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—— [(6S,7S)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C24H27N5OS
[(6S,7S)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2S)-2-methylcyclohexyl]hexanamide —— C25H37N3O5
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2S)-2-methylcyclohexyl]hexanamide
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2R)-2-methylcyclohexyl]hexanamide —— C25H37N3O5
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2R)-2-methylcyclohexyl]hexanamide
—— 6-(3-Chlorophenoxy)-5-nitroimidazo[2,1-b][1,3]thiazole —— C11H6ClN3O3S
6-(3-Chlorophenoxy)-5-nitroimidazo[2,1-b][1,3]thiazole
—— (6R,7R)-6-(4-chlorophenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H22ClN5O2S
(6R,7R)-6-(4-chlorophenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S,8R)-6-methoxy-6,7-dimethyl-8-naphthalen-1-yl-7,8-dihydro-[1,3]dioxolo[4,5-g]chromene —— C23H22O4
(6S,7S,8R)-6-methoxy-6,7-dimethyl-8-naphthalen-1-yl-7,8-dihydro-[1,3]dioxolo[4,5-g]chromene
—— (6S,7S)-6-(4-fluorophenyl)-N-[(4-methoxyphenyl)methyl]-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C25H22FN5O2S
(6S,7S)-6-(4-fluorophenyl)-N-[(4-methoxyphenyl)methyl]-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]hexanamide —— C26H39N3O5
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]hexanamide
—— (6R,7S)-6-(4-chlorophenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H22ClN5OS
(6R,7S)-6-(4-chlorophenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7R)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20ClN5O2S
(6R,7R)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[[(1R)-1-[(1,3-dioxoisoindol-2-yl)methyl]-3,4-dihydro-1H-isoquinolin-2-yl]sulfonyl]-1,4-dihydroquinoxaline-2,3-dione —— C26H20N4O6S
6-[[(1R)-1-[(1,3-dioxoisoindol-2-yl)methyl]-3,4-dihydro-1H-isoquinolin-2-yl]sulfonyl]-1,4-dihydroquinoxaline-2,3-dione
—— (6R,7S)-N-(furan-2-ylmethyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C23H21N5O2S
(6R,7S)-N-(furan-2-ylmethyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7R)-6-(4-chlorophenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H22ClN5OS
(6R,7R)-6-(4-chlorophenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S)-N-(3-methoxyphenyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C25H23N5O2S
(6S,7S)-N-(3-methoxyphenyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-(4-Methoxyphenyl)-2-[(3,4,4-trifluoro-3-butenyl)sulfanyl][1,2,4]triazolo[1,5-a]pyrimidin-7-ylamine —— C16H14F3N5OS
6-(4-Methoxyphenyl)-2-[(3,4,4-trifluoro-3-butenyl)sulfanyl][1,2,4]triazolo[1,5-a]pyrimidin-7-ylamine
—— [(6-Methyl-2,3-dihydrothiochromen-4-ylidene)amino] 4-fluorobenzoate —— C17H14FNO2S
[(6-Methyl-2,3-dihydrothiochromen-4-ylidene)amino] 4-fluorobenzoate
—— [(6R,7R)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C24H27N5OS
[(6R,7R)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— 6-(5-ethoxy-6-oxocyclohexa-2,4-dien-1-ylidene)-3-(4-ethoxyphenyl)-1,2-dihydropyrazolo[3,4-b]pyridine-4-carboxylic acid —— C23H21N3O5
6-(5-ethoxy-6-oxocyclohexa-2,4-dien-1-ylidene)-3-(4-ethoxyphenyl)-1,2-dihydropyrazolo[3,4-b]pyridine-4-carboxylic acid
—— 6-[3-(dimethylamino)acryloyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C11H11N3O2S
6-[3-(dimethylamino)acryloyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— [(6S,7S)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C22H23N5O3S
[(6S,7S)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— [(6R,7S)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C24H27N5OS
[(6R,7S)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— 6-[(5R,10bR)-9-bromo-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C22H18BrN3O2
6-[(5R,10bR)-9-bromo-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6S,7R)-N-(furan-2-ylmethyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C23H21N5O2S
(6S,7R)-N-(furan-2-ylmethyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-(4-Methoxyphenyl)-5-methyl-3-(2-pyridinyl)pyrazolo[1,5-a]pyrimidin-7-ylamine —— C19H17N5O
6-(4-Methoxyphenyl)-5-methyl-3-(2-pyridinyl)pyrazolo[1,5-a]pyrimidin-7-ylamine
—— [(6R,7R)-6-(4-ethoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C25H29N5O2S
