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—— 6-(3-methylpyridine-4-carbonyl)-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27N5O4
6-(3-methylpyridine-4-carbonyl)-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine —— C22H28N4O2
6-[1-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine
—— 6-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine —— C21H26N4O2
6-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine
—— (6-methoxypyridin-3-yl)-[(2S)-2-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]pyrrolidin-1-yl]methanone —— C22H23N5O2
(6-methoxypyridin-3-yl)-[(2S)-2-[2-methyl-5-(3-methylpyridin-4-yl)pyrimidin-4-yl]pyrrolidin-1-yl]methanone
—— 6-methyl-1-[4-(2-phenylethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C26H26N2O
6-methyl-1-[4-(2-phenylethoxy)phenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— 6-[1-[(5-tert-butyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine —— C20H28N6
6-[1-[(5-tert-butyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine
—— 6-Chloro-2-(3-ethoxyphenyl)-8-fluoroquinoline-4-carboxylic acid —— C18H13ClFNO3
6-Chloro-2-(3-ethoxyphenyl)-8-fluoroquinoline-4-carboxylic acid
—— 6,8-Dichloro-2-(furan-2-yl)quinoline-4-carboxylic acid —— C14H7Cl2NO3
6,8-Dichloro-2-(furan-2-yl)quinoline-4-carboxylic acid
—— 6,7-Dimethoxy-1-[4-(2-methylpropoxy)phenyl]-1,2,3,4-tetrahydroisoquinoline —— C21H27NO3
6,7-Dimethoxy-1-[4-(2-methylpropoxy)phenyl]-1,2,3,4-tetrahydroisoquinoline
—— 6-Chloro-2-(2-ethoxyphenyl)-8-methylquinoline-4-carboxylic acid —— C19H16ClNO3
6-Chloro-2-(2-ethoxyphenyl)-8-methylquinoline-4-carboxylic acid
—— 6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27N5O4
6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,6-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H23N5O3
6-[(2,6-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H21N5O2
6-[(2-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,3-Dichlorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H17Cl2N5O
6-[(2,3-Dichlorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H23N5O3S
6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H21N5O2
6-[(4-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H24N6O3
6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,5-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H23N5O3
6-[(2,5-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,4-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H23N5O3
6-[(2,4-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H18FN5O
6-[(2-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(3S)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O2S
6-(cyclopropanecarbonyl)-2-[(3S)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-Dichlorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H17Cl2N5O
6-[(3,4-Dichlorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,5-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H23N5O3
6-[(3,5-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-Methoxy-2,3-dimethylphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H25N5O2
6-[(4-Methoxy-2,3-dimethylphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(3-chlorophenyl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine —— C19H21ClN4
6-[1-[(3-chlorophenyl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine
—— 6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H24N6O3
6-(3-methylpyridine-4-carbonyl)-2-[(2S)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(5-methylpyrazine-2-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C27H28N4O2
(6S)-1-(5-methylpyrazine-2-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[(2,3-Difluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H17F2N5O
6-[(2,3-Difluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-N-[(1S)-2-(6-oxo-2-propan-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H24N6O2
6-methyl-N-[(1S)-2-(6-oxo-2-propan-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-[(3,4-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H23N5O3
6-[(3,4-Dimethoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H18FN5O
6-[(3-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(5-methylpyrazine-2-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C27H28N4O2
(6R)-1-(5-methylpyrazine-2-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O3S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H21N5O2
6-[(3-Methoxyphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H18FN5O
6-[(4-Fluorophenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O3S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine —— C18H24N6
6-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-3-methyl-5H-pyrrolo[2,3-b]pyrazine
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(2-pyridin-2-ylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27N5O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(2-pyridin-2-ylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2,2-Diphenylacetyl)-2-(3-methoxyphenyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C28H25N3O3
6-(2,2-Diphenylacetyl)-2-(3-methoxyphenyl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O3S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H28N4O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(3R)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H28N4O2S
6-(cyclopropanecarbonyl)-2-[(3R)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H28N4O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[3-(5-methylpyrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C26H30N4O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[3-(5-methylpyrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— 6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O2S
6-[(3-methylthiophen-2-yl)methyl]-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one