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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-1-(4-ethylthiadiazole-5-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C23H24N4O2S
(6R)-1-(4-ethylthiadiazole-5-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-ethyl-5-methyl-2-oxo-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]-1H-pyridine-3-carboxamide —— C22H22N6O2S
6-ethyl-5-methyl-2-oxo-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]-1H-pyridine-3-carboxamide
—— 6-[[1-(3-Chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-methylpropyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H22ClN5OS
6-[[1-(3-Chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-methylpropyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-ethyl-3-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C20H21F3N4O
6-ethyl-3-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— 6-ethyl-5-methyl-3-[4-[6-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H23F3N4O3
6-ethyl-5-methyl-3-[4-[6-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (6S)-1-(4-ethylthiadiazole-5-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C23H24N4O2S
(6S)-1-(4-ethylthiadiazole-5-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-ethyl-N-[2-[3-(4-fluorophenyl)-5-pyridin-3-ylpyrazol-1-yl]ethyl]-5-methyl-2-oxo-1H-pyridine-3-carboxamide —— C25H24FN5O2
6-ethyl-N-[2-[3-(4-fluorophenyl)-5-pyridin-3-ylpyrazol-1-yl]ethyl]-5-methyl-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-4-ethyl-1-(4-ethylthiadiazole-5-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6R)-4-ethyl-1-(4-ethylthiadiazole-5-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-ethyl-5-methyl-3-[(3R)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H23F3N4O3
6-ethyl-5-methyl-3-[(3R)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (6R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O3
(6R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O3
(6S)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[3-[16-[3-(3,8-Diamino-5-methylphenanthridin-5-ium-6-yl)phenoxy]hexadecoxy]phenyl]-5-methylphenanthridin-5-ium-3,8-diamine —— C56H66N6O2+2
6-[3-[16-[3-(3,8-Diamino-5-methylphenanthridin-5-ium-6-yl)phenoxy]hexadecoxy]phenyl]-5-methylphenanthridin-5-ium-3,8-diamine
—— (6R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O4
(6R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-bromo-1-(2,4-difluorophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C17H13BrF2N2
6-bromo-1-(2,4-difluorophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— (6S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O4
(6S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-bromo-1-[3-methoxy-4-(2-phenylethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C26H25BrN2O2
6-bromo-1-[3-methoxy-4-(2-phenylethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-[[1-(3,5-Dichlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-methylpropyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H21Cl2N5OS
6-[[1-(3,5-Dichlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-methylpropyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-1-(5-ethyl-2,4-dimethylpyrazole-3-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H32N4O2
(6R)-1-(5-ethyl-2,4-dimethylpyrazole-3-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-(5-ethyl-2,4-dimethylpyrazole-3-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H32N4O2
(6S)-1-(5-ethyl-2,4-dimethylpyrazole-3-carbonyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O4
(6R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H29N3O4
(6S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H22N4O3
6-[1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H22N4O3
6-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[3-[8-[3-(3,8-Diamino-5-methylphenanthridin-5-ium-6-yl)phenoxy]octoxy]phenyl]-5-methylphenanthridin-5-ium-3,8-diamine —— C48H50N6O2+2
6-[3-[8-[3-(3,8-Diamino-5-methylphenanthridin-5-ium-6-yl)phenoxy]octoxy]phenyl]-5-methylphenanthridin-5-ium-3,8-diamine
—— 6-[4-(3-Methoxyphenyl)piperazine-1-carbonyl]-2-(3-methylphenyl)-4,5-dihydropyridazin-3-one —— C23H26N4O3
6-[4-(3-Methoxyphenyl)piperazine-1-carbonyl]-2-(3-methylphenyl)-4,5-dihydropyridazin-3-one
—— 6-ethylsulfonyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H25N5O4S
6-ethylsulfonyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-(1-ethylsulfonylpiperidine-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H28N4O4S
6-[1-(1-ethylsulfonylpiperidine-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-(cyclohexanecarbonyl)-2-[(2R)-1-ethylsulfonylpiperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H32N4O4S
6-(cyclohexanecarbonyl)-2-[(2R)-1-ethylsulfonylpiperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Furan-2-ylmethylidene)-3-(4-methylphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C16H11N3O2S
6-(Furan-2-ylmethylidene)-3-(4-methylphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-ethylsulfonyl-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2R)-1-(2-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(thiophene-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H24N4O4S2
6-ethylsulfonyl-2-[(2S)-1-(thiophene-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2R)-1-(4-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2R)-1-(4-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(3R)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(3R)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(3R)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H23N5O4S
6-ethylsulfonyl-2-[(3R)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-ethylsulfonyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C21H26N2O4S
(6R)-1-ethylsulfonyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-ethylsulfonyl-2-[(3S)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(3S)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H25N5O4S
6-ethylsulfonyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(2-ethoxybenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N2O3S
(6S)-1-(2-ethoxybenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-ethylsulfonyl-2-[(3S)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H23N5O4S
6-ethylsulfonyl-2-[(3S)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(3R)-1-[2-(4-methylphenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(3R)-1-[2-(4-methylphenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-ethylsulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C21H25FN2O4S
(6R)-1-ethylsulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-ethylsulfonyl-2-[(2R)-1-(2-pyridin-3-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H27N5O4S
6-ethylsulfonyl-2-[(2R)-1-(2-pyridin-3-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H25FN4O4S
6-ethylsulfonyl-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H25FN4O4S
6-ethylsulfonyl-2-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(3S)-1-(2-phenylacetyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H26N4O4S
6-ethylsulfonyl-2-[(3S)-1-(2-phenylacetyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H25N5O4S
6-ethylsulfonyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethylsulfonyl-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O4S
6-ethylsulfonyl-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-ethylsulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C21H25FN2O4S
(6S)-1-ethylsulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one