[(6R,7R)-6-(4-ethoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— (6S,7S)-6-(4-methoxyphenyl)-3-phenyl-N,N-dipropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C24H29N5O2S
(6S,7S)-6-(4-methoxyphenyl)-3-phenyl-N,N-dipropyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7R)-6-(4-methylphenyl)-3-phenyl-N-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C27H27N5OS
(6S,7R)-6-(4-methylphenyl)-3-phenyl-N-(2,4,6-trimethylphenyl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bS)-9-bromo-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C22H18BrN3O2
6-[(5R,10bS)-9-bromo-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6S,7S)-N-(furan-2-ylmethyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C23H21N5O2S
(6S,7S)-N-(furan-2-ylmethyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— [(6S,7S)-6-(4-ethoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C25H29N5O2S
[(6S,7S)-6-(4-ethoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— (6S,7R)-6-(4-chlorophenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H22ClN5O2S
(6S,7R)-6-(4-chlorophenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— [(6R,7S)-6-(4-ethoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone —— C25H29N5O2S
[(6R,7S)-6-(4-ethoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-[(2S)-2-methylpiperidin-1-yl]methanone
—— [(6R,7R)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C22H23N5O3S
[(6R,7R)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— 6-(methylsulfanyl)-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl 3-(trifluoromethyl)phenyl ether —— C19H13F3N4OS
6-(methylsulfanyl)-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl 3-(trifluoromethyl)phenyl ether
—— (6R,7R)-N-(3-methoxyphenyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C25H23N5O2S
(6R,7R)-N-(3-methoxyphenyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20ClN5O2S
(6S,7S)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bS)-9-bromo-5-pyridin-4-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C22H18BrN3O3
6-[(5R,10bS)-9-bromo-5-pyridin-4-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— (6S,7R)-N-(3-methoxyphenyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C25H23N5O2S
(6S,7R)-N-(3-methoxyphenyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bR)-9-bromo-5-pyridin-4-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C22H18BrN3O3
6-[(5R,10bR)-9-bromo-5-pyridin-4-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-9-bromo-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C22H18BrN3O3
6-[(5R,10bS)-9-bromo-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]hexanamide —— C26H39N3O5
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]hexanamide
—— [(6R,7S)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C22H23N5O3S
[(6R,7S)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— (6S,7S)-6-(4-methoxyphenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C22H25N5O3S
(6S,7S)-6-(4-methoxyphenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6-((2,4-Dichlorophenyl)sulfanyl)-2-methyl-4-pyrimidinyl)methyl phenyl sulfone —— C18H14Cl2N2O2S2
(6-((2,4-Dichlorophenyl)sulfanyl)-2-methyl-4-pyrimidinyl)methyl phenyl sulfone
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[[(2S)-oxolan-2-yl]methyl]hexanamide —— C23H33N3O6
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[[(2S)-oxolan-2-yl]methyl]hexanamide
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]hexanamide —— C26H39N3O5
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]hexanamide
—— 6-chloro-1-{[(dimethylamino)carbonyl]oxy}-2-(4-methoxyphenyl)-1H-1,3-benzimidazole —— C17H16ClN3O3
6-chloro-1-{[(dimethylamino)carbonyl]oxy}-2-(4-methoxyphenyl)-1H-1,3-benzimidazole
—— 6-(3,4-dichlorophenyl)-2H-pyrazolo[3,4-b]pyridin-3-amine —— C12H8Cl2N4
6-(3,4-dichlorophenyl)-2H-pyrazolo[3,4-b]pyridin-3-amine
—— 6-[(E)-3-(dimethylamino)prop-2-enoyl]-4-methyl-2-[4-(trifluoromethyl)phenyl]-1,2,4-triazine-3,5-dione —— C16H15F3N4O3
6-[(E)-3-(dimethylamino)prop-2-enoyl]-4-methyl-2-[4-(trifluoromethyl)phenyl]-1,2,4-triazine-3,5-dione
—— 6-(4-Chlorophenyl)-2-(2,4-difluorophenoxy)-4-(trifluoromethyl)pyridine-3-carbonitrile —— C19H8ClF5N2O
6-(4-Chlorophenyl)-2-(2,4-difluorophenoxy)-4-(trifluoromethyl)pyridine-3-carbonitrile