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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Bromo-3',5'-DI-tert-butyl-2-(4-nitrophenyl)-2,4-dihydrospiro[1,4-benzoxazine-3,1'-cyclohexane]-2',5'-dien-4'-one —— C27H29BrN2O4
6-Bromo-3',5'-DI-tert-butyl-2-(4-nitrophenyl)-2,4-dihydrospiro[1,4-benzoxazine-3,1'-cyclohexane]-2',5'-dien-4'-one
—— (6-methyl-1H-indol-2-yl)-[4-(1H-pyrrolo[3,2-b]pyridin-2-yl)piperidin-1-yl]methanone —— C22H22N4O
(6-methyl-1H-indol-2-yl)-[4-(1H-pyrrolo[3,2-b]pyridin-2-yl)piperidin-1-yl]methanone
—— 6-(cyclopentanecarbonyl)-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-(cyclopentanecarbonyl)-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-N-[(2R)-1-[(3S)-3-(2-methylsulfonylacetyl)piperidin-1-yl]-1-oxopropan-2-yl]-1H-indole-2-carboxamide —— C21H27N3O5S
6-methyl-N-[(2R)-1-[(3S)-3-(2-methylsulfonylacetyl)piperidin-1-yl]-1-oxopropan-2-yl]-1H-indole-2-carboxamide
—— (6-methyl-1H-indol-2-yl)-[4-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone —— C23H21F3N4O
(6-methyl-1H-indol-2-yl)-[4-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone
—— (6-methyl-1H-indol-2-yl)-[(3S)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone —— C23H21F3N4O
(6-methyl-1H-indol-2-yl)-[(3S)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone
—— 6-(2-methoxyacetyl)-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28N4O4
6-(2-methoxyacetyl)-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28N4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6-methyl-1H-indol-2-yl)-[(3R)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone —— C23H21F3N4O
(6-methyl-1H-indol-2-yl)-[(3R)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone
—— (6R)-1-(5-methyl-1-benzofuran-2-carbonyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H25N3O3
(6R)-1-(5-methyl-1-benzofuran-2-carbonyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(5-methyl-1-benzofuran-2-carbonyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H25N3O3
(6S)-1-(5-methyl-1-benzofuran-2-carbonyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Hydroxy-5-[[6-hydroxy-1-(2-methylphenyl)-4-oxo-2-sulfanylidenepyrimidin-5-yl]-[4-methoxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-1-(2-methylphenyl)-2-sulfanylidenepyrimidin-4-one —— C35H35N5O6S2
6-Hydroxy-5-[[6-hydroxy-1-(2-methylphenyl)-4-oxo-2-sulfanylidenepyrimidin-5-yl]-[4-methoxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-1-(2-methylphenyl)-2-sulfanylidenepyrimidin-4-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-bromo-5-methoxy-4-propoxybenzoate —— C20H20BrNO8
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-bromo-5-methoxy-4-propoxybenzoate
—— 6-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C32H39N5O6
6-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-methyl-1-[[(2S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C24H27F3N4O
6-methyl-1-[[(2S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-1-[[(2R)-1-[(5-methyl-1-prop-2-enylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C24H27F3N4O
6-methyl-1-[[(2R)-1-[(5-methyl-1-prop-2-enylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6,8-Difluoro-2-pyridin-2-ylquinoline-4-carboxylic acid —— C15H8F2N2O2
6,8-Difluoro-2-pyridin-2-ylquinoline-4-carboxylic acid
—— 6-methyl-1-[[(2S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C22H24F3N5O
6-methyl-1-[[(2S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-2-oxo-4-(4-propan-2-ylphenyl)-N-[2-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C22H22F3N3O2
6-methyl-2-oxo-4-(4-propan-2-ylphenyl)-N-[2-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 6-methyl-1-[[(2S)-1-[(5-methyl-1-prop-2-enylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C24H27F3N4O
6-methyl-1-[[(2S)-1-[(5-methyl-1-prop-2-enylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C32H39N3O6
6-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-methyl-1-[[(2R)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C22H23F3N4OS
6-methyl-1-[[(2R)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-1-[[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C21H23F3N4O
6-methyl-1-[[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-1-[[(2R)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C24H27F3N4O
6-methyl-1-[[(2R)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-1-[[(2S)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C22H23F3N4OS
