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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(1R)-1-imidazol-1-ylethyl]-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrimidin-4-one —— C15H21N5O
6-[(1R)-1-imidazol-1-ylethyl]-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H34N4O3
6-(4-methylcyclohexyl)-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N4O2S
6-(4-methylcyclohexyl)-2-[(2S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O2
6-(4-methylcyclohexyl)-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C27H36N4O2
6-(4-methylcyclohexyl)-2-[(2R)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H34N4O3
6-(4-methylcyclohexyl)-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O2S
6-(4-methylcyclohexyl)-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3S)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O2
6-(4-methylcyclohexyl)-2-[(3S)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(4-methylcyclohexyl)-2-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3S)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O2
6-(4-methylcyclohexyl)-2-[(3S)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3S)-1-(oxane-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H38N4O3
6-(4-methylcyclohexyl)-2-[(3S)-1-(oxane-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6aS)-5-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione —— C20H25N3O3
(6aS)-5-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepine-6,11-dione
—— 6-(4-methylcyclohexyl)-2-[(3R)-1-(oxane-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H38N4O3
6-(4-methylcyclohexyl)-2-[(3R)-1-(oxane-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N4O2S
6-(4-methylcyclohexyl)-2-[(2S)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H34N4O2
6-(4-methylcyclohexyl)-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3S)-1-(pyridine-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(4-methylcyclohexyl)-2-[(3S)-1-(pyridine-4-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[4-[(4-chlorophenyl)methoxy]-3-methoxyphenyl]-4-oxo-2-sulfanylidene-1H-pyrimidine-5-carbonitrile —— C19H14ClN3O3S
6-[4-[(4-chlorophenyl)methoxy]-3-methoxyphenyl]-4-oxo-2-sulfanylidene-1H-pyrimidine-5-carbonitrile
—— 6-(Dimethylsulfamoyl)-2-(2-ethoxyphenyl)quinoline-4-carboxylic acid —— C20H20N2O5S
6-(Dimethylsulfamoyl)-2-(2-ethoxyphenyl)quinoline-4-carboxylic acid
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N4O2S
6-(4-methylcyclohexyl)-2-[(2R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O2
6-(4-methylcyclohexyl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[4-[(4-Chlorophenyl)methyl]piperazine-1-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one —— C22H23ClN4O2
6-[4-[(4-Chlorophenyl)methyl]piperazine-1-carbonyl]-2-phenyl-4,5-dihydropyridazin-3-one
—— 6-Amino-4-(5-nitrothiophen-2-yl)-3-(pyridin-2-yl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C16H10N6O3S
6-Amino-4-(5-nitrothiophen-2-yl)-3-(pyridin-2-yl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H34N4O2
6-(4-methylcyclohexyl)-2-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3R)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O2
6-(4-methylcyclohexyl)-2-[(3R)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O2
6-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(3R)-1-(pyridine-3-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(4-methylcyclohexyl)-2-[(3R)-1-(pyridine-3-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H28N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O2S
6-(4-methylcyclohexyl)-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1S,2S)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1S,2S)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one
—— 6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexanecarbonyl)-2-[(2R)-1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(cyclohexanecarbonyl)-2-[(2R)-1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-acetyl-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H26N4O3
6-acetyl-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexanecarbonyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(cyclohexanecarbonyl)-2-[(2R)-1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(2-cyclopentylacetyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O2
6-(4-methylcyclohexyl)-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Chloro-3-ethyl-2-[1-(3-methylpiperazin-1-yl)ethyl]quinazolin-4-one —— C17H23ClN4O
6-Chloro-3-ethyl-2-[1-(3-methylpiperazin-1-yl)ethyl]quinazolin-4-one
—— (6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1R,2S)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1R,2S)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one
—— 6-Chloro-2-(3,4-dimethylphenyl)-8-fluoroquinoline-4-carboxylic acid —— C18H13ClFNO2
6-Chloro-2-(3,4-dimethylphenyl)-8-fluoroquinoline-4-carboxylic acid
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C27H36N4O2
6-(4-methylcyclohexyl)-2-[(2S)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H28N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexanecarbonyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-(cyclohexanecarbonyl)-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-acetyl-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H26N4O3
6-acetyl-2-[(2R)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H28N4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-acetyl-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H26N4O3
6-acetyl-2-[(2R)-1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one