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—— 6-[(3-chlorophenyl)methylsulfonyl]-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C20H26ClN5O2S
6-[(3-chlorophenyl)methylsulfonyl]-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-[(2S)-1-(1-ethylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C20H30N4O4S
6-[(2S)-1-(1-ethylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2S)-1-(4-methoxy-2-methyl-5-propan-2-ylphenyl)sulfonylpyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C22H29N3O4S
6-[(2S)-1-(4-methoxy-2-methyl-5-propan-2-ylphenyl)sulfonylpyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-(4-ethoxyphenyl)-3-(4-ethylphenyl)-2,5-bis(sulfanylidene)-4H-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C21H19N3O2S3
6-(4-ethoxyphenyl)-3-(4-ethylphenyl)-2,5-bis(sulfanylidene)-4H-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 6-[(2R)-1-[4-(2-fluorophenoxy)butanoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C22H26FN3O3
6-[(2R)-1-[4-(2-fluorophenoxy)butanoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2S)-1-[4-(2-fluorophenoxy)butanoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C22H26FN3O3
6-[(2S)-1-[4-(2-fluorophenoxy)butanoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2R)-1-[(1-ethylimidazol-2-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H28FN5O
6-[(2R)-1-[(1-ethylimidazol-2-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H25FN4O3
6-[(2S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-(1,3-dimethyl-2-oxobenzimidazol-5-yl)sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C21H25N5O4S
6-[(2S)-1-(1,3-dimethyl-2-oxobenzimidazol-5-yl)sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C25H30FN5O
6-[(2R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C25H29FN6O
6-[(2S)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[[3-(4-methoxyphenyl)phenyl]methyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C25H27N3O2
6-[(2R)-1-[[3-(4-methoxyphenyl)phenyl]methyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H25FN4O3
6-[(2R)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H25FN4O3
6-[(2S)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C26H30FN5O
6-[(2S)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[2-[cyclohexyl(methylsulfonyl)amino]acetyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C20H30N4O4S
6-[(2R)-1-[2-[cyclohexyl(methylsulfonyl)amino]acetyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[1-[(4-fluorophenyl)methyl]piperidine-4-carbonyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C24H29FN4O2
6-[(2R)-1-[1-[(4-fluorophenyl)methyl]piperidine-4-carbonyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-(1,3-dimethyl-2-oxobenzimidazol-5-yl)sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C21H25N5O4S
6-[(2R)-1-(1,3-dimethyl-2-oxobenzimidazol-5-yl)sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2R)-1-(1-ethylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C20H30N4O4S
6-[(2R)-1-(1-ethylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2R)-1-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C22H28N4O4S
6-[(2R)-1-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2S)-1-[2-fluoro-5-(methylsulfamoyl)benzoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C20H23FN4O4S
6-[(2S)-1-[2-fluoro-5-(methylsulfamoyl)benzoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-[(2R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H25FN4O3
6-[(2R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H28FN5O
6-[(2S)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C25H29FN6O
6-[(2R)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-(4-Hydroxyphenyl)-9-(3,4,5-trimethoxyphenyl)-5,6,6a,8,9,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H28N2O5
6-(4-Hydroxyphenyl)-9-(3,4,5-trimethoxyphenyl)-5,6,6a,8,9,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[(2R)-1-(4-methoxy-2-methyl-5-propan-2-ylphenyl)sulfonylpyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C22H29N3O4S
6-[(2R)-1-(4-methoxy-2-methyl-5-propan-2-ylphenyl)sulfonylpyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C26H30FN5O
6-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-(benzenesulfonyl)-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C19H25N5O2S
6-(benzenesulfonyl)-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-[(2S)-1-[1-[(4-fluorophenyl)methyl]piperidine-4-carbonyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C24H29FN4O2
6-[(2S)-1-[1-[(4-fluorophenyl)methyl]piperidine-4-carbonyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-[[3-(4-methoxyphenyl)phenyl]methyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C25H27N3O2