6-methyl-1-[[(2S)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-1-[[(2R)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C22H24F3N5O
6-methyl-1-[[(2R)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— 6-methyl-1'-[2-[(4R)-2-oxo-4-phenylpyrrolidin-1-yl]acetyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H28N2O4
6-methyl-1'-[2-[(4R)-2-oxo-4-phenylpyrrolidin-1-yl]acetyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[(3S)-3-(1,2,4-triazol-1-yl)butanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C20H24N4O3
6-methyl-1'-[(3S)-3-(1,2,4-triazol-1-yl)butanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[2-[(4S)-2-oxo-4-phenylpyrrolidin-1-yl]acetyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H28N2O4
6-methyl-1'-[2-[(4S)-2-oxo-4-phenylpyrrolidin-1-yl]acetyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl-(3,6-dimethyl-1-benzofuran-2-yl)methanone —— C16H16N4O2
6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl-(3,6-dimethyl-1-benzofuran-2-yl)methanone
—— 6-methyl-1'-[2-oxo-2-(4-pyridin-2-ylpiperazin-1-yl)ethyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C25H30N4O3
6-methyl-1'-[2-oxo-2-(4-pyridin-2-ylpiperazin-1-yl)ethyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[2-(2-propan-2-ylbenzimidazol-1-yl)acetyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H29N3O3
6-methyl-1'-[2-(2-propan-2-ylbenzimidazol-1-yl)acetyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C21H25N3O3
6-methyl-1'-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[(2R)-2-(4-oxo-3H-phthalazin-1-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C25H25N3O4
6-methyl-1'-[(2R)-2-(4-oxo-3H-phthalazin-1-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6'-Bromo-2'-oxohexahydrospiro[cyclopropane-1,4'-[1]oxa[3,5]methanocyclopenta[b]furan]-7'-carboxylic acid —— C11H11BrO4
6'-Bromo-2'-oxohexahydrospiro[cyclopropane-1,4'-[1]oxa[3,5]methanocyclopenta[b]furan]-7'-carboxylic acid
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H26N4O4S
6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-1'-(3-methyl-4-morpholin-4-ylbenzoyl)spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H30N2O4
6-methyl-1'-(3-methyl-4-morpholin-4-ylbenzoyl)spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[(2R)-2-(4-oxoquinazolin-3-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C25H25N3O4
6-methyl-1'-[(2R)-2-(4-oxoquinazolin-3-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[(2S)-2-(4-oxo-3H-phthalazin-1-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C25H25N3O4
6-methyl-1'-[(2S)-2-(4-oxo-3H-phthalazin-1-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-[3-(2-hydroxyethoxy)phenyl]-1,2'-dioxo-3,4-diphenyl-1-N'-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1',8-dicarboxamide —— C44H40N4O7
6-[3-(2-hydroxyethoxy)phenyl]-1,2'-dioxo-3,4-diphenyl-1-N'-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1',8-dicarboxamide
—— 6-methyl-1'-[(3R)-3-(1,2,4-triazol-1-yl)butanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C20H24N4O3
6-methyl-1'-[(3R)-3-(1,2,4-triazol-1-yl)butanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-methyl-1'-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C21H25N3O3
6-methyl-1'-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6'-[4-(2-hydroxyethoxy)phenyl]-5-[2-(4-methoxyphenyl)ethynyl]-3',4'-diphenyl-8'-(4-pyrimidin-2-ylpiperazine-1-carbonyl)spiro[1H-indole-3,7'-4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine]-1',2-dione —— C52H46N6O7
6'-[4-(2-hydroxyethoxy)phenyl]-5-[2-(4-methoxyphenyl)ethynyl]-3',4'-diphenyl-8'-(4-pyrimidin-2-ylpiperazine-1-carbonyl)spiro[1H-indole-3,7'-4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine]-1',2-dione
—— 6-methyl-1'-[1-(pyridin-3-ylmethyl)piperidine-4-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H31N3O3
6-methyl-1'-[1-(pyridin-3-ylmethyl)piperidine-4-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H26N4O4S
6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H26N4O4S
6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H26N4O4S
6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(5-methylthiophene-2-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C24H24N2O2S
(6R)-1-(5-methylthiophene-2-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H26N4O4S
6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one