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—— (6R)-6-N-benzyl-2-N-[2-(3,4-diethoxyphenyl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C29H35N5O5
(6R)-6-N-benzyl-2-N-[2-(3,4-diethoxyphenyl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-N-cyclopentyl-5-ethyl-6-methyl-2-[4-(4-nitrophenyl)piperazine-1-carbonyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H33N7O5
(6S)-N-cyclopentyl-5-ethyl-6-methyl-2-[4-(4-nitrophenyl)piperazine-1-carbonyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-N-[3-(azepan-1-yl)propyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H40N6O3
(6S)-2-N-[3-(azepan-1-yl)propyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C22H33N5O5
(6S)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H28FN5O5
(6S)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-6-N-benzyl-5,6-dimethyl-4-oxo-2-N-[(3,4,5-trimethoxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H31N5O6
(6S)-6-N-benzyl-5,6-dimethyl-4-oxo-2-N-[(3,4,5-trimethoxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-[3-(azepan-1-yl)propyl]-6-N-benzyl-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H36N6O3
(6R)-2-N-[3-(azepan-1-yl)propyl]-6-N-benzyl-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-N-cyclopentyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C22H31N5O5
(6S)-N-cyclopentyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-(azepane-1-carbonyl)-N-benzyl-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H29N5O3
(6R)-2-(azepane-1-carbonyl)-N-benzyl-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H35N5O5
(6R)-N-cycloheptyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H33N5O5
(6R)-N-cyclohexyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-N-[(4-butoxyphenyl)methyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H37N5O4
(6R)-2-N-[(4-butoxyphenyl)methyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-[3-(azepan-1-yl)propyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H40N6O3
(6R)-2-N-[3-(azepan-1-yl)propyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(4-ethoxyphenyl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C28H39N5O4
(6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(4-ethoxyphenyl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H31N5O5
(6R)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-N-[2-(azepan-1-yl)ethyl]-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33FN6O3
(6R)-2-N-[2-(azepan-1-yl)ethyl]-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C22H33N5O5
(6R)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-(azepane-1-carbonyl)-N-cyclopentyl-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H35N5O3
(6S)-2-(azepane-1-carbonyl)-N-cyclopentyl-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-N-cyclooctyl-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H32FN5O3
(6S)-2-N-cyclooctyl-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-[3-(azepan-1-yl)propyl]-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H38N6O3
(6R)-2-N-[3-(azepan-1-yl)propyl]-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-benzyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H29N5O5
(6R)-N-benzyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-N-(3-butylsulfanylpropyl)-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H35N5O3S
(6S)-2-N-(3-butylsulfanylpropyl)-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H28FN5O5
(6R)-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-N-cyclooctyl-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H32FN5O3
(6R)-2-N-cyclooctyl-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-cyclopentyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H35N5O5
(6R)-N-cyclopentyl-2-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-amino-1-benzyl-3-ethyl-5-[2-[methyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]acetyl]pyrimidine-2,4-dione —— C25H26N6O4
6-amino-1-benzyl-3-ethyl-5-[2-[methyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]acetyl]pyrimidine-2,4-dione
—— 6-[[1-(2-Chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H24ClN5OS
6-[[1-(2-Chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[[1-(5-Chloro-2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-methyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H20ClN5O3S
6-[[1-(5-Chloro-2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-methyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-Amino-4-(2-chlorophenyl)-3-(thiophen-2-yl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C17H11ClN4OS