6-[(2S)-1-[[3-(4-methoxyphenyl)phenyl]methyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2S)-1-[2-[cyclohexyl(methylsulfonyl)amino]acetyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide —— C20H30N4O4S
6-[(2S)-1-[2-[cyclohexyl(methylsulfonyl)amino]acetyl]pyrrolidin-2-yl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H28FN5O
6-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— (6-fluoro-1H-indol-2-yl)-[3-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone —— C20H23FN6O
(6-fluoro-1H-indol-2-yl)-[3-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone
—— (6-chloro-1H-indol-2-yl)-[3-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone —— C20H23ClN6O
(6-chloro-1H-indol-2-yl)-[3-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone
—— (6-fluoro-1H-indol-2-yl)-[3-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone —— C20H23FN6O
(6-fluoro-1H-indol-2-yl)-[3-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone
—— (6-chloro-1H-indol-2-yl)-[3-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone —— C20H23ClN6O
(6-chloro-1H-indol-2-yl)-[3-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone
—— 6a,9a-Dichloro-6-(2-chloro-4-hydroxyphenyl)-2-(4-iodophenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C32H17Cl3F5IN2O5
6a,9a-Dichloro-6-(2-chloro-4-hydroxyphenyl)-2-(4-iodophenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-[6a-(4-chlorophenyl)-8-(4-fluoroanilino)-6-(2-hydroxy-6-methoxyphenyl)-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C39H37ClFN3O8
6-[6a-(4-chlorophenyl)-8-(4-fluoroanilino)-6-(2-hydroxy-6-methoxyphenyl)-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— 6-bromo-3,3-bis(morpholin-4-ylmethyl)-8-nitro-2H-chromen-4-one —— C19H24BrN3O6
6-bromo-3,3-bis(morpholin-4-ylmethyl)-8-nitro-2H-chromen-4-one
—— 6-(3-Bromo-4-hydroxy-5-methoxyphenyl)-8-(bromomethyl)-6a,9a-dichloro-2-(4-ethenylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C30H24Br2Cl2N2O6
6-(3-Bromo-4-hydroxy-5-methoxyphenyl)-8-(bromomethyl)-6a,9a-dichloro-2-(4-ethenylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6a,9a-Dichloro-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-(2-hydroxy-3-methylphenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H24Cl2F5N5O9
6a,9a-Dichloro-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-(2-hydroxy-3-methylphenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6-fluoro-1H-indol-2-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone —— C19H21FN6O
(6-fluoro-1H-indol-2-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone
—— 6-(3-Bromo-4-hydroxy-5-methoxyphenyl)-6a,9a-dichloro-2-(4-nitrophenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C33H19BrCl2F5N3O8
6-(3-Bromo-4-hydroxy-5-methoxyphenyl)-6a,9a-dichloro-2-(4-nitrophenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6a,9a-Dichloro-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-(3-ethoxy-4-hydroxyphenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C44H33Cl2F5N2O8
6a,9a-Dichloro-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-(3-ethoxy-4-hydroxyphenyl)-8-(2,3,4,5,6-pentafluorophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— [6-[[3-[[1-Hydroxy-5-[(2-methylpropan-2-yl)oxy]-5-oxopentan-2-yl]amino]-3-oxopropyl]carbamoyl]-2,2-diphenyl-3a,4,5,7a-tetrahydro-1,3-benzodioxol-4-yl] 3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]benzoate —— C47H54N2O10
[6-[[3-[[1-Hydroxy-5-[(2-methylpropan-2-yl)oxy]-5-oxopentan-2-yl]amino]-3-oxopropyl]carbamoyl]-2,2-diphenyl-3a,4,5,7a-tetrahydro-1,3-benzodioxol-4-yl] 3-[2-(7-oxabicyclo[4.1.0]heptan-3-yl)ethenyl]benzoate
—— (6-chloro-1H-indol-2-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone —— C19H21ClN6O
(6-chloro-1H-indol-2-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone
—— [6'-[[3-(2-Hydroxyethylcarbamoyl)phenyl]methylcarbamoyl]spiro[1,3-dihydroindene-2,2'-3a,4,5,7a-tetrahydro-1,3-benzodioxole]-4'-yl] 3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]benzoate —— C38H35F3N2O9
[6'-[[3-(2-Hydroxyethylcarbamoyl)phenyl]methylcarbamoyl]spiro[1,3-dihydroindene-2,2'-3a,4,5,7a-tetrahydro-1,3-benzodioxole]-4'-yl] 3-[3-oxo-3-(2,2,2-trifluoroethoxy)prop-1-enyl]benzoate
—— (6-chloro-1H-indol-2-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone —— C19H21ClN6O
(6-chloro-1H-indol-2-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone
—— 6-Amino-4-(3-bromophenyl)-3-(2-naphthyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C23H15BrN4O
6-Amino-4-(3-bromophenyl)-3-(2-naphthyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-(benzenesulfonyl)-N-methyl-2-(1-methylpiperidin-4-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C20H27N5O2S
6-(benzenesulfonyl)-N-methyl-2-(1-methylpiperidin-4-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine