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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-4-ethyl-1-(3-methoxybenzoyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6S)-4-ethyl-1-(3-methoxybenzoyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[2-(4-methyltriazol-1-yl)acetyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[2-(4-methyltriazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclobutanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H32N2O3
(6R)-1-(cyclobutanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O3
(6R)-4-ethyl-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(6-methylpyridin-2-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H30N4O
(6S)-4-ethyl-1-[(6-methylpyridin-2-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-benzyl-4-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C26H38N6
6-benzyl-4-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-1-[(1S)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C28H34N2O3
(6R)-1-[(1S)-cyclohex-3-ene-1-carbonyl]-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(1-propan-2-ylpyrazole-4-carbonyl)-1,4-diazepan-5-one —— C27H32N4O2
(6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(1-propan-2-ylpyrazole-4-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O2
(6S)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one —— C28H36N2O3
(6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O2
(6R)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one —— C26H30N4O3
(6R)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(1-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-5-one —— C26H29N3O
(6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-methoxybenzoyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6R)-4-ethyl-1-(2-methoxybenzoyl)-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-5-one —— C24H27N5O2
(6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H30N4O2
(6R)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(5-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one —— C26H30N4O3
(6S)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(5-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
—— (6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O3
(6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C26H29N3O
(6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(pyridin-3-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6S)-4-ethyl-1-(pyridin-3-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclobutanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H32N2O3
(6S)-1-(cyclobutanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(6-methoxypyridine-3-carbonyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H28N4O3
(6S)-4-ethyl-1-(6-methoxypyridine-3-carbonyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-chloro-3-[(4-phenylphenyl)methylidene]-1H-indol-2-one —— C21H14ClNO
6-chloro-3-[(4-phenylphenyl)methylidene]-1H-indol-2-one
—— (6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(2-pyrazol-1-ylacetyl)-1,4-diazepan-5-one —— C25H28N4O2
(6S)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(2-pyrazol-1-ylacetyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6S)-4-ethyl-1-(pyridin-2-ylmethyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(4-methoxyphenyl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O2
(6S)-4-ethyl-1-[(4-methoxyphenyl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-ethyl-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H32N2O2
(6R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)-4-ethyl-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(3-pyridin-4-ylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2S
(6S)-4-ethyl-1-(3-pyridin-4-ylpropanoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one —— C28H36N2O3
(6S)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[3-[(2S)-oxolan-2-yl]propanoyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H24N4O3S
(6S)-4-ethyl-1-(6-oxo-1H-pyridazine-3-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-ethyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6S)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-ethyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N3O3
(6R)-4-ethyl-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C26H29N3O
(6R)-4-ethyl-6-[(2-phenylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O3
(6S)-4-ethyl-1-[2-(2-oxopyrrolidin-1-yl)acetyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one —— C25H28FN3O3
(6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4O2S
(6R)-4-ethyl-1-(5-methyl-1H-pyrazole-4-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N5O
(6S)-4-ethyl-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[(3-phenylphenyl)methyl]-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one —— C26H27N3O2
(6R)-4-ethyl-6-[(3-phenylphenyl)methyl]-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H32N2O3S
(6R)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-propan-2-ylpyrazole-4-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-4-ethyl-1-(1-propan-2-ylpyrazole-4-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O2
(6S)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-pyrazol-1-ylacetyl)-1,4-diazepan-5-one —— C26H30N4O3
(6S)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-pyrazol-1-ylacetyl)-1,4-diazepan-5-one
—— (6S)-1-(cyclopentanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H34N2O3
(6S)-1-(cyclopentanecarbonyl)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H30N4O2
(6S)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(5-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one —— C26H30N4O2
(6S)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(5-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N3O3
(6S)-4-ethyl-1-[(2R)-2-(2-oxopyrrolidin-1-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(4-methylthiadiazole-5-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C24H26N4O2S
(6S)-4-ethyl-1-(4-methylthiadiazole-5-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one —— C26H26FN3O2
(6S)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H33N5O
(6R)-4-ethyl-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(6-oxo-1H-pyridazine-3-carbonyl)-1,4-diazepan-5-one —— C26H28N4O3
(6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-(6-oxo-1H-pyridazine-3-carbonyl)-1,4-diazepan-5-one