6-Amino-4-(2-chlorophenyl)-3-(thiophen-2-yl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-[[1-(5-Chloro-2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H18ClN5O3S
6-[[1-(5-Chloro-2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-N-(3-{[3-(trifluoromethyl)phenyl]sulfamoyl}phenyl)pyridine-3-carboxamide —— C19H13ClF3N3O3S
6-chloro-N-(3-{[3-(trifluoromethyl)phenyl]sulfamoyl}phenyl)pyridine-3-carboxamide
—— 6-[[5-[[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]sulfonyl]thiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione —— C21H23N3O4S2
6-[[5-[[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]sulfonyl]thiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-thiophen-2-ylprop-2-enoate —— C16H13NO6S
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 3-thiophen-2-ylprop-2-enoate
—— 6-[[5-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonylthiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione —— C19H21N3O4S2
6-[[5-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonylthiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-[[5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylthiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione —— C19H21N3O4S2
6-[[5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylthiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-Nitro-2-[2-(3-phenylmethoxyphenyl)ethenyl]-1,3-benzothiazole —— C22H16N2O3S
6-Nitro-2-[2-(3-phenylmethoxyphenyl)ethenyl]-1,3-benzothiazole
—— 6-chloro-4-phenyl-3-{[4-(prop-2-en-1-yl)-5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}quinolin-2(1H)-one —— C25H18ClN5OS
6-chloro-4-phenyl-3-{[4-(prop-2-en-1-yl)-5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}quinolin-2(1H)-one
—— 6-chloro-1-(4-chlorophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C17H14Cl2N2
6-chloro-1-(4-chlorophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-[[3-Ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O4S
6-[[3-Ethoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[[4-[4-[(Dibenzylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C39H44N2O6
6-[[4-[4-[(Dibenzylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-amino-1-benzyl-3-methyl-5-[2-(3H-[1,2,4]triazolo[4,3-a]benzimidazol-1-ylsulfanyl)acetyl]pyrimidine-2,4-dione —— C22H19N7O3S
6-amino-1-benzyl-3-methyl-5-[2-(3H-[1,2,4]triazolo[4,3-a]benzimidazol-1-ylsulfanyl)acetyl]pyrimidine-2,4-dione
—— 6-acetyl-2-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one —— C28H23BrN2O5S
6-acetyl-2-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one
—— 6-fluoro-1-[3-(2-phenylethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C25H23FN2O
6-fluoro-1-[3-(2-phenylethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-chloro-N-(3-chloro-4-methylphenyl)-2-methylquinolin-1-ium-4-amine —— C17H15Cl2N2+
6-chloro-N-(3-chloro-4-methylphenyl)-2-methylquinolin-1-ium-4-amine
—— 6-acetyl-2-[[4-(diethylamino)-2-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one —— C32H33N3O4S
6-acetyl-2-[[4-(diethylamino)-2-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one
—— 6-[(5-Bromo-2-methoxyphenyl)methylidene]-5-imino-2-thiophen-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C17H11BrN4O2S2
6-[(5-Bromo-2-methoxyphenyl)methylidene]-5-imino-2-thiophen-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-acetyl-2-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one —— C35H29FN2O5S
6-acetyl-2-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one
—— 6-acetyl-2-[(4-hydroxyphenyl)methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one —— C27H22N2O4S
6-acetyl-2-[(4-hydroxyphenyl)methylidene]-5-(2-methoxynaphthalen-1-yl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-3-one
—— 6-Hydroxy-5-[[6-hydroxy-1-(2-methylphenyl)-4-oxo-2-sulfanylidenepyrimidin-5-yl]-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-1-(2-methylphenyl)-2-sulfanylidenepyrimidin-4-one —— C35H35N5O5S2
6-Hydroxy-5-[[6-hydroxy-1-(2-methylphenyl)-4-oxo-2-sulfanylidenepyrimidin-5-yl]-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-1-(2-methylphenyl)-2-sulfanylidenepyrimidin-4-one
—— 6-Hydroxy-5-{[4-hydroxy-1-(2-methylphenyl)-6-oxo-2-sulfanyl-1,6-dihydropyrimidin-5-yl][4-methoxy-3-(pyrrolidinium-1-ylmethyl)phenyl]methyl}-1-(2-methylphenyl)-4-oxo-1,4-dihydropyrimidine-2-thiolate —— C35H35N5O5S2
6-Hydroxy-5-{[4-hydroxy-1-(2-methylphenyl)-6-oxo-2-sulfanyl-1,6-dihydropyrimidin-5-yl][4-methoxy-3-(pyrrolidinium-1-ylmethyl)phenyl]methyl}-1-(2-methylphenyl)-4-oxo-1,4-dihydropyrimidine-2-thiolate