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—— (6S)-6-[[2-(3-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one —— C25H29FN2O3
(6S)-6-[[2-(3-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one
—— (6R)-1-(2-methoxyacetyl)-6-[(2-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C24H28N2O3
(6R)-1-(2-methoxyacetyl)-6-[(2-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-(2-methoxyacetyl)-2-[(2R)-1-(3-methoxybenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28N4O5
6-(2-methoxyacetyl)-2-[(2R)-1-(3-methoxybenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one —— C25H29FN2O3
(6S)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H28N4O4
6-(cyclopropanecarbonyl)-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H26N4O4
6-(cyclopropanecarbonyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H34N4O3
6-(cyclohexylmethyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-cyclohexylacetyl)-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N4O4
6-(2-cyclohexylacetyl)-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(2-methoxyacetyl)-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H27N3O3
(6S)-1-(2-methoxyacetyl)-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[1-[(1R,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H27N3O3
6-[1-[(1R,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6R)-1-(3-methoxypropanoyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C25H30N2O3
(6R)-1-(3-methoxypropanoyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[(3R)-1-(cyclopropanecarbonyl)piperidin-3-yl]-2-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrimidin-4-one —— C21H30N4O4
6-[(3R)-1-(cyclopropanecarbonyl)piperidin-3-yl]-2-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrimidin-4-one
—— 6-(2-methoxyacetyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H26N4O4S
6-(2-methoxyacetyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H27N3O3
6-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H27N3O3
6-[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6S)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one —— C25H29FN2O3
(6S)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[(3R)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C17H20N4O3
6-[(3R)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H30N4O4
6-(cyclopentanecarbonyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one —— C25H29FN2O3
(6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(3-methoxypropanoyl)-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-(2-cyclopentylacetyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N4O4
6-(2-cyclopentylacetyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(3-methoxypropanoyl)-6-[(2-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C25H30N2O3
(6R)-1-(3-methoxypropanoyl)-6-[(2-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-(4-fluorobenzoyl)-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H23FN4O4
6-(4-fluorobenzoyl)-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-methoxyacetyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H25N5O4
6-(2-methoxyacetyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexanecarbonyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N4O4
6-(cyclohexanecarbonyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine —— C24H29N5O2
6-[1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[(3S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C19H22N6OS
6-[(3S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— (6S)-1-(3-methoxypropanoyl)-4-prop-2-enyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O3
(6S)-1-(3-methoxypropanoyl)-4-prop-2-enyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(2-cyclopentylacetyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N4O4
6-(2-cyclopentylacetyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H30N4O4
6-(cyclopentanecarbonyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H26N4O4
6-(cyclopropanecarbonyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3S)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine —— C24H29N5O2
6-[(3S)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyrazin-2-ylpyrimidin-4-amine —— C22H25FN6O
6-[1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyrazin-2-ylpyrimidin-4-amine
—— 6-[(3R)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine —— C22H24FN5
6-[(3R)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-Tert-butyl-N,N-diethyl-2-(2-fluorobenzamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H31FN2O2S
6-Tert-butyl-N,N-diethyl-2-(2-fluorobenzamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(3R)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine —— C23H26FN5O
6-[(3R)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[(3R)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C21H22FN5O2S
6-[(3R)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— (6-methoxycarbonyl-2-methyl-4-oxo-1H-quinolin-3-yl)methyl-methyl-(1-methylpiperidin-1-ium-4-yl)azanium —— C20H29N3O3+2
(6-methoxycarbonyl-2-methyl-4-oxo-1H-quinolin-3-yl)methyl-methyl-(1-methylpiperidin-1-ium-4-yl)azanium
—— 6-cyclopropyl-2-[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C20H29N3O3
6-cyclopropyl-2-[1-[(1S,3S)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— 6-cyclopropyl-2-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C20H29N3O3
6-cyclopropyl-2-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— 6-[(3S)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine —— C22H24FN5
6-[(3S)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[1-(2-methoxyphenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C22H25N5O3S
6-[1-(2-methoxyphenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C22H25N5O3S
6-[(3R)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-(1-cyclopentylpiperidin-4-yl)-N-methyl-2-pyridin-4-ylpyrimidin-4-amine —— C20H27N5
6-(1-cyclopentylpiperidin-4-yl)-N-methyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[1-(4-fluorophenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C21H22FN5O2S
6-[1-(4-fluorophenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C23H27N5O
6-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[(3R)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C22H24FN5
6-[(3R)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-cyclopropyl-2-[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C20H29N3O3
6-cyclopropyl-2-[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— (6,7-dimethoxy-1-thiophen-2-yl-3,4-dihydro-1H-isoquinolin-2-yl)-(4-phenylphenyl)methanone —— C28H25NO3S
(6,7-dimethoxy-1-thiophen-2-yl-3,4-dihydro-1H-isoquinolin-2-yl)-(4-phenylphenyl)methanone
—— (6S)-1-(2-methoxyacetyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C24H28N2O3
(6S)-1-(2-methoxyacetyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C24H29N5O2
6-[1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine