4O2
(6S)-N-cyclooctyl-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide