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—— 6-fluoro-2-[(3S)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O3
6-fluoro-2-[(3S)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-(4-Methoxyphenyl)sulfonyl-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H17N5O4S
6-(4-Methoxyphenyl)sulfonyl-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-2-[(3R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]quinoline-3-carboxamide —— C24H24FN3O3
6-fluoro-2-[(3R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3R)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide —— C25H26FN3O3
6-fluoro-2-[(3R)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3S)-1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]quinoline-3-carboxamide —— C22H21FN4O3
6-fluoro-2-[(3S)-1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-fluoro-2-[(3R)-1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]quinoline-3-carboxamide —— C22H21FN4O3
6-fluoro-2-[(3R)-1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-benzyl-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-N,N-dimethyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-amine —— C23H31N5O2
6-benzyl-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-N,N-dimethyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-amine
—— 6-Amino-5-[2-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3-methyl-1-(2-methylpropyl)pyrimidine-2,4-dione —— C20H23ClN6O3S
6-Amino-5-[2-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3-methyl-1-(2-methylpropyl)pyrimidine-2,4-dione
—— 6-benzyl-N,N-dimethyl-4-(4-piperidin-1-ylpiperidin-1-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-amine —— C26H38N6
6-benzyl-N,N-dimethyl-4-(4-piperidin-1-ylpiperidin-1-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-amine
—— 6-benzyl-4-[4-(2-methoxyethyl)piperazin-1-yl]-N,N-dimethyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-amine —— C23H34N6O
6-benzyl-4-[4-(2-methoxyethyl)piperazin-1-yl]-N,N-dimethyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-amine
—— 6-(2-Methoxypyridine-4-carbonyl)-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H16N6O3
6-(2-Methoxypyridine-4-carbonyl)-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— [6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C20H17FN4O2S2
[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— [6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C20H17FN4O2S2
[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— [6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2R)-2-(methoxymethyl)piperidin-1-yl]methanone —— C21H25N3O2S
[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2R)-2-(methoxymethyl)piperidin-1-yl]methanone
—— 6-Benzyl-4-<4-methyl-piperazino>-2-pyrrolidino-5,6,7,8-tetrahydro-pyrido<4,3-d>pyrimidin 7212-05-7 C23H32N6
6-Benzyl-4-<4-methyl-piperazino>-2-pyrrolidino-5,6,7,8-tetrahydro-pyrido<4,3-d>pyrimidin
—— [6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2S)-2-(methoxymethyl)piperidin-1-yl]methanone —— C21H25N3O2S
[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-[(2S)-2-(methoxymethyl)piperidin-1-yl]methanone
—— 6-(5-Ethyl-1,2-oxazole-3-carbonyl)-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C17H16N6O3
6-(5-Ethyl-1,2-oxazole-3-carbonyl)-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[2-(1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H21N7O2
6-ethyl-5-methyl-2-[(2R)-1-[2-(1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-amino-4-(4-butoxyphenyl)-3-phenyl-2H,4H-pyrano[2,3-c]pyrazole-5-carbonitrile —— C23H22N4O2
6-amino-4-(4-butoxyphenyl)-3-phenyl-2H,4H-pyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-ethyl-5-methyl-2-[(3S)-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O
6-ethyl-5-methyl-2-[(3S)-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
6-ethyl-2-[(3S)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
6-ethyl-2-[(3S)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(3R)-1-pyrrolidin-1-ylsulfonylpyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H25N5O3S
6-ethyl-5-methyl-2-[(3R)-1-pyrrolidin-1-ylsulfonylpyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6'-amino-1-benzyl-2-oxo-1',3'-diphenyl-1,2-dihydro-1'H-spiro[indole-3,4'-pyrano[2,3-c]pyrazole]-5'-carbonitrile —— C33H23N5O2
6'-amino-1-benzyl-2-oxo-1',3'-diphenyl-1,2-dihydro-1'H-spiro[indole-3,4'-pyrano[2,3-c]pyrazole]-5'-carbonitrile
—— 6-ethyl-2-[(3R)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H30N4O3
6-ethyl-2-[(3R)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
6-ethyl-2-[(3S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3R)-1-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H30N4O3
6-ethyl-2-[(3R)-1-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H25N5O3
6-ethyl-5-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3R)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23FN4O
6-ethyl-2-[(3R)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
6-ethyl-2-[(3R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-Amino-1-(3-chlorophenyl)-3-methyl-4-(2-nitrophenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C20H14ClN5O3
6-Amino-1-(3-chlorophenyl)-3-methyl-4-(2-nitrophenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-ethyl-2-[(3R)-1-[[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H30N4O2
6-ethyl-2-[(3R)-1-[[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-N-(2-methoxyethyl)-5-methyl-2-(5-methyl-1,2-oxazol-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine —— C16H21N5O2
6-ethyl-N-(2-methoxyethyl)-5-methyl-2-(5-methyl-1,2-oxazol-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 6-ethyl-5-methyl-2-[(3R)-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O
6-ethyl-5-methyl-2-[(3R)-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H30N4O3
6-ethyl-2-[(3S)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H30N4O2
6-ethyl-2-[(3S)-1-[[4-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H20N6O2
6-ethyl-5-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O2
6-ethyl-5-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O2
6-ethyl-5-methyl-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23FN4O
6-ethyl-2-[(3S)-1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H22N6O2
6-ethyl-5-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3R)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N4O2
6-ethyl-2-[(3R)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H20N6O2
6-ethyl-5-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(3S)-1-pyrrolidin-1-ylsulfonylpyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H25N5O3S
6-ethyl-5-methyl-2-[(3S)-1-pyrrolidin-1-ylsulfonylpyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3S)-1-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H30N4O3
6-ethyl-2-[(3S)-1-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H25N5O3
6-ethyl-5-methyl-2-[(2S)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-(5-methyl-1,2-oxazol-3-yl)-N-(2-pyrrolidin-1-ylethyl)pyrazolo[1,5-a]pyrimidin-7-amine —— C19H26N6O
6-ethyl-5-methyl-2-(5-methyl-1,2-oxazol-3-yl)-N-(2-pyrrolidin-1-ylethyl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 6-ethyl-2-[(3R)-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23FN4O
6-ethyl-2-[(3R)-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[(2S)-2-(1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H23N7O2
6-ethyl-5-methyl-2-[(2R)-1-[(2S)-2-(1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(3R)-1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23FN4O
6-ethyl-2-[(3R)-1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one